-
1دورية أكاديمية
المؤلفون: Paul A Clarke, Maria-Jesus Ortiz-Ruiz, Robert TePoele, Olajumoke Adeniji-Popoola, Gary Box, Will Court, Stephanie Czasch, Samer El Bawab, Christina Esdar, Ken Ewan, Sharon Gowan, Alexis De Haven Brandon, Phillip Hewitt, Stephen M Hobbs, Wolfgang Kaufmann, Aurélie Mallinger, Florence Raynaud, Toby Roe, Felix Rohdich, Kai Schiemann, Stephanie Simon, Richard Schneider, Melanie Valenti, Stefan Weigt, Julian Blagg, Andree Blaukat, Trevor C Dale, Suzanne A Eccles, Stefan Hecht, Klaus Urbahns, Paul Workman, Dirk Wienke
المصدر: eLife, Vol 5 (2016)
مصطلحات موضوعية: CDK8, inhibitor, Mediator complex, Wnt, super-enhancer, Medicine, Science, Biology (General), QH301-705.5
وصف الملف: electronic resource
-
2
المؤلفون: Loredana Puca, Michele S. Dowless, Carmen M. Perez-Ferreiro, Maria Jesus Ortiz-Ruiz, Gregory P. Donoho, Andrew Capen, Lysiane Huber, Sarah M. Bogner, Dongling Fei, Jason R. Manro, Chun Ping Yu, Wei Guo Xu, Rui Wang, Shuang Chen, Mark A. Hicks, Parisa Zolfaghari, Andrew Faber, Raymond Gilmour, Monica D. Ramstetter, Matthew T. Chang, Maria Jose Lallena, Xuequian Gong, David M. Hyman, Lillian M. Smyth, Barbara J. Brandhuber, Barry S. Taylor, Anke Klippel
المصدر: Cancer Research. 83:P4-08
مصطلحات موضوعية: Cancer Research, Oncology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::527fc9e133f9687e3e79e24c582b9519
https://doi.org/10.1158/1538-7445.sabcs22-p4-08-02 -
3
المؤلفون: Djordje Musil, Suzanne A. Eccles, Daniel Schwarz, Klaus Urbahns, Trevor Clive Dale, Paul A. Clarke, Christina Esdar, Paul Czodrowski, Maria-Jesus Ortiz-Ruiz, Oliver Pöschke, Florence I. Raynaud, Aurélie Mallinger, Dirk Wienke, Kai Schiemann, Richard Schneider, Felix Rohdich, Michael Busch, Julian Blagg
المصدر: Journal of Medicinal Chemistry. 59:9337-9349
مصطلحات موضوعية: 0301 basic medicine, High-throughput screening, Mice, Nude, Antineoplastic Agents, Pharmacology, Mice, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Cyclin-dependent kinase, Thiadiazoles, Drug Discovery, Biomarkers, Tumor, Animals, Humans, Structure–activity relationship, Protein Kinase Inhibitors, Cell Proliferation, Dose-Response Relationship, Drug, Molecular Structure, Oncogene, biology, Drug discovery, Kinase, Chemistry, Imidazoles, Wnt signaling pathway, Neoplasms, Experimental, Cyclin-Dependent Kinase 8, High-Throughput Screening Assays, 030104 developmental biology, 030220 oncology & carcinogenesis, biology.protein, Molecular Medicine, Cyclin-dependent kinase 8, Female, Drug Screening Assays, Antitumor
وصف الملف: application/pdf
-
4
المؤلفون: Alexis De Haven Brandon, Paul Workman, Aurélie Mallinger, Elizabeth Fraser, Mark Stubbs, Paul Czodrowski, Andree Blaukat, Richard Schneider, Julian Blagg, Djordje Musil, Melanie Valenti, Daniel Schwarz, Rahul S. Samant, Klaus Schneider, Kai Schiemann, Sharon Gowan, Christina Esdar, Florence I. Raynaud, Suzanne A. Eccles, Robert TePoele, Dennis Waalboer, Gary Box, Dirk Wienke, Oliver Poeschke, Paul A. Clarke, Maria-Jesus Ortiz-Ruiz, Kenneth Burnside Ramsay Ewan, Trevor Clive Dale, Felix Rohdich, Olajumoke Adeniji-Popoola, Will Court
