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1
المؤلفون: Catherine Abbadie, Raul F. Alvaro, Lin-Lin Shiao, Mark Rosenbach, Lisa F. Frey, Marc D. Chioda, Ravi P. Nargund, Richard Hajdu, Kathleen Sullivan, Robert J. DeVita, Joseph F. Leone, Kevin M. Belyk, Jenna L. Terebetski, Amanda K. Makarewicz, Elliot J. Martel, Gino Salituro, Bindhu V. Karanam, Raman K. Bakshi, James Dellureficio, Selena Fung, Ping Liu, Linda Chang, Nina Jochnowitz, Shruti Mistry, Joyce Shuman, Linus S. Lin, Yan Guo, Maria Madeira, Shane W. Krska, Mark McLaughlin, Erin McGowan, Harry R. Chobanian, Jessica Alexander, Matthew J. Wyvratt, Qingmei Hong, Thomas J. Lanza
المصدر: ACS Medicinal Chemistry Letters. 5:717-721
مصطلحات موضوعية: business.industry, Organic Chemistry, Pharmacology, Biochemistry, In vitro, chemistry.chemical_compound, Pharmacokinetics, chemistry, In vivo, Fatty acid amide hydrolase, Drug Discovery, Neuropathic pain, Medicine, Potency, lipids (amino acids, peptides, and proteins), business, MK-4409, Oxazole
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2
المؤلفون: Luis Sojo, Alla Yurevna Zenova, Margaret van Heek, David Percival, Andrea Lindgren, Linus S. Lin, Michael Winther, Shaoyi Sun, Pritpaul Samra, Celene Grayson, Jianmin Fu, Qi Jia, Jing Zhong, Richard A. Dean, Zaihui Zhang, Clark Xie
المصدر: Bioorganic & Medicinal Chemistry. 21:7724-7734
مصطلحات موضوعية: Male, Endothelial lipase, Pyrrolidines, Clinical Biochemistry, Pharmaceutical Science, Hdl metabolism, Pharmacology, Benzoates, Biochemistry, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, Anthranilic acid, medicine, Animals, Enzyme Inhibitors, Molecular Biology, ADME, Mice, Knockout, Dose-Response Relationship, Drug, Molecular Structure, Cholesterol, Cholesterol, HDL, Organic Chemistry, Lipase, medicine.disease, Mice, Inbred C57BL, chemistry, Molecular Medicine, Dyslipidemia
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3
المؤلفون: Richard Hargreaves, Maria Madeira, Patricia Miller, Joyce Powell, Richard Hajdu, Selena Fung, Lin-Lin Shiao, Mark Rosenbach, Ping Liu, Zhizhen Zeng, Qingmei Hong, Catherine Abbadie, Tsing-Bau Chen, Aniket Joshi, Wenping Li, Suzanne M. Mandala, Diane Posavec, Jacquelynn J. Cook, Bindhu V. Karanam, Ling Xu, Jenna L. Terebetski, Marc D. Chioda, Kerry Riffel, Nina Jochnowitz, Robert J. DeVita, Joseph F. Leone, David L. Williams, Mangay Williams, Ravi P. Nargund, Stacey O'Malley, Marie A. Holahan, Linus S. Lin, Sandra Sanabria, Raman K. Bakshi, Mona Purcell, Kathleen A. Sullivan, Yan Guo, Terence G. Hamill, James Dellureficio, Linda Chang, Harry R. Chobanian, Jessica Alexander, Gino Salituro, Hong Jin
المصدر: ACS Medicinal Chemistry Letters. 4:509-513
مصطلحات موضوعية: medicine.diagnostic_test, Organic Chemistry, Pyrazole, Imaging brain, Biochemistry, chemistry.chemical_compound, nervous system, chemistry, Fatty acid amide hydrolase, Positron emission tomography, Physical chemical, Drug Discovery, Lipophilicity, medicine, Imidazole, lipids (amino acids, peptides, and proteins), Pet tracer, psychological phenomena and processes
