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1دورية أكاديمية
المؤلفون: Laura Braconi, Chiara Riganti, Astrid Parenti, Marta Cecchi, Alessio Nocentini, Gianluca Bartolucci, Marta Menicatti, Marialessandra Contino, Nicola Antonio Colabufo, Dina Manetti, Maria Novella Romanelli, Claudiu T. Supuran, Elisabetta Teodori
المصدر: Molecules, Vol 29, Iss 14, p 3290 (2024)
مصطلحات موضوعية: MDR reversers, P-gp modulators, CA XII inhibitors, K562/DOX, HT29/DOX, A549/DOX, Organic chemistry, QD241-441
وصف الملف: electronic resource
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2دورية أكاديمية
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3دورية أكاديمية
المؤلفون: Laura Braconi, Gianluca Bartolucci, Marialessandra Contino, Niccolò Chiaramonte, Roberta Giampietro, Dina Manetti, Maria Grazia Perrone, Maria Novella Romanelli, Nicola Antonio Colabufo, Chiara Riganti, Silvia Dei, Elisabetta Teodori
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 974-992 (2020)
مصطلحات موضوعية: tetrahydroisoquinoline, mdr reversers, p-gp modulators, co-administration assay, cytotoxicity, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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4دورية أكاديمية
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5دورية أكاديمية
المؤلفون: Elisabetta Teodori, Laura Braconi, Silvia Bua, Andrea Lapucci, Gianluca Bartolucci, Dina Manetti, Maria Novella Romanelli, Silvia Dei, Claudiu T. Supuran, Marcella Coronnello
المصدر: Molecules, Vol 25, Iss 7, p 1748 (2020)
مصطلحات موضوعية: MDR reversers, P-gp modulators, CA XII inhibitors, K562/DOX, LoVo/DOX, hybrid compounds, Organic chemistry, QD241-441
وصف الملف: electronic resource
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المؤلفون: Braconi, Laura, Bartolucci, Gianluca, Contino, Marialessandra, Chiaramonte, Niccolò, Giampietro, Roberta, Manetti, Dina, Perrone, Maria Grazia, Romanelli, Maria Novella, Colabufo, Nicola Antonio, Riganti, Chiara, Dei, Silvia, Teodori, Elisabetta
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 974-992 (2020)مصطلحات موضوعية: Tariquidar, Antineoplastic Agents, ATP-binding cassette transporter, RM1-950, co-administration assay, cytotoxicity, MDR reversers, P-gp modulators, Tetrahydroisoquinoline, 01 natural sciences, Structure-Activity Relationship, chemistry.chemical_compound, Hydrolysis, Dogs, Neoplasms, Tetrahydroisoquinolines, Enzymatic hydrolysis, Amide, Drug Discovery, medicine, Animals, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, Cells, Cultured, Pharmacology, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Aryl, Esters, General Medicine, Amides, Combinatorial chemistry, Drug Resistance, Multiple, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry, Doxorubicin, Drug Resistance, Neoplasm, Therapeutics. Pharmacology, Drug Screening Assays, Antitumor, Selectivity, Research Paper, medicine.drug
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المؤلفون: Maria Novella Romanelli, Elisabetta Teodori, Dina Manetti, Claudiu T. Supuran, Gianluca Bartolucci, Marcella Coronnello, Laura Braconi, Silvia Bua, Andrea Lapucci, Silvia Dei
المصدر: Molecules
Volume 25
Issue 7
Molecules, Vol 25, Iss 1748, p 1748 (2020)مصطلحات موضوعية: Pharmaceutical Science, hybrid compounds, Analytical Chemistry, 0302 clinical medicine, Drug Stability, Drug Discovery, Cytotoxicity, Carbonic Anhydrase Inhibitors, P-glycoprotein, Carbonic Anhydrases, 0303 health sciences, biology, Molecular Structure, Chemistry, Drug Resistance, Multiple, LoVo/DOX, Chemistry (miscellaneous), 030220 oncology & carcinogenesis, selective chemosensitizers, Molecular Medicine, Efflux, MDR reversers, medicine.drug, circulatory and respiratory physiology, animal structures, PH reduction, Antineoplastic Agents, Article, lcsh:QD241-441, 03 medical and health sciences, Structure-Activity Relationship, lcsh:Organic chemistry, medicine, Humans, Doxorubicin, cardiovascular diseases, ATP Binding Cassette Transporter, Subfamily B, Member 1, Physical and Theoretical Chemistry, 030304 developmental biology, CA XII inhibitors, Dual P-gp/CA XII inhibitory activity, Hybrid compounds, K562/DOX, Multitarget ligands, P-gp modulators, Selective chemosensitizers, multitarget ligands, Organic Chemistry, Biological Transport, Molecular biology, Multiple drug resistance, Drug Resistance, Neoplasm, Cancer cell, biology.protein, dual P-gp/CA XII inhibitory activity, K562 Cells, K562 cells
وصف الملف: application/pdf
