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1
المؤلفون: Christopher L. Carpenter, Eldridge N. Nartey, Dominic Suarez, Elisabeth A. Minthorn, Jesus R. Medina, Louis V. LaFrance, Ralph A. Rivero, James F. Mack, Charles F. McHugh, Xinrong Tian, Dirk A. Heerding, Christina Ng Di Marco, Thomas J. Berrodin, Aishwarya Bhaskar, Biju Mangatt, William Hoi Hong Li, Brackley James, Martyr Cuthbert, Lorena A. Kallal, Michael Butticello, Jacob Rubin
المصدر: Journal of Medicinal Chemistry. 64:16056-16087
مصطلحات موضوعية: Gene knockdown, Oncogene, Drug discovery, Chemistry, Drug Discovery, Molecular Medicine, Structure–activity relationship, Computational biology, Small molecule binding, Pharmacophore, Small molecule, Function (biology)
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2
المؤلفون: Jesús R, Medina, Xinrong, Tian, William H, Li, Dominic, Suarez, James F, Mack, Louis, LaFrance, Cuthbert, Martyr, James, Brackley, Christina, Di Marco, Ralph, Rivero, Dirk A, Heerding, Charles, McHugh, Elisabeth, Minthorn, Aishwarya, Bhaskar, Jacob, Rubin, Michael, Butticello, Christopher, Carpenter, Eldridge N, Nartey, Thomas J, Berrodin, Lorena A, Kallal, Biju, Mangatt
المصدر: Journal of medicinal chemistry. 64(21)
مصطلحات موضوعية: Proto-Oncogene Proteins c-myc, Small Molecule Libraries, Structure-Activity Relationship, Area Under Curve, Cell Line, Tumor, Drug Discovery, Animals, Humans, Xenograft Model Antitumor Assays, Half-Life, Rats
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3
المؤلفون: Widdowson Katherine L, Lorena A. Kallal, Yvett Sosa, Matthew S. Steiginga, Michael T. Ouellette, Myles H. Akabas, I. J. Frame, Andrew J. Pope, Roman Deniskin, Todd L. Graybill, Deepak Bandyopadhyay, Robert J. Young
المصدر: ACS Infectious Diseases. 5:1738-1753
مصطلحات موضوعية: 0301 basic medicine, Purine, Drug, Drug discovery, media_common.quotation_subject, Auxotrophy, 030106 microbiology, Equilibrative nucleoside transporter, Plasmodium falciparum, Biology, biology.organism_classification, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, Infectious Diseases, chemistry, Biochemistry, Drug development, Purine metabolism, media_common
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4دورية أكاديمية
المؤلفون: David J Rickard, Clark A Sehon, Viera Kasparcova, Lorena A Kallal, Pamela A Haile, Xin Zeng, Monica N Montoute, Derek D Poore, Hu Li, Zining Wu, Patrick M Eidam, John G Emery, Robert W Marquis, Peter J Gough, John Bertin
المصدر: PLoS ONE, Vol 9, Iss 5, p e96737 (2014)
وصف الملف: electronic resource
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5High-Throughput Screening and Triage Assays Identify Small Molecules Targeting c-MYC in Cancer Cells
المؤلفون: Jon-Paul Jaworski, Lisa A. Payne, Anna Waszkiewicz, Biju Mangatt, Anthony J. Jurewicz, Lorena A. Kallal, Jesus R. Medina, Pat Brady, Xin Zeng, Thomas J. Berrodin, Carolyn Doepner-Buser, Anthony Della Pietra
المصدر: SLAS discovery : advancing life sciences RD. 26(2)
مصطلحات موضوعية: 0301 basic medicine, High-throughput screening, Genes, myc, Biochemistry, Analytical Chemistry, Flow cytometry, Small Molecule Libraries, 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, medicine, Fluorescence Resonance Energy Transfer, Humans, Transcription factor, Reporter gene, medicine.diagnostic_test, Cell growth, Chemistry, Reverse Transcriptase Polymerase Chain Reaction, Cell cycle, Gene signature, Flow Cytometry, Molecular biology, High-Throughput Screening Assays, Gene Expression Regulation, Neoplastic, 030104 developmental biology, 030220 oncology & carcinogenesis, Cancer cell, Molecular Medicine, Drug Screening Assays, Antitumor, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0dbee602aec0943dd6af57df9d435d52