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المؤلفون: Linda Chang, Yanqing Kan, Alison M. Strack, Yan Guo, Judith N. Gorski, Linus S. Lin, Maria Madeira, Oksana C. Palyha, Thomas J. Lanza, Randy R. Miller, Jasminka Dragovic, Theresa M. Kelly, Ping Liu, Marc L. Reitman, Ravi P. Nargund, Joseph M. Metzger, Harry R. Chobanian, Donald J. Marsh, Kathy Lyons, Jianmei Pang, Kate A. Raustad, Marc D. Chioda, Xiao-Ming Guan, Sheng-Ping Wang
المصدر: ACS Medicinal Chemistry Letters. 3:252-256
مصطلحات موضوعية: Agonist, Benzodiazepine, Atropisomer, medicine.drug_class, business.industry, Organic Chemistry, Pharmacology, Biochemistry, chemistry.chemical_compound, chemistry, Pharmacokinetics, Pharmacodynamics, Drug Discovery, medicine, Bombesin Receptor Subtype-3, Penetrant (biochemical), business
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المؤلفون: Oksana C. Palyha, Terry D. Faidley, Joseph M. Metzger, Xiao-Ming Guan, Sheng-Ping Wang, Jennifer A. Kosinski, Ravi P. Nargund, Stephanie K. Spann, Marc L. Reitman, Liming Yang, Linus S. Lin, Lauren P. Shearman, Kate A. Raustad, Donald J. Marsh, Kathy Lyons, Theresa M. Kelly, Stephanie Craw, Alison M. Strack, Yanqing Kan, Hong Yu, Jasminka Dragovic, Iyassu K. Sebhat
المصدر: Journal of Pharmacology and Experimental Therapeutics. 336:356-364
مصطلحات موضوعية: Male, Agonist, medicine.medical_specialty, medicine.drug_class, Blood Pressure, Pharmacology, Energy homeostasis, Rats, Sprague-Dawley, Eating, Mice, Dogs, Heart Rate, Weight loss, Internal medicine, medicine, Animals, Receptor, Dose-Response Relationship, Drug, Chemistry, Body Weight, Imidazoles, Rats, Bombesin receptor, Mice, Inbred C57BL, Receptors, Bombesin, Dose–response relationship, Blood pressure, Endocrinology, Pyrazoles, Molecular Medicine, Bombesin Receptor Subtype-3, Anti-Obesity Agents, medicine.symptom, Energy Metabolism
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4f83aba6c5ca83619726b27f1351081f
https://doi.org/10.1124/jpet.110.174763 -
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المؤلفون: Laurie G. Castonguay, Sookhee Ha, Lex H.T. Van der Ploeg, Chun-Pyn Shen, Ihor E. Kopka, Zhege J. Lao, Mark T. Goulet, Linus S. Lin, William K. Hagmann, Tung M. Fong, James P. Jewell, Thomas J. Lanza
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:4757-4761
مصطلحات موضوعية: Models, Molecular, Molecular model, Pyridines, medicine.drug_class, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Carboxamide, Context (language use), Biochemistry, Chemical synthesis, Taranabant, Receptor, Cannabinoid, CB1, Drug Discovery, medicine, Humans, Inverse agonist, Computer Simulation, Homology modeling, Molecular Biology, Chemistry, Organic Chemistry, Amides, Molecular Medicine, Anti-Obesity Agents, Cannabinoid, Protein Binding, medicine.drug
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المؤلفون: Nathan X. Yu, Thomas J. Lanza, Koppara Samuel, Sanjeev Kumar, George A. Doss, Vijay Bhasker G. Reddy, Ralph A. Stearns, Bindhu V. Karanam, Linus S. Lin, Conrad E. Raab, Andy Shiqiang Zhang
المصدر: Xenobiotica. 40:650-662