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المؤلفون: Ottavia Spiga, Niccolò Chiaramonte, Milena Salerno, Silvia Dei, Marta Menicatti, Laura Braconi, Chatchanok Udomtanakunchai, Marcella Coronnello, Marialessandra Contino, Maria Grazia Perrone, Gianluca Bartolucci, Nicola Antonio Colabufo, Elisabetta Teodori, Alfonso Trezza, Maria Novella Romanelli, Dina Manetti
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Antineoplastic Agents, 01 natural sciences, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Tumor Cells, Cultured, ATP Binding Cassette Transporter, Subfamily G, Member 2, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, Amines, 030304 developmental biology, P-glycoprotein, Pharmacology, 0303 health sciences, biology, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Aryl, Organic Chemistry, Esters, General Medicine, Drug Resistance, Multiple, 0104 chemical sciences, Neoplasm Proteins, Multiple drug resistance, chemistry, Docking (molecular), Drug Resistance, Neoplasm, biology.protein, Amine gas treating, Multidrug Resistance-Associated Protein 1, Efflux, Caco-2 Cells, Multidrug Resistance-Associated Proteins, K562 Cells, 1-(3-dimethylaminopropyl)-3-ethylcarbodiimmide hydrochloride, 4-Dimethylaminopyridine, Apparent permeability, ATPase activity, BCRP, BCRP modulators, Breast cancer resistance protein, Caco-2 cells, Colorectal adenocarcinoma cells, DMAP, DOX, Doxorubicin, EDCI, Human plasma stability, KEE, Ketoprofen Ethyl Ester, Madin-Darby Canin Kidney, MDCK, MDR reversers, Molecular docking, MRP1, MRP1 modulators, Multidrug resistance associated protein 1, P-gp, P-gp modulators, PBS, PDB, Phosphate buffer solution, Pirarubicin uptake, Protein data bank, Rhd123, Rhodamine-123, Rhodamine-123 efflux, Topological polar surface area, TPSA, Linker, Dimerization
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e6a608570c490ee0bb2e3b1b660300c6
http://hdl.handle.net/2158/1152900 -
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المؤلفون: Milena Salerno, Chiara Riganti, Ottavia Spiga, Elena Gazzano, Dina Manetti, Asimidis Athanasios, Gianluca Bartolucci, Maria Novella Romanelli, Marialessandra Contino, Laura Braconi, Silvia Dei, Elisabetta Teodori, Alfonso Trezza, Nicola Antonio Colabufo, Maria Grazia Perrone, Roberta Giampietro
مصطلحات موضوعية: 01 natural sciences, Madin Darby Canine Kidney Cells, Stereocenter, chemistry.chemical_compound, Drug Discovery, Structural isomer, Amines, Collateral sensitivity, Enantiomers, Human plasma stability, K562 cells, MDCK cells, MDR reversers, Molecular docking, P-gp modulators, Cells, Cultured, 0303 health sciences, Molecular Structure, Esters, Stereoisomerism, General Medicine, Drug Resistance, Multiple, Molecular Docking Simulation, Amine gas treating, Stereochemistry, Antineoplastic Agents, Structure-Activity Relationship, 03 medical and health sciences, Dogs, Animals, Humans, Cell Proliferation, 030304 developmental biology, Pharmacology, Dose-Response Relationship, Drug, 010405 organic chemistry, Aryl, Organic Chemistry, 0104 chemical sciences, Multiple drug resistance, chemistry, Drug Resistance, Neoplasm, Docking (molecular), Drug Design, Drug Screening Assays, Antitumor, Enantiomer, K562 Cells, Methyl group
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::58cf81100cf01c1230b4c3abea16f8cf
http://hdl.handle.net/2158/1175670 -
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المؤلفون: Marcella Coronnello, Elisabetta Teodori, Niccolò Chiaramonte, Maria Novella Romanelli, Milena Salerno, Dina Manetti, Silvia Dei
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, gp modulators, MDR reversers, heterodimers, flavonoids, doxorubicin-resistant human erythroleukemia K562 cells (K562/DOX), pirarubicin uptak, 03 medical and health sciences, chemistry.chemical_compound, Residue (chemistry), Structure-Activity Relationship, 0302 clinical medicine, Drug Discovery, Tumor Cells, Cultured, Molecule, Moiety, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, Amines, Molecular Biology, P-glycoprotein, biology, Dose-Response Relationship, Drug, Molecular Structure, Aryl, Organic Chemistry, Esters, Flavones, Drug Resistance, Multiple, Multiple drug resistance, 030104 developmental biology, chemistry, Chromones, Drug Resistance, Neoplasm, 030220 oncology & carcinogenesis, Drug Design, Chromone, biology.protein, Molecular Medicine, Amine gas treating, K562 Cells, Dimerization
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d2bbe60ffb410153698af31004d333c2
http://hdl.handle.net/2158/1106055