المصدر: Nature chemical biology
مصطلحات موضوعية: Models, Molecular, Pyridines, Article, Mediator, Cyclin-dependent kinase, In vivo, Cell Line, Tumor, Humans, Spiro Compounds, Kinase activity, Protein Kinase Inhibitors, Molecular Biology, Molecular Structure, biology, Kinase, Wnt signaling pathway, Cell Biology, Cyclin-Dependent Kinase 8, Cyclin-Dependent Kinases, Cell biology, Biochemistry, Molecular Probes, Colonic Neoplasms, biology.protein, Cyclin-dependent kinase 8, Phosphorylation
-
5
المؤلفون: Toby Roe, Will Court, Felix Rohdich, Julian Blagg, Wolfgang Kaufmann, Stefan Hecht, Richard Schneider, Stephen M. Hobbs, Christina Esdar, Alexis De Haven Brandon, Samer El Bawab, Phllip Hewitt, Suzanne A. Eccles, Kai Schiemann, Trevor Clive Dale, Paul Workman, Aurélie Mallinger, Stefan Weigt, Klaus Urbahns, Olajumoke Adeniji-Popoola, Andree Blaukat, Stephanie Simon, Robert TePoele, Melanie Valenti, Sharon Gowan, Stefanie Czasch, Paul A. Clarke, Gary Box, Dirk Wienke, Kenneth Burnside Ramsay Ewan, Maria-Jesus Ortiz-Ruiz, Florence I. Raynaud
المصدر: eLife
eLife, Vol 5 (2016)مصطلحات موضوعية: 0301 basic medicine, Anti-Inflammatory Agents, Pharmacology, Mice, Neoplasms, Biology (General), media_common, Cancer Biology, Mediator Complex, Kinase, General Neuroscience, Wnt signaling pathway, General Medicine, Cyclin-Dependent Kinases, inhibitor, Treatment Outcome, Medicine, Heterografts, Stem cell, Research Article, Human, Drug, QH301-705.5, Science, media_common.quotation_subject, CDK8, Antineoplastic Agents, Biology, General Biochemistry, Genetics and Molecular Biology, 03 medical and health sciences, Wnt, Immune system, Cyclin-dependent kinase, super-enhancer, medicine, Animals, Humans, Human Biology and Medicine, Protein Kinase Inhibitors, Hyperplasia, General Immunology and Microbiology, Cancer, medicine.disease, Cyclin-Dependent Kinase 8, Disease Models, Animal, 030104 developmental biology, Cancer cell, biology.protein
وصف الملف: application/pdf
-
6
المؤلفون: Andree Blaukat, Sharon Gowan, Richard Schneider, Suzanne A. Eccles, Gary Box, Dirk Wienke, Paul Workman, Robert TePoele, Stefan Hecht, Kai Schiemann, Trevor Clive Dale, Paul A. Clarke, Melanie Valenti, Toby Roe, Felix Rohdich, Wolfgang Kaufmann, Stephanie Czasch, Maria-Jesus Ortiz-Ruiz, Christina Esdar, Stefan Weigt, Kenneth Burnside Ramsay Ewan, Aurélie Mallinger, Alexis De Haven Brandon, Phillip Hewitt, Olajumoke Adeniji-Popoola, Will Court, Florence I. Raynaud, Stephen M. Hobbs, Stephanie Simon, Julian Blagg, Samer El Bawab, Klaus Urbahns
مصطلحات موضوعية: Mediator, Chemistry, Kinase, Mechanism (biology), Cell biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::4fdc132145578e222df38589324159b5
https://doi.org/10.7554/elife.20722.047 -
7
