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1دورية أكاديمية
المؤلفون: Leslie W Tari, Xiaoming Li, Michael Trzoss, Daniel C Bensen, Zhiyong Chen, Thanh Lam, Junhu Zhang, Suk Joong Lee, Grayson Hough, Doug Phillipson, Suzanne Akers-Rodriguez, Mark L Cunningham, Bryan P Kwan, Kirk J Nelson, Amanda Castellano, Jeff B Locke, Vickie Brown-Driver, Timothy M Murphy, Voon S Ong, Chris M Pillar, Dean L Shinabarger, Jay Nix, Felice C Lightstone, Sergio E Wong, Toan B Nguyen, Karen J Shaw, John Finn
المصدر: PLoS ONE, Vol 8, Iss 12, p e84409 (2013)
وصف الملف: electronic resource
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المؤلفون: Gabriel M. Simon, Cheryl A. Grice, Micah J. Niphakis, Olivia D. Weber, R. Alan B. Ezekowitz, Nhi Ngo, Rachel A. Herbst, Jason R. Clapper, Justin S. Cisar, Iain P. Fraser, Jacqueline L. Blankman, Dylan M. Herbst, Mark L. Cunningham, Gary P. O'Neill, Todd K. Jones, Anna M. Knize, Alex Reed, Cassandra L. Henry, Aundrea R. Coppola, Andreu Viader, Jessica P. Alexander
المصدر: The Journal of pharmacology and experimental therapeutics. 367(3)
مصطلحات موضوعية: 0301 basic medicine, Male, Analgesic, Pain, Rodentia, Arachidonic Acids, Pharmacology, Degradative enzyme, Glycerides, Rats, Sprague-Dawley, 03 medical and health sciences, chemistry.chemical_compound, Mice, Piperidines, Cell Line, Tumor, medicine, Animals, Humans, Cyclooxygenase Inhibitors, Enzyme Inhibitors, ED50, Analgesics, Mice, Inbred ICR, biology, Hydrolysis, Prostanoid, Brain, Human brain, Antipruritics, Endocannabinoid system, Monoacylglycerol Lipases, Rats, Monoacylglycerol lipase, 030104 developmental biology, medicine.anatomical_structure, chemistry, PC-3 Cells, biology.protein, Prostaglandins, Molecular Medicine, Cyclooxygenase, Endocannabinoids
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ef38160293a49bd7fff58ad8eba72dc0
https://pubmed.ncbi.nlm.nih.gov/30305428 -
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المؤلفون: Bryan P. Kwan, Kirk J. Nelson, Grayson Hough, John T. Finn, Karen Joy Shaw, Mark Hilgers, Mark L. Cunningham, Thanh Lam, Michael Trzoss, Vickie Brown-Driver, Voon Ong
المصدر: Journal of Medicinal Chemistry. 57:651-668
مصطلحات موضوعية: Models, Molecular, Staphylococcus aureus, Benzimidazole, Stereochemistry, Microbial Sensitivity Tests, Cofactor, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Sepsis, Drug Resistance, Bacterial, Drug Discovery, Dihydrofolate reductase, Animals, Humans, Potency, Structure–activity relationship, chemistry.chemical_classification, biology, Wild type, Staphylococcal Infections, Anti-Bacterial Agents, Tetrahydrofolate Dehydrogenase, Streptococcus pneumoniae, Enzyme, chemistry, Quinazolines, biology.protein, Folic Acid Antagonists, Molecular Medicine, Benzimidazoles
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المصدر: SLAS Discovery. 18:1018-1026
مصطلحات موضوعية: DNA, Bacterial, Staphylococcus aureus, Topoisomerase IV, Cefepime, Microbial Sensitivity Tests, Biochemistry, DNA gyrase, Analytical Chemistry, Minimum inhibitory concentration, chemistry.chemical_compound, Bacterial Proteins, Cell Wall, Drug Discovery, Escherichia coli, medicine, biology, Chloramphenicol, Kanamycin, Anti-Bacterial Agents, RNA, Bacterial, chemistry, DNA Gyrase, biology.protein, Molecular Medicine, Vancomycin, Biological Assay, Tedizolid, Biotechnology, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a345debe45ef8d15b8d1dc6858616212
https://doi.org/10.1177/1087057113487208 -
