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1Impact of Cancer-Associated Mutations in CC Chemokine Receptor 2 on Receptor Function and Antagonism
المؤلفون: Lisa S. den Hollander, Olivier J.M. Béquignon, Xuesong Wang, Kim van Wezel, Jeremy Broekhuis, Marina Gorostiola González, Karin E. de Visser, Adriaan P. IJzerman, Gerard J. P. van Westen, Laura H. Heitman
المصدر: SSRN Electronic Journal.
مصطلحات موضوعية: History, Polymers and Plastics, Business and International Management, Industrial and Manufacturing Engineering
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::03a9a2c7d27bd4a57b7a799147a7505e
https://doi.org/10.2139/ssrn.4250690 -
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المؤلفون: Joseph Openy, Adriaan P. IJzerman, Burak Dogan, Ya-Yun Hsiao, Eelke B. Lenselink, Jacobus P. D. van Veldhoven, Natalia V. Ortiz Zacarías, Laura H. Heitman, Lisa S den Hollander
المصدر: Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, 62(24), 11035-11053مصطلحات موضوعية: CCR2, Receptors, CCR5, Receptors, CCR2, animal diseases, Antineoplastic Agents, Bone Neoplasms, Pharmacology, Ligands, 01 natural sciences, Article, Radioligand Assay, Structure-Activity Relationship, 03 medical and health sciences, Chemokine receptor, parasitic diseases, Drug Discovery, Tumor Cells, Cultured, Humans, Structure–activity relationship, Binding site, Receptor, Cell Proliferation, 030304 developmental biology, Osteosarcoma, 0303 health sciences, Binding Sites, Molecular Structure, Chemistry, hemic and immune systems, Biological activity, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Purines, Molecular Medicine, Intracellular, Protein Binding