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المؤلفون: Bruce A. Ruggeri, Giorgio Inghirami, Bruce D. Dorsey, Mark A. Ator, Cristina Abele, Rodolfo Machiorlatti, Flavio Cristofani, Lisa D. Aimone, Thelma S. Angeles, Mark S. Albom, Weihua Wan, Lihui Lu, Gregory R. Ott, Diane E. Gingrich, Matthew R. Quail, Mangeng Cheng
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b6a0a50e0c286d90b24603959f90aa4c
https://doi.org/10.1158/1535-7163.22498291 -
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المؤلفون: Bruce A. Ruggeri, Giorgio Inghirami, Bruce D. Dorsey, Mark A. Ator, Cristina Abele, Rodolfo Machiorlatti, Flavio Cristofani, Lisa D. Aimone, Thelma S. Angeles, Mark S. Albom, Weihua Wan, Lihui Lu, Gregory R. Ott, Diane E. Gingrich, Matthew R. Quail, Mangeng Cheng
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::36ff3acce277a3f9ee6d65f11bbc8c38
https://doi.org/10.1158/1535-7163.22498288 -
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المؤلفون: Robert L. Hudkins, Joanne R. Mathiasen, Rita Raddatz, Edward R. Bacon, Michael J. Marino, Mark A. Ator, Michael Williams, Lisa D. Aimone, John A. Gruner
المصدر: Neuropharmacology. 106:37-45
مصطلحات موضوعية: Male, 0301 basic medicine, medicine.medical_specialty, Drug Inverse Agonism, Drinking, Drug Evaluation, Preclinical, Administration, Oral, Biological Availability, Motor Activity, Pharmacology, Histamine agonist, Histamine Agonists, Rats, Sprague-Dawley, 03 medical and health sciences, Cellular and Molecular Neuroscience, Histamine receptor, chemistry.chemical_compound, Dogs, 0302 clinical medicine, Therapeutic index, Piperidines, Internal medicine, medicine, Animals, Humans, Receptors, Histamine H3, Inverse agonist, Spiro Compounds, Wakefulness, Chemistry, Methylhistamines, Antagonist, Brain, Macaca fascicularis, 030104 developmental biology, Endocrinology, Pyrazines, Histamine H3 receptor, Sleep, 030217 neurology & neurosurgery, Histamine, Histamine H3 Antagonists
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المؤلفون: Nadine C. Becknell, Joanne R. Mathiasen, Jacquelyn A. Lyons, John A. Gruner, Robert L. Hudkins, Mark A. Olsen, Lisa D. Aimone, Rita Raddatz, R. Curtis Haltiwanger
المصدر: European Journal of Medicinal Chemistry. 95:349-356
مصطلحات موضوعية: Pyrrolidines, Drug Inverse Agonism, Stereochemistry, Histamine Antagonists, Structure-Activity Relationship, chemistry.chemical_compound, Irdabisant, Drug Discovery, Animals, Humans, Receptors, Histamine H3, Inverse agonist, Wakefulness, Receptor, Pharmacology, Dose-Response Relationship, Drug, Bicyclic molecule, Organic Chemistry, Diastereomer, Stereoisomerism, General Medicine, Combinatorial chemistry, Rats, Functional antagonism, Pyridazines, chemistry, Drug Design, Selectivity, Histamine
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المؤلفون: R. Curtis Haltiwanger, Mark A. Olsen, Mark A. Ator, Emily Kordwitz, Gregory R. Ott, Jason C. Wagner, Bruce D. Dorsey, Zeqi Huang, Mangeng Cheng, Bruce Ruggeri, Eugen F. Mesaros, Weihua Wan, Lihui Lu, Amy J. Landis, Lisa D. Aimone, Mark S. Albom, Thelma S. Angeles
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:1047-1052
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Clinical Biochemistry, Diol, Pharmaceutical Science, Antineoplastic Agents, Mice, SCID, Crystallography, X-Ray, Biochemistry, Rats, Sprague-Dawley, chemistry.chemical_compound, Piperidines, In vivo, Cell Line, Tumor, hemic and lymphatic diseases, Drug Discovery, Animals, Humans, Anaplastic lymphoma kinase, Anaplastic Lymphoma Kinase, Pyrroles, Protein Kinase Inhibitors, Molecular Biology, Triazine, Triazines, Kinase, Organic Chemistry, Autophosphorylation, Receptor Protein-Tyrosine Kinases, Biological activity, chemistry, Lymphoma, Large-Cell, Anaplastic, Molecular Medicine, Piperidine
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المؤلفون: Sankar Chatterjee, John A. Gruner, Yin G. Lin, Brigitte Lesur, Lisa D. Aimone, Edward R. Bacon, Val R. Marcy
