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المؤلفون: Arie Zask, Pawel Nowak, Robert T. Abraham, James J. Gibbons, Tarek S. Mansour, Semiramis Ayral-Kaloustian, John Ellingboe, Derek C. Cole, David J. Malwitz, Kevin Curran, Jeroen Verheijen, Jamie Kim, Boris Shor, Judy Lucas, Wei-Guo Zhang, Celine Shi, Lourdes Toral-Barza, Ker Yu
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::af5af9a5271aa0276274bef18b48d37d
https://doi.org/10.1158/0008-5472.22378673.v1 -
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المؤلفون: Xiaoran S. Yang, Michael D. Arensman, Mary Mileski, Fang Wang, Christina H. Eng, Jeremy S. Myers, Robert T. Abraham, Danielle Leahy, Lourdes Toral-Barza, Shibing Deng, Edward Rosfjord
المصدر: Proceedings of the National Academy of Sciences of the United States of America
مصطلحات موضوعية: Medical Sciences, Amino Acid Transport System y+, medicine.medical_treatment, T cell, T-Lymphocytes, T cells, Antigen-Presenting Cells, Biology, medicine.disease_cause, Cell Line, Mice, Immune system, In vivo, medicine, cancer, Animals, Cell Proliferation, chemistry.chemical_classification, cystine, Mice, Knockout, Reactive oxygen species, Multidisciplinary, xCT, Cancer, Immunotherapy, Neoplasms, Experimental, Biological Sciences, medicine.disease, Glutathione, medicine.anatomical_structure, chemistry, PNAS Plus, Cancer cell, Cancer research, Immunologic Memory, Oxidative stress, Gene Deletion
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::33dbe7ee0e6b5a6ef16144037f68c55b
http://europepmc.org/articles/PMC6511047 -
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المؤلفون: Jiang Wu, Ker Yu, Xuesai Zhang, Yaqing Chen, Hui Zhao, Celine Shi, Jianchang Qian, Qun He, Lourdes Toral-Barza
المصدر: Oncotarget
مصطلحات موضوعية: 0301 basic medicine, medicine.medical_specialty, ATP citrate lyase, Class I Phosphatidylinositol 3-Kinases, Receptor, ErbB-2, cancer metabolism, Breast Neoplasms, mTORC1, Mechanistic Target of Rapamycin Complex 2, Biology, mTORC2, 03 medical and health sciences, 0302 clinical medicine, breast cancer, Acetyl Coenzyme A, Internal medicine, Cell Line, Tumor, medicine, lipid synthesis, Humans, skin and connective tissue diseases, Mechanistic target of rapamycin, PI3K/AKT/mTOR pathway, Kinase, Cell growth, Lipogenesis, TOR Serine-Threonine Kinases, musculoskeletal system, 030104 developmental biology, Endocrinology, Oncology, 030220 oncology & carcinogenesis, Cancer research, biology.protein, ATP Citrate (pro-S)-Lyase, Female, Research Paper
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::04b381de86fd84fb0d7b5bc60f5cad69
http://europepmc.org/articles/PMC5041899 -
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المؤلفون: Christina H. Eng, Lourdes Toral-Barza, Judy Lucas, Elizabeth George, Leon Murphy, Stephanie Fitzgerald, Zuncai Wang, Kevin Bray, Valeria Fantin, Rowena De Jesus, Gregory McAllister, Gregory R. Hoffman, Diane Tkach, Beat Nyfeler, Shanming Liu, Luanna Lemon, Robert T. Abraham, Elizabeth Frias, Nadire Cochran, Savuth Ugwonali
المصدر: Proceedings of the National Academy of Sciences of the United States of America. 113(1)