المؤلفون: Julian Blagg, Suzanne A. Eccles, Phllip Hewitt, Olajumoke Adeniji-Popoola, Felix Rohdich, Maria-Jesus Ortiz-Ruiz, Aurélie Mallinger, Alexis De Haven Brandon, Kenneth Burnside Ramsay Ewan, Melanie Valenti, Paul A. Clarke, Christina Esdar, Gary Box, Paul Workman, Dirk Wienke, Richard Schneider, Robert te Poele, Kai Schiemann, Florence I. Raynaud, Wolfgang Kaufmann, Sharon Gowan, Stephanie Simon, Trevor Clive Dale
المصدر: Cancer Research. 77:129-129
مصطلحات موضوعية: Cancer Research, Mediator, Oncology, Chemistry, Mechanism (biology), Kinase, Cyclin-dependent kinase 8, Cell biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::683dfd73d2b6f076d885de97182d8459
https://doi.org/10.1158/1538-7445.am2017-129 -
8
المؤلفون: S M Hobbs, Julian Blagg, Will Court, Aurélie Mallinger, Olajumoke O. Popoola, Dirk Wienke, Christina Esdar, Kai Schiemann, Paul A. Clarke, Rahul S. Samant, Paul Workman, Sue Eccles, Maria-Jesus Ortiz-Ruiz, Mark Stubbs, Rosemary Burke, Robert TePoele
المصدر: Cancer Research. 76:3869-3869
مصطلحات موضوعية: Genetics, Cancer Research, Pregnane X receptor, Oncology, Cell culture, Kinase, Wnt signaling pathway, Cyclin-dependent kinase 8, Phosphorylation, Signal transduction, Biology, Transcription factor, Molecular biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::90af652c2c380e8401260272d6d280e9
https://doi.org/10.1158/1538-7445.am2016-3869 -
9
المؤلفون: Paul Czodrowski, Andree Blaukat, Frank Stieber, Julian Blagg, Djordje Musil, Felix Rohdich, Simon Crumpler, Rosemary Burke, Michael Busch, Kai Schiemann, Sharon Gowan, Michel Calderini, Stephanie Simon, Richard Schneider, Suzanne A. Eccles, Robert TePoele, Maria-Jesus Ortiz-Ruiz, Oliver Poeschke, Trevor Clive Dale, Florence I. Raynaud, Klaus Urbahns, Olajumoke Adeniji-Popoola, Wolfgang Kaufmann, Daniel Schwarz, Klaus Schneider, Aurélie Mallinger, Rahul S. Samant, Christian Rink, Christina Esdar, Mark Stubbs, Dennis Waalboer, Paul Workman, Paul A. Clarke, Dirk Wienke
المصدر: Cancer Research. 76:3025-3025
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Kinase, Wnt signaling pathway, Cancer, Context (language use), Pharmacology, Biology, medicine.disease, MED12, 03 medical and health sciences, 030104 developmental biology, Mediator, Oncology, In vivo, medicine, Cyclin-dependent kinase 8
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::205048a11978c437f58e8b431a90eeaa
https://doi.org/10.1158/1538-7445.am2016-3025 -
10
المؤلفون: Aurélie Mallinger, Trevor Clive Dale, Maria-Jesus Ortiz-Ruiz, Kai Schiemann, Christina Esdar, Robert te Poele, Suzanne A. Eccles, Kenneth Burnside Ramsay Ewan, Julian Blagg, Sharon Gowan, Olajumoke Adeniji-Popoola, Paul Workman, Dennis Waalboer, Dirk Wienke, Paul A. Clarke
المصدر: Molecular Cancer Therapeutics. 14:PR02-PR02
مصطلحات موضوعية: Cancer Research, Oncology, Kinase, Stable isotope labeling by amino acids in cell culture, Wnt signaling pathway, Cyclin-dependent kinase 8, Biology, Kinase activity, Proteomics, DNA-binding protein, Small molecule, Molecular biology, Cell biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::0f781a8c9722175dd6ccfb6d99a36d8b
https://doi.org/10.1158/1535-7163.targ-15-pr02