المصدر: Chemical Biology & Drug Design. 81:429-432
مصطلحات موضوعية: Pharmacology, Stereochemistry, Aryl, Organic Chemistry, Modafinil, Biochemistry, chemistry.chemical_compound, Wakefulness-Promoting Agents, chemistry, Drug Discovery, medicine, Molecular Medicine, psychological phenomena and processes, medicine.drug
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المؤلفون: Nathan Anderson, Diane E. Gingrich, Arup K. Ghose, Mark S. Albom, Bruce D. Dorsey, Lisa D. Aimone, Elizabeth Bruckheimer, Jason C. Wagner, Matthew A. Curry, Lihui Lu, Jay Friedman, Mark A. Ator, Bruce Ruggeri, Eugen F. Mesaros, Mangeng Cheng, Zeqi Huang, Keith S. Learn, Matthew R. Quail, Thelma S. Angeles, Pawel Dobrzanski, Gregory R. Ott, Sandra V. Fernandez, Joseph G. Lisko, Kevin J. Wells-Knecht, Weihua Wan
المصدر: Journal of medicinal chemistry. 59(16)
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, medicine.drug_class, Administration, Oral, Mice, Nude, Mice, SCID, Metastasis, Focal adhesion, 03 medical and health sciences, Mice, Structure-Activity Relationship, 0302 clinical medicine, In vivo, hemic and lymphatic diseases, Cell Line, Tumor, Drug Discovery, medicine, Anaplastic lymphoma kinase, Animals, Humans, Anaplastic Lymphoma Kinase, Protein Kinase Inhibitors, Cell Proliferation, Dose-Response Relationship, Drug, Molecular Structure, Cell growth, Chemistry, Drug discovery, Receptor Protein-Tyrosine Kinases, Neoplasms, Experimental, medicine.disease, In vitro, ALK inhibitor, Benzocycloheptenes, 030104 developmental biology, Biochemistry, 030220 oncology & carcinogenesis, Focal Adhesion Kinase 1, Benzamides, Cancer research, Molecular Medicine, Female, Drug Screening Assays, Antitumor
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المصدر: Bioorganic & Medicinal Chemistry Letters. 22:4198-4202
مصطلحات موضوعية: Pyrrolidines, Drug Inverse Agonism, Stereochemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, CHO Cells, Biochemistry, Histamine Agonists, Structure-Activity Relationship, chemistry.chemical_compound, Irdabisant, Cricetinae, Drug Discovery, Animals, Receptors, Histamine H3, Inverse agonist, Potency, Molecular Biology, Nootropic Agents, Dose-Response Relationship, Drug, Molecular Structure, biology, Cell Membrane, Organic Chemistry, Combinatorial chemistry, Rats, Pyridazines, chemistry, biology.protein, Molecular Medicine, Histamine H3 receptor, Selectivity, Heterocyclic Compounds, 3-Ring, Linker, Histamine, Histamine H3 Antagonists
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المؤلفون: Robert L. Hudkins, Allison L. Zulli, Rita Raddatz, Lisa D. Aimone, John A. Gruner, Edward R. Bacon, Joanne R. Mathiasen
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:2807-2810
مصطلحات موضوعية: Pyrrolidines, Ketone, Drug Inverse Agonism, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, 1-Propanol, Biochemistry, Histamine Agonists, Methylamines, chemistry.chemical_compound, Phenols, Pharmacokinetics, Sleep Disorders, Circadian Rhythm, In vivo, Diamine, Drug Discovery, Animals, Humans, Inverse agonist, Molecule, Wakefulness, Receptor, Molecular Biology, chemistry.chemical_classification, Organic Chemistry, Ketones, Rats, chemistry, Molecular Medicine, Histamine
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المؤلفون: Thomas J. Connors, Jie Qian, Zeck Huang, Joanne R. Mathiasen, Edward R. Bacon, Thelma S. Angeles, Mark J. Huffman, Emir Duzic, Joseph M. Salvino, Beth Ann McKenna, Hervé Schaffhauser, Robert J. McHugh, Lily D. Lu, George C. Morton, Beverly P. Holskin, Karla Kopec, Amy DiCamillo, Gerard C. Rosse, Chrysanthe Spais, Rabindranath Tripathy, Lisa D. Aimone
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:1421-1426
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Stereoisomerism, Biochemistry, Sulfone, chemistry.chemical_compound, In vivo, Drug Discovery, 5-HT6 receptor, Molecular Medicine, Pharmacophore, Receptor, Molecular Biology, 5-HT receptor