مصطلحات موضوعية: 0301 basic medicine, Indoles, Antineoplastic Agents, Ubiquitin-Activating Enzymes, Biology, medicine.disease_cause, Autophagy-Related Protein 7, Radiation Tolerance, Proto-Oncogene Proteins p21(ras), 03 medical and health sciences, chemistry.chemical_compound, Erlotinib Hydrochloride, Gene Knockout Techniques, Chloroquine, Cell Line, Tumor, medicine, Autophagy, Sunitinib, Humans, Pyrroles, Protein Kinase Inhibitors, Cell Proliferation, Multidisciplinary, Cell growth, Biological Sciences, 030104 developmental biology, Cell Transformation, Neoplastic, chemistry, Drug Resistance, Neoplasm, Mutation, Cancer research, Erlotinib, KRAS, Growth inhibition, Carcinogenesis, Tyrosine kinase, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::acb4a85f8fc633e0ef94a495d525798c
https://pubmed.ncbi.nlm.nih.gov/26677873 -
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المؤلفون: Hwei-Ru Tsou, George Theodore Grosu, Semiramis Ayral-Kaloustian, Natasja Brooijmans, Joel Bard, Ker Yu, Matthew Gregory Bursavich, Tarek S. Mansour, Gary Harold Birnberg, Irwin Hollander, Lourdes Toral-Barza, Gloria Jean Macewan
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:2321-2325
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Clinical Biochemistry, Mice, Nude, Pharmaceutical Science, Antineoplastic Agents, Protein Serine-Threonine Kinases, Crystallography, X-Ray, Biochemistry, Inhibitory Concentration 50, Mice, Phosphatidylinositol 3-Kinases, Structure-Activity Relationship, chemistry.chemical_compound, Adenosine Triphosphate, Microsomes, Neoplasms, Drug Discovery, Animals, Humans, Transferase, Methylene, Protein Kinase Inhibitors, Molecular Biology, PI3K/AKT/mTOR pathway, Benzofurans, Serine/threonine-specific protein kinase, Phosphoinositide 3-kinase, biology, Hydrogen bond, Chemistry, Kinase, TOR Serine-Threonine Kinases, Organic Chemistry, Intracellular Signaling Peptides and Proteins, biology.protein, Molecular Medicine, Selectivity
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المؤلفون: Judy Lucas, Ker Yu, Kevin J. Curran, David J. Richard, Lourdes Toral-Barza, Jeroen C. Verheijen, Joshua Kaplan, Irwin Hollander, Arie Zask
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:2644-2647
مصطلحات موضوعية: Stereochemistry, Morpholines, Clinical Biochemistry, Mice, Nude, Pharmaceutical Science, Protein Serine-Threonine Kinases, Biochemistry, Inhibitory Concentration 50, Mice, chemistry.chemical_compound, Adenosine Triphosphate, Nude mouse, In vivo, Morpholine, Drug Discovery, Animals, Molecular Biology, PI3K/AKT/mTOR pathway, Triazine, biology, Triazines, Drug discovery, Kinase, TOR Serine-Threonine Kinases, Organic Chemistry, Intracellular Signaling Peptides and Proteins, biology.organism_classification, In vitro, chemistry, Molecular Medicine
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المؤلفون: Irwin Hollander, Arie Zask, Ker Yu, Lourdes Toral-Barza, Jeroen C. Verheijen
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:375-379
مصطلحات موضوعية: Stereochemistry, Morpholines, Clinical Biochemistry, Pharmaceutical Science, Protein Serine-Threonine Kinases, Biochemistry, Chemical synthesis, Phosphatidylinositol 3-Kinases, Structure-Activity Relationship, chemistry.chemical_compound, Cell Line, Tumor, Morpholine, Drug Discovery, Humans, Structure–activity relationship, Molecular Biology, PI3K/AKT/mTOR pathway, Phosphoinositide-3 Kinase Inhibitors, Octane, chemistry.chemical_classification, Bicyclic molecule, Chemistry, TOR Serine-Threonine Kinases, Organic Chemistry, Intracellular Signaling Peptides and Proteins, Pyrimidines, Enzyme, Molecular Medicine, Selectivity, Tropanes