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1
المؤلفون: Jean-Yves Christophe Chiva, Peter Pyun, Andrew John Keats, Linos Lazarides, Karine G. Poullennec, Neil Andrew Dunbar, Brian E. Schultz, Mingzhe Ji, Gregory M. Watt, Karki Kapil Kumar, Ruby Cai, Carina E. Cannizzaro, Uli Schmitz, David Kenneth Dean, Yu-Jen Lee, Sangi Michael, Victoria Alexandra Steadman, Adam J. Schrier, Simon B. Pettit, Hans G. Fliri, Adrian John Highton, Todd C. Appleby, Carol Austin, Richard L. Mackman, Caroline A. Blakemore, Hui Hon Chung, Dustin Siegel, Gregory Chin, Bernard P. Murray, Hai Yang, Yang Tian, George Stepan, Jonathan Sanvoisin, Albert Liclican, Mish Michael R, David Sperandio, Rex Santos, Petr Jansa, Haolun Jin
المصدر: Journal of Medicinal Chemistry. 61:9473-9499
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Protein Conformation, Administration, Oral, Biological Availability, Hepacivirus, Isomerase, Pharmacology, Antiviral Agents, 01 natural sciences, Virus, Cell Line, Cyclophilins, Lactones, 03 medical and health sciences, Protein structure, Drug Discovery, Spiro Compounds, Enzyme Inhibitors, Cyclophilin, 010405 organic chemistry, Chemistry, Total synthesis, 0104 chemical sciences, Bioavailability, Ring size, 030104 developmental biology, Cell culture, Drug Design, Molecular Medicine
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المؤلفون: Yu-Jen Lee, Andrew John Keats, Karine G. Poullennec, Uli Schmitz, Todd C. Appleby, Hans G. Fliri, Linos Lazarides, Albert Liclican, Steven J. Stanway, David Kenneth Dean, Debi Jin, Victoria Alexandra Steadman, Simon B. Pettit, Stephanie A. Leavitt, Yang Tian, Jonathan Sanvoisin, Petr Jansa, Brian E. Schultz, Christian R. Frey, Melanie H. Wong, Gregory M. Watt, Richard L. Mackman, Carol Austin
المصدر: Journal of Medicinal Chemistry. 60:1000-1017
مصطلحات موضوعية: Spectrometry, Mass, Electrospray Ionization, Stereochemistry, Proton Magnetic Resonance Spectroscopy, Tripeptide, Crystallography, X-Ray, 010402 general chemistry, 01 natural sciences, Chemical synthesis, Stereocenter, Cyclophilins, Lactones, Structure-Activity Relationship, Residue (chemistry), chemistry.chemical_compound, Cyclophilin A, Drug Discovery, Humans, Moiety, Spiro Compounds, Cells, Cultured, Cyclophilin, Natural product, 010405 organic chemistry, Hydrogen Bonding, Surface Plasmon Resonance, 0104 chemical sciences, chemistry, Thermodynamics, Molecular Medicine, Chromatography, Liquid
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المؤلفون: Linos Lazarides, J. Y. C. Chiva, M. Jones, Victoria Alexandra Steadman
مصطلحات موضوعية: biology, Eleftheria terrae, medicine.drug_class, Antibiotics, Teixobactin, Vancomycin-Resistant Enterococci, biochemical phenomena, metabolism, and nutrition, medicine.disease_cause, biology.organism_classification, Methicillin-resistant Staphylococcus aureus, Microbiology, medicine, Antibacterial activity, Bacteria
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::f1d0143332251a48baccb2de461da9c8
https://doi.org/10.1039/9781782629870-00127 -
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المؤلفون: Victoria Weller, Poonam Shah, David N. Mallett, Mark Price, Joanne O. Hessey, Diane M. Coe, Stephen C. Hughes, Charlotte J. Hardy, Amanda Lucas, Xiao Qing Lewell, Doug Ball, Bob H. Gibbon, Stephen A. Smith, Anesh Sitaram, Linos Lazarides, Keith Biggadike, Daphne Tsitoura, Stephen A. Hermitage, Richard Stocker, Chris D. Edwards, Mahbub Ahmed, Diana Quint, Fiona Priest, Deidre Dalmas Wilk, Aimee Hillegas, Naimisha Trivedi
المصدر: Journal of medicinal chemistry. 59(5)
مصطلحات موضوعية: 0301 basic medicine, Agonist, medicine.drug_class, Pharmacology, Compound 32, 03 medical and health sciences, Structure-Activity Relationship, 0302 clinical medicine, Downregulation and upregulation, Piperidines, In vivo, Drug Discovery, medicine, Structure–activity relationship, Potency, Humans, Administration, Intranasal, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Adenine, TLR7, Asthma, 030104 developmental biology, Toll-Like Receptor 7, 030220 oncology & carcinogenesis, Molecular Medicine, Nasal administration
