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1دورية أكاديمية
المؤلفون: Andreas Masch, Abed Nasereddin, Arne Alder, Megan J. Bird, Sandra I. Schweda, Lutz Preu, Christian Doerig, Ron Dzikowski, Tim W. Gilberger, Conrad Kunick
المصدر: Malaria Journal, Vol 18, Iss 1, Pp 1-10 (2019)
مصطلحات موضوعية: Anti-malarial drugs, Atropisomers, Axial chirality, Drug discovery, Malaria, PfGSK-3, Arctic medicine. Tropical medicine, RC955-962, Infectious and parasitic diseases, RC109-216
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Hilke Burmeister, Pascal Dietze, Lutz Preu, Julia E. Bandow, Ingo Ott
المصدر: Molecules, Vol 26, Iss 14, p 4282 (2021)
مصطلحات موضوعية: antibacterial, N-heterocyclic carbenes, ruthenium, thioredoxin reductase, Organic chemistry, QD241-441
وصف الملف: electronic resource
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3دورية أكاديمية
المؤلفون: Thomas Weidner, Leonardo Lucantoni, Abed Nasereddin, Lutz Preu, Peter G. Jones, Ron Dzikowski, Vicky M. Avery, Conrad Kunick
المصدر: Malaria Journal, Vol 16, Iss 1, Pp 1-10 (2017)
مصطلحات موضوعية: Anti-malaria drugs, Coenzyme A synthesis, Drug discovery, Malaria, 1,3,4-Oxadiazole, Oxazole, Arctic medicine. Tropical medicine, RC955-962, Infectious and parasitic diseases, RC109-216
وصف الملف: electronic resource
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4دورية أكاديمية
المؤلفون: Anne Walter, Apirat Chaikuad, Renate Helmer, Nadège Loaëc, Lutz Preu, Ingo Ott, Stefan Knapp, Laurent Meijer, Conrad Kunick
المصدر: PLoS ONE, Vol 13, Iss 5, p e0196761 (2018)
وصف الملف: electronic resource
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5دورية أكاديمية
المؤلفون: Rosanna Meine, Walter Becker, Hannes Falke, Lutz Preu, Nadège Loaëc, Laurent Meijer, Conrad Kunick
المصدر: Molecules, Vol 23, Iss 2, p 64 (2018)
مصطلحات موضوعية: DYRK1A, fraction of saturation, fragment-based drug development, indole, lipophilicity, molecular docking, protein kinase inhibitor, solubility, Organic chemistry, QD241-441
وصف الملف: electronic resource
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6دورية أكاديمية
المؤلفون: Thomas Weidner, Abed Nasereddin, Lutz Preu, Johann Grünefeld, Ron Dzikowski, Conrad Kunick
المصدر: Molecules, Vol 21, Iss 2, p 223 (2016)
مصطلحات موضوعية: diarylether, luciferase, Malaria, 2-phenoxyanilide, Plasmodium falciparum, TCAMS, TCMDC-137332, Organic chemistry, QD241-441
وصف الملف: electronic resource
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7
المؤلفون: Julia E. Bandow, Ingo Ott, Hilke Burmeister, Pascal Dietze, Lutz Preu
المصدر: Molecules, Vol 26, Iss 4282, p 4282 (2021)
Molecules
Volume 26
Issue 14مصطلحات موضوعية: Models, Molecular, Thioredoxin-Disulfide Reductase, Stereochemistry, Thioredoxin reductase, N-heterocyclic carbenes, Pharmaceutical Science, chemistry.chemical_element, Organic chemistry, Bacillus subtilis, 010402 general chemistry, medicine.disease_cause, 01 natural sciences, Article, Analytical Chemistry, chemistry.chemical_compound, QD241-441, Bacterial Proteins, Coordination Complexes, Heterocyclic Compounds, Drug Discovery, medicine, Humans, Physical and Theoretical Chemistry, Candida albicans, ruthenium, Escherichia coli, chemistry.chemical_classification, biology, Bacteria, 010405 organic chemistry, thioredoxin reductase, Bacterial Infections, biology.organism_classification, 0104 chemical sciences, Ruthenium, Anti-Bacterial Agents, antibacterial, Enzyme, chemistry, Chemistry (miscellaneous), Molecular Medicine, Carbene, Methane
وصف الملف: application/pdf
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8
المؤلفون: Till Beuerle, David Kaufholdt, Robert Hänsch, Ludger Beerhues, Mariam Gaid, Poonam Singh, Lutz Preu
المصدر: The Plant journal : for cell and molecular biologyREFERENCES. 104(6)
مصطلحات موضوعية: 0106 biological sciences, 0301 basic medicine, Coenzyme A, Xanthones, Plant Science, 01 natural sciences, 03 medical and health sciences, chemistry.chemical_compound, Cytosol, Biosynthesis, Xanthone, Coenzyme A Ligases, Genetics, Peroxisomes, Cloning, Molecular, Peroxisomal targeting signal, Phylogeny, Benzoic acid, Plant Proteins, chemistry.chemical_classification, DNA ligase, biology, Active site, Cell Biology, Molecular Docking Simulation, 030104 developmental biology, Enzyme, Biochemistry, chemistry, biology.protein, Acyl Coenzyme A, Hypericum, Metabolic Networks and Pathways, 010606 plant biology & botany
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9Scaffold hopping identifies 6,8-disubstituted purines as novel anaplastic lymphoma kinase inhibitors
المؤلفون: Michael H.G. Kubbutat, Markus Immer, Frank Totzke, Lutz Preu, Conrad Kunick, Christoph Schächtele, Laura Schlütke
المصدر: European Journal of Pharmaceutics and Biopharmaceutics. 126:89-94
مصطلحات موضوعية: 0301 basic medicine, Purine, C-Met, medicine.drug_class, Receptor Protein-Tyrosine Kinases, Pharmaceutical Science, Antineoplastic Agents, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, hemic and lymphatic diseases, medicine, Humans, Structure–activity relationship, Anaplastic lymphoma kinase, Anaplastic Lymphoma Kinase, Binding site, Purine metabolism, Protein Kinase Inhibitors, Binding Sites, General Medicine, Protein kinase inhibitor, Protein Structure, Tertiary, Molecular Docking Simulation, 030104 developmental biology, chemistry, Biochemistry, Purines, 030220 oncology & carcinogenesis, Biotechnology
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10
المؤلفون: Andreas, Masch, Abed, Nasereddin, Arne, Alder, Megan J, Bird, Sandra I, Schweda, Lutz, Preu, Christian, Doerig, Ron, Dzikowski, Tim W, Gilberger, Conrad, Kunick
المصدر: Malaria Journal
مصطلحات موضوعية: Thienopyridines, Pyridines, Drug discovery, PfGSK-3, Research, Plasmodium falciparum, Protozoan Proteins, Atropisomers, Axial chirality, Protein kinase, Malaria, Anti-malaria drugs, Antimalarials, Glycogen Synthase Kinase 3, Structure-Activity Relationship, HEK293 Cells, Humans, Malaria, Falciparum, Thorpe cyclization