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المؤلفون: Ken Chen, Adam F. Dukes, Chris Harris, Mark D. Mason, Elizabeth L. Appelbaum, Jennifer Ivanovich, Justin T. Lolofie, Michael D. McLellan, Lei Chen, Benjamin J. Oberkfell, Lisa Cook, Jeremy Hoog, Devin P. Locke, Shunqiang Li, Jennifer S. Hodges, Scott M. Smith, Feiyu Du, Dong-Wei Shen, Amy Hawkins, Gabriel E. Sanderson, Rachel Abbott, Lucinda Fulton, John W. Wallis, Mark A. Watson, Sherri R. Davies, George M. Weinstock, Michelle D O'Laughlin, Richard K. Wilson, Joelle Kalicki, Jacqueline E. Snider, Joshua F. McMichael, Charles M. Perou, Heather K. Schmidt, Nathan D. Dees, Tammi L. Vickery, Jerry S. Reed, Glendoria Elliott, Robert S. Fulton, William Schierding, Li-li Lin, Robert J. Crowder, Timothy J. Ley, James M. Eldred, Josh B. Peck, Craig Pohl, Dominic M. Thompson, David J. Dooling, Paul J. Goodfellow, Michael C. Wendl, Vincent Magrini, Therese Guintoli, Katherine DeSchryver, Li Ding, Kelly E. Bernard, Kim D. Delehaunty, David E. Larson, Qunyuan Zhang, Kimberley A. Pape, Mark L. Cunningham, Matthew J. Ellis, Madeline E. Wiechert, Sean McGrath, Rebecca Aft, Ling Lin, Elaine R. Mardis, Jody S. Robinson, Catrina Fronick, Yu Long Tao, Daniel C. Koboldt
المصدر: Nature
مصطلحات موضوعية: Adult, DNA Copy Number Variations, DNA Mutational Analysis, Transplantation, Heterologous, Breast Neoplasms, Biology, Bioinformatics, medicine.disease_cause, Translocation, Genetic, Article, Metastasis, 03 medical and health sciences, 0302 clinical medicine, Breast cancer, Gene Frequency, medicine, Humans, 030304 developmental biology, 0303 health sciences, Mutation, Multidisciplinary, Brain Neoplasms, Genome, Human, Cancer, Genomics, Cell cycle, medicine.disease, Transplantation, 030220 oncology & carcinogenesis, Disease Progression, Cancer research, Human genome, Female, alpha Catenin, Neoplasm Transplantation, Brain metastasis
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المؤلفون: Victor Nizet, Mark L. Cunningham, Bryan P. Kwan, Wdee Thienphrapa, Kyoung Hwa Jang, Leo Lin, Evaristus Soubih, Nina M. Haste, Dan N. Tran, Mary E. Hensler, William Fenical, Karen Joy Shaw, Lisa Vuong
المصدر: The Journal of antibiotics
The Journal of antibiotics, vol 67, iss 8مصطلحات موضوعية: Methicillin-Resistant Staphylococcus aureus, Staphylococcus aureus, medicine.drug_class, Medicinal & Biomolecular Chemistry, Antibiotics, Microbial Sensitivity Tests, Biology, Peritonitis, medicine.disease_cause, Staphylococcal infections, Microbiology, Article, Anthracimycin, Methicillin, Mice, novel antibiotic, anthracimycin, In vivo, Vancomycin, Drug Discovery, medicine, Animals, Humans, Pharmacology, Molecular Structure, Vancomycin Resistance, Pharmacology and Pharmaceutical Sciences, biochemical phenomena, metabolism, and nutrition, Staphylococcal Infections, medicine.disease, biology.organism_classification, methicillin-resistant, Methicillin-resistant Staphylococcus aureus, 3. Good health, Bacillus anthracis, Anti-Bacterial Agents, Hela Cells, Polyketides, Methicillin Resistance, medicine.drug, HeLa Cells
وصف الملف: application/pdf
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المؤلفون: Mark L. Cunningham, Allen J. Borchardt, Grayson Hough, Mark Hilgers, Bryan P. Kwan, Karen J. Shaw, Jeffrey B. Locke, Sunny Abraham, Gregory Haley, John T. Finn, Min Teng, Courtney Hall
المصدر: Journal of medicinal chemistry. 56(4)
مصطلحات موضوعية: Models, Molecular, Burkholderia, Yersinia pestis, Mutant, Microbial Sensitivity Tests, medicine.disease_cause, Crystallography, X-Ray, Haemophilus influenzae, Substrate Specificity, Structure-Activity Relationship, Bacterial Proteins, Drug Discovery, Drug Resistance, Bacterial, medicine, Escherichia coli, Threonine-tRNA Ligase, Humans, Binding site, Binding Sites, biology, Burkholderia thailandensis, Molecular Structure, Chemistry, Escherichia coli Proteins, Substrate (chemistry), Stereoisomerism, biology.organism_classification, Antimicrobial, Anti-Bacterial Agents, Biochemistry, Mutation, Quinazolines, Molecular Medicine, Bacteria, Protein Binding
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المؤلفون: Mark L. Cunningham, Doug Phillipson, Bryan P. Kwan, John T. Finn, