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1
المؤلفون: Janeta Popovici-Muller, Lenny Dang, Scott A. Biller, Nelamangala Nagaraja, Hua Yang, Shinsan M. Su, Yue Chen, Liping Yan, Hyeryun Kim, Lemieux Rene M, Luke Utley, Bin Fan
المصدر: Drug Metabolism and Disposition. 49:870-881
مصطلحات موضوعية: IDH1, CYP2B6, Metabolic Clearance Rate, Pyridines, Glycine, Pharmaceutical Science, Antineoplastic Agents, Drug Elimination Routes, Pharmacology, Glutarates, Mice, Dogs, Cytochrome P-450 Enzyme System, Pharmacokinetics, In vivo, Animals, Humans, Point Mutation, Drug Interactions, Dose-Response Relationship, Drug, CYP3A4, Chemistry, Myeloid leukemia, Haplorhini, Xenograft Model Antitumor Assays, Isocitrate Dehydrogenase, Rats, Leukemia, Myeloid, Acute, Isocitrate dehydrogenase, Ketoglutaric Acids, Drug metabolism, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3f57647f928757a03f343f00f8fa0f98
https://doi.org/10.1124/dmd.120.000234 -
2
المؤلفون: Jennifer R. Molina, Joseph M. Gozgit, Melissa M. Vasbinder, Ryan P. Abo, Kaiko kunii, Kristy G. Kuplast-Barr, Bin Gui, Sunaina P. Nayak, Elena Minissale, Kerren K. Swinger, Tim J. Wigle, Alvin Z. Lu, Danielle J. Blackwell, Christina R. Majer, Yue Ren, Ellen Bamberg, Mario Niepel, Jan-Rung Mo, William D. Church, Ahmed S. Mady, Jeff Song, Zacharenia A. Varsamis, Luke Utley, Patricia E. Rao, Timoty J. Mitchison, Kevin W. Kuntz, Victoria M. Richon, Kristen McEachern, Heike Keilhack
المصدر: Cancer Research. 82:2154-2154
مصطلحات موضوعية: Cancer Research, Oncology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::138b6edb388c9ff28b5c6026a9134c0a
https://doi.org/10.1158/1538-7445.am2022-2154 -
3
المؤلفون: Tim J. Wigle, Luke Utley, Kevin Wayne Kuntz, Jeff Song, Jan-Rung Mo, W. David Church, Sunaina P. Nayak, Heike Keilhack, Yue Ren, Alvin Lu, Danielle J. Blackwell, Ryan Abo, Kaiko Kunii, Christina R. Majer, Ahmed S.A. Mady, Melissa M. Vasbinder, Ellen Bamberg, Kerren Kalai Swinger, Bin Gui, Victoria M. Richon, Mario Niepel, Patricia E. Rao, Kristy Kuplast-Barr, Jennifer R. Molina, Timothy J. Mitchison, Joseph M. Gozgit, Elena Minissale, Zacharenia A. Varsamis
المصدر: Cancer cell. 39(9)
مصطلحات موضوعية: Cancer Research, Cell Survival, Nucleoside Transport Proteins, Adaptive Immunity, Small Molecule Libraries, Mice, Immune system, Interferon, Cell Line, Tumor, Neoplasms, medicine, Animals, Humans, Lung cancer, Cell Proliferation, Innate immune system, Chemistry, Cell growth, Cancer, medicine.disease, Xenograft Model Antitumor Assays, HEK293 Cells, Oncology, Drug Resistance, Neoplasm, Cancer cell, Interferon Type I, Cancer research, Nucleic acid, Tumor Escape, medicine.drug, HeLa Cells, Signal Transduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::07edb791c59df419eedd1a9ffce03541
https://pubmed.ncbi.nlm.nih.gov/34375612 -
4
المؤلفون: Thomas R Parr, Luke Utley, Thomas Zabawa, Akash Jain, Michael J. Pucci
المصدر: Expert Review of Anti-infective Therapy. 16:513-522
مصطلحات موضوعية: Adult, 0301 basic medicine, Microbiology (medical), Carbapenem, medicine.medical_specialty, medicine.drug_class, Tebipenem, 030106 microbiology, Antibiotics, Administration, Oral, Microbiology, Unmet needs, Beta-lactam, 03 medical and health sciences, chemistry.chemical_compound, Antibiotic resistance, Virology, Drug Resistance, Bacterial, Gram-Negative Bacteria, polycyclic compounds, medicine, Animals, Humans, Prodrugs, Intensive care medicine, business.industry, biochemical phenomena, metabolism, and nutrition, bacterial infections and mycoses, Anti-Bacterial Agents, Infectious Diseases, Carbapenems, chemistry, Drug Design, Community setting, Gram-Negative Bacterial Infections, business, medicine.drug
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5
المؤلفون: Hua Yang, Muriel D. David, Jeffrey O. Saunders, Lemieux Rene M, Gui Yao, Luke Utley, Véronique Saada, Xiaobing Lv, Yue Chen, Fang Wang, Shengfang Jin, Ping Chen, Erin Artin, Stéphane de Botton, Cheng Fang, Hyeryun Kim, Giovanni Cianchetta, Stefan Gross, Lenny Dang, Zhenwei Cai, Scott A. Biller, Andrew J. Olaharski, Erica Tobin, Cui Dawei, Katharine E. Yen, Virginie Penard-Lacronique, Liping Yan, Ding Zhou, Lee Silverman, Cyril Quivoron, Zhiyong Luo, Jeremy Travins, Janeta Popovici-Muller, Shinsan M. Su, Kimberly Straley, Zhiwei Gu, Francesco G. Salituro
المصدر: ACS Medicinal Chemistry Letters
مصطلحات موضوعية: mutant IDH1, 0301 basic medicine, Letter, IDH1, ivosidenib, Cellular differentiation, Point mutation, Organic Chemistry, Mutant, 2-hydroxyglutarate, Biology, Biochemistry, AG-120, 03 medical and health sciences, differentiation therapy, 030104 developmental biology, 0302 clinical medicine, Isocitrate dehydrogenase, Differentiation therapy, 030220 oncology & carcinogenesis, Drug Discovery, Cancer cell, Cancer research, isocitrate dehydrogenase, Ex vivo
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6
المؤلفون: Luke Utley, Kaiko Kunii, Danielle J. Blackwell, Ryan Abo, Jan-Rung Mo, Mario Niepel, Yue Ren, David Church, Joseph M. Gozgit, Kevin Wayne Kuntz, Patricia E. Rao, Kerren Kalai Swinger, Jeff Song, Melissa Vasbinder, Kristy Kuplast-Barr, Victoria M. Richon, Timothy J. Mitchison, Christina R. Majer, Alvin Lu, Bin Gui, Jennifer R. Molina, Elena Minissale, Heike Keilhack, Tim J. Wigle, Ellen Bamberg
المصدر: Cancer Research. 81:48-48
مصطلحات موضوعية: Cancer Research, biology, Chemistry, Acquired immune system, Olaparib, chemistry.chemical_compound, Immune system, Oncology, Interferon, Cancer cell, biology.protein, medicine, Cancer research, Cytotoxic T cell, STAT1, CD8, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::cbbdce3f5b4baab19e0042b551ef0b95
https://doi.org/10.1158/1538-7445.am2021-48 -
7
المؤلفون: Kaiko Kunii, W. David Church, Danielle J. Blackwell, Kevin Wayne Kuntz, Tim J. Wigle, Kristen McEachern, Heike Keilhack, Yue Ren, Laurie B. Schenkel, Ellen Bamberg, Prashant Shambharkar, Melissa Vasbinder, Kristy Kuplast-Barr, Christina R. Majer, Joseph M. Gozgit, Jenkins L. Lemera, Luke Utley, Victoria M. Richon, Mario Niepel
المصدر: Cancer Research. 81:1344-1344
مصطلحات موضوعية: Cancer Research, Chemistry, Effector, T cell, CD38, medicine.anatomical_structure, Immune system, Oncology, Cancer cell, medicine, Cancer research, Extracellular, NAD+ kinase, Intracellular
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::0c751ca50b9bf2528b2979338f802eef
https://doi.org/10.1158/1538-7445.am2021-1344 -
8
المؤلفون: Gerald Steven Falchook, Erika Manyak, Kristen McEachern, Viviana Bozon, Sudha Parasuraman, Kristy Kuplast-Barr, Luke Utley, Lisa D. Cleary, Timothy A. Yap, Melissa Lynne Johnson, Manish R. Patel
المصدر: Journal of Clinical Oncology. 39:3000-3000
مصطلحات موضوعية: Cancer Research, Oncology, business.industry, Interferon, Cancer research, Nucleic acid, Medicine, In patient, First in human, business, Therapeutic strategy, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::0a78ba58d8c6989cf34e182b20cad0cf
https://doi.org/10.1200/jco.2021.39.15_suppl.3000 -
9
المؤلفون: Grayson Moore, Luke Utley, Erika Manyak, Akash Jain, Susannah M. Walpole, Aaron Dane, David Melnick, Paul B. Eckburg
المصدر: Antimicrobial Agents and Chemotherapy
مصطلحات موضوعية: Adult, Diarrhea, Male, medicine.medical_specialty, Carbapenem, Tebipenem, Cmax, Administration, Oral, Urine, Clinical Therapeutics, Placebo, Gastroenterology, carbapenem, Food-Drug Interactions, oral, 03 medical and health sciences, chemistry.chemical_compound, Pharmacokinetics, tebipenem, Internal medicine, Humans, Medicine, Prodrugs, Pharmacology (medical), Adverse effect, 030304 developmental biology, Pharmacology, 0303 health sciences, 030306 microbiology, business.industry, Fasting, Healthy Volunteers, Anti-Bacterial Agents, Infectious Diseases, Carbapenems, chemistry, Female, medicine.symptom, business, pharmacokinetics, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c736b1dd9ae03c7f8608361a4acdafae
https://doi.org/10.1128/aac.00618-19 -
10
المؤلفون: Tim Keutzer, Scott Coleman, John Tomayko, Troy Lister, Susannah M. Walpole, Paul B. Eckburg, Luke Utley, Ellen Kopp, Nicholas Farinola
المصدر: Antimicrobial Agents and Chemotherapy
مصطلحات موضوعية: Adult, Male, medicine.drug_class, Antibiotics, Cmax, Aztreonam, Pharmacology, Clinical Therapeutics, Placebo, beta-Lactams, Ceftazidime, SPR741, Drug Administration Schedule, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, Double-Blind Method, medicine, Humans, Pharmacology (medical), Drug Interactions, 030212 general & internal medicine, 0303 health sciences, drug interaction, Dose-Response Relationship, Drug, 030306 microbiology, business.industry, potentiator, Drug interaction, Healthy Volunteers, Anti-Bacterial Agents, Infectious Diseases, Piperacillin, Tazobactam Drug Combination, Tolerability, chemistry, Area Under Curve, lipids (amino acids, peptides, and proteins), Administration, Intravenous, Female, business, pharmacokinetics, Polymyxin B, medicine.drug, Antimicrobial Cationic Peptides
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::01a2253c57e6da616e6099402042864d
http://europepmc.org/articles/PMC6709486