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1
المؤلفون: Richard Martyn Angell, David W. Brown, Katherine Louise Jones, Smith Kathryn Jane, Ann Louise Walker, Penny A. Smee, Tim Longstaff, Paul Bamborough, Tony D. Angell, Stuart G. Cockerill, Chris D. Edwards, Don O. Somers, Murray J. B. Brown, Jacky B. Buckton, Malcolm Willson
المصدر: Bioorganicmedicinal chemistry letters. 18(1)
مصطلحات موضوعية: Models, Molecular, Stereochemistry, p38 mitogen-activated protein kinases, Clinical Biochemistry, Biphenyl derivatives, Molecular Conformation, Pharmaceutical Science, Administration, Oral, Non-specific serine/threonine protein kinase, Crystallography, X-Ray, Biochemistry, p38 Mitogen-Activated Protein Kinases, Piperazines, chemistry.chemical_compound, Structure-Activity Relationship, In vivo, Amide, Drug Discovery, Animals, Molecular Biology, Protein Kinase Inhibitors, chemistry.chemical_classification, Biphenyl, Oxadiazoles, Organic Chemistry, Biphenyl Compounds, Amides, Arthritis, Experimental, Rats, Enzyme, chemistry, Molecular Medicine, Protein Binding
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2
المؤلفون: David Spalding, Stuart Cockerill, Malcolm Clive Carter, Peter Topley, Lindy L. Thomsen, D. J. Hayes, Patrick M. Woollard, Jeremy N. Stables, Karen Affleck, Malcolm Willson, Colin Stubberfield, Robert D. Shaw, Amanda Jowett, Steve McKeown, Kathryn Jane Smith, Stephen Barry Guntrip
المصدر: Bioorganicmedicinal chemistry letters. 11(11)
مصطلحات موضوعية: Receptor, ErbB-2, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Mice, SCID, Biochemistry, Receptor tyrosine kinase, Mice, Epidermal growth factor, Drug Discovery, Tumor Cells, Cultured, Animals, Receptor, Molecular Biology, chemistry.chemical_classification, biology, Chemistry, Kinase, Organic Chemistry, Xenograft Model Antitumor Assays, ErbB Receptors, Disease Models, Animal, Enzyme, Pyrimidines, Enzyme inhibitor, Cell culture, Cancer research, biology.protein, Quinazolines, Molecular Medicine, Signal transduction, Cell Division