https://pubmed.ncbi.nlm.nih.gov/33482073 -
6دورية أكاديمية
المؤلفون: David J Rickard, Clark A Sehon, Viera Kasparcova, Lorena A Kallal, Xin Zeng, Monica N Montoute, Tushar Chordia, Derek D Poore, Hu Li, Zining Wu, Patrick M Eidam, Pamela A Haile, Jong Yu, John G Emery, Robert W Marquis, Peter J Gough, John Bertin
المصدر: PLoS ONE, Vol 8, Iss 8, p e69619 (2013)
وصف الملف: electronic resource
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7
المؤلفون: Anton Simeonov, Lorena A. Kallal, Marc A. Holbert, Mark J. Henderson
المصدر: SLAS discovery : advancing life sciences RD. 25(2)
مصطلحات موضوعية: 0301 basic medicine, Biomedical Research, Computer science, Drug discovery, Target engagement, Context (language use), Computational biology, Biochemical Activity, Ligands, 01 natural sciences, Biochemistry, 0104 chemical sciences, Analytical Chemistry, High-Throughput Screening Assays, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, Microtiter plate, 030104 developmental biology, Protein structure, Drug Discovery, Molecular Medicine, Humans, Protein target, Throughput (business), Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e74cfb093214f5a721178267cf4505b9
https://pubmed.ncbi.nlm.nih.gov/31566060 -
8
المؤلفون: Yvett, Sosa, Roman, Deniskin, I J, Frame, Matthew S, Steiginga, Deepak, Bandyopadhyay, Todd L, Graybill, Lorena A, Kallal, Michael T, Ouellette, Andrew J, Pope, Katherine L, Widdowson, Robert J, Young, Myles H, Akabas
المصدر: ACS Infect Dis
مصطلحات موضوعية: Erythrocytes, Plasmodium falciparum, Protozoan Proteins, Biological Transport, Hep G2 Cells, Article, High-Throughput Screening Assays, Malaria, Antimalarials, Gene Knockout Techniques, Purines, Yeasts, Drug Discovery, Humans, Malaria, Falciparum, Transcriptome, Nucleobase, Nucleoside, Nucleotide, and Nucleic Acid Transport Proteins, Cell Proliferation
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9
المؤلفون: Elizabeth Nixon, Lorena A. Kallal, Michael Weglos, Snehal Bhatt, Maggie Truong, Jeffrey W. Gross, Sue Crimmin
المصدر: SLAS technology. 24(3)
مصطلحات موضوعية: Sample handling, 0303 health sciences, Emerging technologies, Drug discovery, Science and engineering, Stem Cells, Cytological Techniques, Drug Evaluation, Preclinical, 02 engineering and technology, Microfluidic Analytical Techniques, 021001 nanoscience & nanotechnology, Data science, Computer Science Applications, High-Throughput Screening Assays, 03 medical and health sciences, Medical Laboratory Technology, Drug Discovery, Humans, 0210 nano-technology, Cells, Cultured, 030304 developmental biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a6e435326763cd8daf3e6f65cad3a35c
https://pubmed.ncbi.nlm.nih.gov/30726680 -
10
المؤلفون: Quinn Lu, Tiger W. Bee, Pankaj K. Agarwal, Dwight M. Morrow, Xin Zeng, Zining Wu, Monica N. Montoute, Hong Lin, Andrew J. Pope, Yan Liu, Da-Yuan Wang, Lorena A. Kallal
المصدر: SLAS Discovery. 21:260-268
مصطلحات موضوعية: 0301 basic medicine, Beta-catenin, Multiprotein complex, Adenomatous polyposis coli, Cell, Antineoplastic Agents, Biochemistry, Analytical Chemistry, Small Molecule Libraries, Inhibitory Concentration 50, 03 medical and health sciences, Antibody Specificity, Cell Line, Tumor, medicine, Humans, Wnt Signaling Pathway, beta Catenin, Dose-Response Relationship, Drug, biology, Wnt signaling pathway, Antibodies, Monoclonal, Molecular biology, High-Throughput Screening Assays, Cell biology, 030104 developmental biology, medicine.anatomical_structure, Adenomatous Polyposis Coli, Proteasome, Catenin, biology.protein, Molecular Medicine, Drug Screening Assays, Antitumor, Signal transduction, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::98f29be05bd84e79ed27e00301943936
https://doi.org/10.1177/1087057115620169