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المؤلفون: Jannik N. Andersen, Shikhar Sharma, Wylie S. Palmer, Philip Jones, Giulio Draetta, Dafydd R. Owen, Dominique Verhelle, Alessia Petrocchi, Carlo Toniatti, Joseph R. Marszalek, Timothy P. Heffernan, Mike Peoples, Trang N. Tieu, Andrew Futreal, Alexei Protopopov, Harshad S. Mahadeshwar, Elisabetta Leo, Yanai Zhan, Xi Shi, Lisa Nottebaum, Maria Kost-Alimova, Parantu K. Shah, Thomas A. Paul, Bhavatarini Vangamudi
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0ccf7d378c7bc490374b9266a8d53305
https://doi.org/10.1158/0008-5472.22407462.v1 -
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المؤلفون: Jannik N. Andersen, Shikhar Sharma, Wylie S. Palmer, Philip Jones, Giulio Draetta, Dafydd R. Owen, Dominique Verhelle, Alessia Petrocchi, Carlo Toniatti, Joseph R. Marszalek, Timothy P. Heffernan, Mike Peoples, Trang N. Tieu, Andrew Futreal, Alexei Protopopov, Harshad S. Mahadeshwar, Elisabetta Leo, Yanai Zhan, Xi Shi, Lisa Nottebaum, Maria Kost-Alimova, Parantu K. Shah, Thomas A. Paul, Bhavatarini Vangamudi
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0badb0679a64bcc92e6b33f08070943f
https://doi.org/10.1158/0008-5472.22407459 -
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المؤلفون: Anthony R. Harris, Susan M. Lotarski, Michael Aaron Brodney, Michael Popiolek, Catherine A. Thorn, Stephen Jenkinson, Che Wah Lee, Jennifer E. Davoren, Stefanus J. Steyn, Lei Zhang, Terrence Peter Kenakin, Betty Pettersen, Sarah Grimwood, Damien Webb, Michelle R. Garnsey, Simeon Ramsey, John T. Lazzaro, Steven Victor O'neil, Lisa Nottebaum, Jean-Philippe Fortin, Jeremy R. Edgerton
المصدر: Journal of Medicinal Chemistry. 60:6649-6663
مصطلحات موضوعية: 0301 basic medicine, Agonist, Allosteric modulator, medicine.drug_class, Chemistry, Allosteric regulation, Muscarinic acetylcholine receptor M1, Pharmacology, 03 medical and health sciences, 030104 developmental biology, Drug Discovery, Convulsion, medicine, Molecular Medicine, Cholinergic, Structure–activity relationship, medicine.symptom, Receptor
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المؤلفون: Asser Bassyouni, Stephen Jenkinson, John T. Lazzaro, Lisa Nottebaum, Betty Pettersen, Jennifer Elizabeth Davoren
المصدر: Journal of Pharmacological and Toxicological Methods. 99:106595
مصطلحات موضوعية: Pharmacology, business.industry, Medicine, Motility, M1 muscarinic receptor, Toxicology, business
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المؤلفون: Jennifer E, Davoren, Michelle, Garnsey, Betty, Pettersen, Michael A, Brodney, Jeremy R, Edgerton, Jean-Philippe, Fortin, Sarah, Grimwood, Anthony R, Harris, Stephen, Jenkinson, Terry, Kenakin, John T, Lazzaro, Che-Wah, Lee, Susan M, Lotarski, Lisa, Nottebaum, Steven V, O'Neil, Michael, Popiolek, Simeon, Ramsey, Stefanus J, Steyn, Catherine A, Thorn, Lei, Zhang, Damien, Webb
المصدر: Journal of medicinal chemistry. 60(15)
مصطلحات موضوعية: Diarrhea, Male, Lactams, Vomiting, Scopolamine, Isoindoles, Structure-Activity Relationship, Dogs, Allosteric Regulation, Piperidines, Seizures, Thiadiazoles, Animals, Humans, Donepezil, Rats, Wistar, Oxazoles, Sulfonamides, Receptor, Muscarinic M1, Mice, Inbred C57BL, Amphetamine, Drug Design, Indans, Microsomes, Liver, Ataxia, Female
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المؤلفون: Deane M. Nason, Keith Dlugolenski, Chewah Lee, Betty Pettersen, Gregory W. Kauffman, Lei Zhang, Carrie Northcott, Stephen Jenkinson, Yuxia Mao, Jennifer E. Davoren, Susan M. Lotarski, Veronica Reinhart, Damien Webb, Michelle R. Garnsey, Sarah Grimwood, John T. Lazzaro, Michael Aaron Brodney, Jeremy R. Edgerton, Jason Cordes, Stefanus J. Steyn, Romelia Salomon-Ferrer, Steven Victor O'neil, Terrence Peter Kenakin, Lisa Nottebaum, Michael Popiolek, Christopher John Helal, Anthony R. Harris
