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1
المؤلفون: Christina N. DiMarco, Anthony L. Gotter, Alan T. Savitz, Joanne Stevens, Joseph G. Bruno, Tamara D. Cabalu, John J. Renger, Jason W. Skudlarek, Pamela L. Tannenbaum, Paul J. Coleman, Scott D. Kuduk, Joseph Brunner, Susan L. Garson, Christopher J. Winrow, Julie A. O'Brien, Charles M. Harrell, Mark H. Pausch
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:2488-2492
مصطلحات موضوعية: Filorexant, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Piperidines, Orexin Receptors, Sleep Initiation and Maintenance Disorders, mental disorders, Drug Discovery, medicine, Animals, Benzamide, Molecular Biology, G protein-coupled receptor, Organic Chemistry, Antagonist, Triazoles, Receptor antagonist, Orexin receptor, Rats, Orexin, Pyrimidines, chemistry, Molecular Medicine, Orexin Receptor Antagonists, Antagonism, Half-Life, Protein Binding, medicine.drug
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2
المؤلفون: Mark H. Pausch, John Dunlop, Stanley Nawoschik, Jean Y. Zhang, Dianne Kowal, Ravikumar Peri
المصدر: ASSAY and Drug Development Technologies. 8:106-113
مصطلحات موضوعية: biology, Phospholipase C, Chemistry, Inositol Phosphates, Chinese hamster ovary cell, Stimulation, CHO Cells, Ligands, biology.organism_classification, Molecular biology, Cricetulus, Förster resonance energy transfer, Biochemistry, Cricetinae, Drug Discovery, Fluorescence Resonance Energy Transfer, Receptor, Serotonin, 5-HT2C, Animals, Humans, Molecular Medicine, Calcium, Serotonin, Receptor, 5-HT receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::948dbefafd3cc39a7dead631bc6979ab
https://doi.org/10.1089/adt.2009.0205 -
3
المؤلفون: Steven M. Grauer, Peter J. Atkinson, Michael A. Olsen, Cody Kelley, Deborah L. Smith, Margaret Lai, Guoming Zhang, Feng Liu, Sharon Rosenzweig-Lipson, Chad E. Beyer, Michael Popiolek, Adam M. Gilbert, Mark Day, Karen L. Marquis, Radka Graf, Rachel Navarra, Claudine Pulicicchio, Farhana Pruthi, Xavier Z. Khawaja, Evguenia Kouranova, Sheree F. Logue, Tom A. Comery, Caitlin Wantuch, Mark H. Pausch, Nicholas J. Brandon
المصدر: Journal of Pharmacology and Experimental Therapeutics. 327:827-839
مصطلحات موضوعية: Allosteric modulator, Receptor, Metabotropic Glutamate 5, Allosteric regulation, Drug Evaluation, Preclinical, Prefrontal Cortex, CDPPB, Pharmacology, Receptors, Metabotropic Glutamate, Hippocampus, Cell Line, Cognition, Allosteric Regulation, Piperidines, Dopamine, Avoidance Learning, medicine, Animals, Humans, Phencyclidine, Brain Chemistry, Oxadiazoles, Dose-Response Relationship, Drug, Metabotropic glutamate receptor 5, Chemistry, Glutamate receptor, Rats, Metabotropic glutamate receptor, Molecular Medicine, Antipsychotic Agents, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7619d349d85d8c5594fdd5c791082951
https://doi.org/10.1124/jpet.108.136580 -
4
المؤلفون: Eugene Tseng, Ying Sun, Maria Blatcher, Jeremy Johnson, Lynn Zhang, Noel Taylor, Sreekumar Raman Kodangattil, Janet E. Paulsen, Stan P. Nawoschik, Brian Bates, David C. Kopsco, Angela Kramer, Hui Min Chen, Qin Shan, Mark H. Pausch
المصدر: Brain Research. 1087:1-14
مصطلحات موضوعية: Gs alpha subunit, G protein, Molecular Sequence Data, Gene Expression, Nerve Tissue Proteins, Biology, Transfection, Models, Biological, Cell Line, Receptors, G-Protein-Coupled, Mice, GTP-Binding Proteins, Genes, Reporter, Two-Hybrid System Techniques, Gene expression, Cyclic AMP, Animals, Humans, Genetic Testing, Cloning, Molecular, Molecular Biology, Gene, In Situ Hybridization, Gene Library, G protein-coupled receptor, Reporter gene, Messenger RNA, General Neuroscience, HEK 293 cells, Brain, Chromosome Mapping, Blotting, Northern, Molecular biology, Neurology (clinical), Developmental Biology
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5
المصدر: Bioinformatics. 20:3490-3499
مصطلحات موضوعية: Statistics and Probability, Computer science, Word error rate, Markov model, Machine learning, computer.software_genre, Biochemistry, Receptors, G-Protein-Coupled, Structure-Activity Relationship, GTP-Binding Proteins, Sequence Analysis, Protein, Protein Interaction Mapping, State space, Computer Simulation, Hidden Markov model, Molecular Biology, Sequence, Binding Sites, Models, Statistical, Sequence Homology, Amino Acid, business.industry, Pattern recognition, Markov Chains, Computer Science Applications, Computational Mathematics, Models, Chemical, Computational Theory and Mathematics, Coupling (computer programming), Test set, Artificial intelligence, business, Sequence Alignment, computer, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ba3d9f6da79c63e82d4821db765554d2