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المؤلفون: Zhi-Jie Ni, Qun Li, Martin John Slater, Wuxin Zou, Linos Lazarides, Yang Liu, Lois L. Wright, Paul Rowland, Liang Liao, Charles Z. Ding, Tadeusz Skarzynski, Jacob J. Plattner, Jackie E. Mordaunt, Don O. Somers, Xianfeng Li, Colin M. Edge, Yong-Kang Zhang, Gemma Victoria White, Malcolm Ellis, Jon Wright, Stephen J. Baker, Dazhong Fan, Wieslaw M. Kazmierski, Gary K. Smith, Pia Thommes, Lewis E. Pennicott, Julia A. Hubbard, Richard L. Jarvest, Bill McDowell, Yasheen Zhou, Xuelei Qian, Pamela Nassau, Richard Martin Grimes
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:3550-3556
مصطلحات موضوعية: Stereochemistry, viruses, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Peptide, Hepacivirus, Viral Nonstructural Proteins, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Catalytic Domain, Drug Discovery, Serine, medicine, Molecular Biology, chemistry.chemical_classification, Serine protease, NS3, Protease, Molecular Structure, biology, Organic Chemistry, virus diseases, Active site, Boronic Acids, digestive system diseases, Protease inhibitor (biology), chemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, medicine.drug
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المؤلفون: A. Mueller, William Millett, Anthony Nitti, Victoria Alexandra Steadman, M. Jones, Aaron J. Peoples, Linos Lazarides, Slava S. Epstein, Kim Lewis, Tanja Schneider, Amy Spoering, Fetterman Ka, Brian P. Conlon, Cintia R. Felix, Losee Lucy Ling, Chao Chen, Dallas Hughes, Ina Engels, Till F. Schäberle, Cohen Dr, Ashley Zullo
المصدر: Nature
مصطلحات موضوعية: Staphylococcus aureus, Time Factors, medicine.drug_class, Molecular Sequence Data, Antibiotics, Teixobactin, Microbial Sensitivity Tests, Peptidoglycan, Drug resistance, Biology, Article, Microbiology, Mice, chemistry.chemical_compound, Antibiotic resistance, Cell Wall, Depsipeptides, medicine, Animals, Biological Products, Teichoic acid, Multidisciplinary, Microbial Viability, Lipid II, Betaproteobacteria, Drug Resistance, Microbial, Mycobacterium tuberculosis, Staphylococcal Infections, Antimicrobial, Anti-Bacterial Agents, Teichoic Acids, Disease Models, Animal, chemistry, Multigene Family, Female
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e0215ff1462df3d8a28a49980fc10cce
https://europepmc.org/articles/PMC7414797/ -
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المؤلفون: Soraya Manaviazar, Paschalis Dimopoulos, Abil E. Aliev, Jonathan H. George, Audrey Athlan, Karl J. Hale, Marcus Walters, Linos Lazarides
المصدر: Organic Letters. 7:5369-5372
مصطلحات موضوعية: Chemistry, Organic Chemistry, Propargyl, Organic chemistry, General Medicine, Physical and Theoretical Chemistry, Biochemistry
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المؤلفون: Linos Lazarides, Karl J. Hale
المصدر: Organic Letters. 4:1903-1906
مصطلحات موضوعية: Antibiotics, Antineoplastic, Magnetic Resonance Spectroscopy, Lactams, Chemistry, Stereochemistry, Organic Chemistry, Condensation, Ring (chemistry), Peptides, Cyclic, Biochemistry, Mass Spectrometry, Anti-Bacterial Agents, Fragment (logic), Depsipeptides, Indicators and Reagents, Physical and Theoretical Chemistry, Peptides
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المؤلفون: Linos Lazarides, Karl J. Hale, J. Cai
المصدر: ChemInform. 33
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, medicine.drug_class, Stereochemistry, Yield (chemistry), Antibiotics, medicine, HATU, General Medicine, Verucopeptin
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المؤلفون: Linos Lazarides, Karl J. Hale
المصدر: ChemInform. 33
مصطلحات موضوعية: Stereochemistry, Chemistry, Fragment (computer graphics), Condensation, General Medicine, Ring (chemistry)