المصدر: Journal of medicinal chemistry. 59(13)
مصطلحات موضوعية: 0301 basic medicine, Agonist, Male, Models, Molecular, Allosteric modulator, Stereochemistry, medicine.drug_class, Carboxamide, Pharmacology, 03 medical and health sciences, chemistry.chemical_compound, Mice, Structure-Activity Relationship, 0302 clinical medicine, Muscarinic acetylcholine receptor, Drug Discovery, medicine, Structure–activity relationship, Animals, Picolinic Acids, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Receptor, Muscarinic M1, Rats, Thiazoles, 030104 developmental biology, Pyran, Molecular Medicine, Cholinergic, Female, Pharmacophore, 030217 neurology & neurosurgery
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المؤلفون: Xi Shi, Alessia Petrocchi, Shikhar Sharma, Lisa Nottebaum, Jannik N. Andersen, Elisabetta Leo, Maria Kost-Alimova, Timothy P. Heffernan, Philip Jones, Bhavatarini Vangamudi, Trang N. Tieu, Dominique Verhelle, Harshad S. Mahadeshwar, Parantu K. Shah, Dafydd R. Owen, Andrew Futreal, Mike Peoples, Giulio Draetta, Thomas A Paul, Yanai Zhan, Wylie S. Palmer, Joseph R. Marszalek, Carlo Toniatti, Alexei Protopopov
المصدر: Cancer research. 75(18)
مصطلحات موضوعية: Cancer Research, DNA, Complementary, Lung Neoplasms, Chromosomal Proteins, Non-Histone, Pyridines, Protein domain, Biology, Binding, Competitive, Catalysis, Article, Gene Knockout Techniques, Sarcoma, Synovial, RNA interference, Cell Line, Tumor, Neoplasms, Humans, Molecular Targeted Therapy, RNA, Small Interfering, Rhabdoid Tumor, Gene knockdown, Genetic Complementation Test, DNA Helicases, Nuclear Proteins, Chromatin Assembly and Disassembly, Microarray Analysis, SWI/SNF, Chromatin, Bromodomain, Neoplasm Proteins, Protein Structure, Tertiary, Oncology, SMARCA4, Cancer research, RNA Interference, Chromatin immunoprecipitation, Azabicyclo Compounds, Transcription Factors
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b46a37cc723ee28ec2ca78b006ca9829
https://pubmed.ncbi.nlm.nih.gov/26139243 -
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المؤلفون: Wylie S. Palmer, Trang N. Tieu, Giulio Draetta, Maria Alimova, Thomas A Paul, Alessia Petrocchi, Jannik N. Andersen, Elisabetta Leo, Bhavatarini Vangamudi, Alexei Protopopov, Mike Peoples, Dafydd R. Owen, Philip Jones, Xi Shi, Timothy P. Heffernan, Shikhar Sharma, Carlo Toniatti, Joseph R. Marszalek, Yanai Zhan, Dominique Verhelle, Lisa Nottebaum, Parantu K. Shah, Harshad S. Mahadeshwar, Andrew Futreal
المصدر: Cancer Research. 75:3528-3528
مصطلحات موضوعية: Cancer Research, Oncology, RNA interference, Cancer cell, Mutant, Cancer research, SMARCA4, Biology, Molecular biology, Chromatin immunoprecipitation, SWI/SNF, Bromodomain, Chromatin
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::95798e37ef386b6f751cd65c78be3853
https://doi.org/10.1158/1538-7445.am2015-3528 -
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المؤلفون: Aileen McHarg, Qing Zong, Lisa Nottebaum, Michelle Hemkens, Julie V. Selkirk, Jonathan R. Heyen
المصدر: Journal of Pharmacological and Toxicological Methods. 64:e31-e32
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, Aldosterone, business.industry, Toxicology, medicine.disease, chemistry.chemical_compound, Endocrinology, chemistry, Internal medicine, Medicine, Endothelial dysfunction, business, Ex vivo
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المصدر: Journal of Pharmacological and Toxicological Methods. 68:e27
مصطلحات موضوعية: Pharmacology, Aorta, business.industry, medicine.artery, medicine, Anatomy, medicine.symptom, Toxicology, business, Vasoconstriction, Nonhuman primate, In vitro model