مصطلحات موضوعية: Male, Magnetic Resonance Spectroscopy, Drug Inverse Agonism, Pyridines, Stereochemistry, Health, Toxicology and Mutagenesis, Metabolite, Pharmacology, Toxicology, Biochemistry, Mass Spectrometry, Hydroxylation, chemistry.chemical_compound, Taranabant, Receptor, Cannabinoid, CB1, medicine, Animals, Humans, Inverse agonist, Receptor, Antibodies, Monoclonal, Brain, Haplorhini, General Medicine, Glutathione, Metabolism, Amides, Propanamide, Body Fluids, Rats, Ketoconazole, Radioactivity, chemistry, Microsomes, Liver, Female, medicine.drug
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المؤلفون: Marc L. Reitman, Cheng Guo, Theresa M. Kelly, Constantin Tamvakopoulos, Joseph M. Metzger, Tianying Jian, Howard Y. Chen, Arthur A. Patchett, Oksana C. Palyha, Alison M. Strack, Allan J. Goodman, Ravi P. Nargund, Peter H. Dobbelaar, Yanqing Kan, Mark Hadden, Larry Yet, Peter R. Guzzo, Qianping Peng, Linus S. Lin, Shuwen He, Lauren P. Shearman, Alan J. Henderson, Carina P. Tan, Sargent Bruce J, Xiao-Ming Guan, Scott D. Feighner, Iyassu K. Sebhat, Jie Pan, Jian Liu, Donald J. Marsh, Matthew J. Wyvratt, Andrew D. Howard, Megan Ruenz
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1913-1917
مصطلحات موضوعية: Agonist, medicine.drug_class, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Potency, Structure–activity relationship, Molecular Biology, Biphenyl, Chemistry, Drug discovery, fungi, Organic Chemistry, Imidazoles, Rats, Bombesin receptor, Bioavailability, Receptors, Bombesin, Molecular Medicine, Bombesin Receptor Subtype-3
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المؤلفون: Gerard R. Kieczykowski, Carrie P. Jones, Ping Liu, Junying Wang, Conrad E. Raab, Qian Si, Xinchun Tong, Thomas J. Lanza, Anne Schuelke, Kelly M. Treonze, Richard A. Mumford, Salony Manior, Stella H. Vincent, James V. Pivnichny, Gloria C. Koo, James P. Jewell, William K. Hagmann, Regina W. Wang, Philip Davies, Linus S. Lin, Malcolm MacCoss
المصدر: Journal of Medicinal Chemistry. 52:3449-3452
مصطلحات موضوعية: chemistry.chemical_classification, Sulfonyl, Dipeptide, Stereochemistry, medicine.drug_class, Antagonist, Peptide, Phenylalanine, Carboxamide, Biological activity, chemistry.chemical_compound, chemistry, Drug Discovery, medicine, Molecular Medicine, Proline
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المؤلفون: Terence G. Hamill, Brett Connolly, Ping Liu, Tung M. Fong, Christine Ryan, Richard Hargreaves, Linus S. Lin, Mark T. Goulet, Amy Vanko, Wai-Si Eng, William K. Hagmann, James P. Jewell, H. Donald Burns, Sandra Sanabria
المصدر: Molecular Imaging and Biology. 11:246-252
مصطلحات موضوعية: Cancer Research, Cannabinoid receptor, Pyridines, medicine.medical_treatment, Ligands, Tritium, Receptor, Cannabinoid, CB1, In vivo, medicine, Animals, Inverse agonist, Tissue Distribution, Radiology, Nuclear Medicine and imaging, Carbon Radioisotopes, IC50, Chemistry, business.industry, Brain, Pet imaging, Ligand (biochemistry), Amides, Macaca mulatta, In vitro, Oncology, Positron-Emission Tomography, Biophysics, Autoradiography, Cannabinoid, Radiopharmaceuticals, Nuclear medicine, business, Protein Binding