https://doi.org/10.1093/bioinformatics/bth434 -
6
المؤلفون: Mark H. Pausch, Lorena A. Kallal, Jeffrey L. Benovic, Beth Noble
المصدر: Journal of Biological Chemistry. 278:47466-47476
مصطلحات موضوعية: G protein-coupled receptor kinase, Growth factor receptor, G-Protein-Coupled Receptor Kinase 5, Biochemistry, Autophosphorylation, 5-HT5A receptor, Cell Biology, Biology, Interleukin-13 receptor, Molecular Biology, Protease-activated receptor 2, Insulin-like growth factor 1 receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::782c82cedf9e4a611cfa06ec7ec3e108
https://doi.org/10.1074/jbc.m308257200 -
7
المؤلفون: Evi Kostenis, Jürgen Wess, Clarice Schmidt, Isolde Erlenbach, Mark H. Pausch, Fadi F. Hamdan
المصدر: Journal of Neurochemistry. 77:1327-1337
مصطلحات موضوعية: Cellular and Molecular Neuroscience, Biochemistry, Muscarinic acetylcholine receptor M5, Muscarinic acetylcholine receptor M3, Muscarinic acetylcholine receptor M2, Class C GPCR, Muscarinic acetylcholine receptor M1, Biology, Receptor, Molecular biology, Rhodopsin-like receptors, G protein-coupled receptor
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8
المؤلفون: Danielle Raufaste, Clarice Schmidt, Mark H. Pausch, Evi Kostenis, Claudine Serradeil-Le Gal, Jürgen Wess, Mark E. Dumont, Isolde Erlenbach
المصدر: Journal of Biological Chemistry. 276:29382-29392
مصطلحات موضوعية: Models, Molecular, Receptors, Vasopressin, Saccharomyces cerevisiae Proteins, Molecular Sequence Data, Saccharomyces cerevisiae, Biology, Polymerase Chain Reaction, Biochemistry, Gamma-aminobutyric acid receptor subunit alpha-1, Protein Structure, Secondary, Animals, Humans, 5-HT5A receptor, Amino Acid Sequence, Cloning, Molecular, GABBR1, Molecular Biology, Nuclear receptor co-repressor 1, Protease-activated receptor 2, DNA Primers, Gene Library, Sequence Deletion, G protein-coupled receptor, G protein-coupled receptor kinase, Base Sequence, Sequence Homology, Amino Acid, Liver receptor homolog-1, Cell Membrane, Cell Biology, Heterotrimeric GTP-Binding Proteins, GTP-Binding Protein alpha Subunits, Arginine Vasopressin, Kinetics, Protein Subunits, Amino Acid Substitution, Oligodeoxyribonucleotides, Mutagenesis, Site-Directed, GTP-Binding Protein alpha Subunits, Gq-G11, Cattle, Sequence Alignment
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a918fc607f94d3eb5bcf6fde33a5b66c
https://doi.org/10.1074/jbc.m103203200 -
9
المصدر: Molecular and Cellular Biology. 15:6188-6195
مصطلحات موضوعية: Receptors, Peptide, G protein, Molecular Sequence Data, Saccharomyces cerevisiae, Pheromones, GTP-Binding Proteins, Animals, Somatostatin receptor 2, Somatostatin receptor 1, Receptors, Somatostatin, Molecular Biology, DNA Primers, Delta cell, Base Sequence, biology, Somatostatin receptor, Cell Membrane, Cell Biology, biology.organism_classification, Recombinant Proteins, Yeast, Rats, Biochemistry, Receptors, Mating Factor, Biological Assay, Signal transduction, Somatostatin, Cell Division, Research Article, Signal Transduction, Transcription Factors
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10
المؤلفون: Pranab K. Chanda, Eckart D. Gundelfinger, John F. Ross, Stephen J. Moss, Mark H. Pausch, Michael Popiolek, Erik I. Charych, Nicholas J. Brandon
المصدر: The Journal of biological chemistry. 286(33)
مصطلحات موضوعية: D-Amino-Acid Oxidase, Male, Immunoprecipitation, Population, D-amino acid oxidase, Presynaptic Terminals, Synaptic Membranes, Nerve Tissue Proteins, Biology, Biochemistry, Receptors, N-Methyl-D-Aspartate, Rats, Sprague-Dawley, chemistry.chemical_compound, Glutamatergic, Neurobiology, Cerebellum, Serine, Animals, Humans, Receptor, education, Neurotransmitter, Molecular Biology, education.field_of_study, Neuropeptides, Cell Biology, Rats, Cytoskeletal Proteins, Membrane protein, chemistry, Schizophrenia, Presynaptic active zone
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a22df65c67226db264a0f5131cec3c70
https://pubmed.ncbi.nlm.nih.gov/21700703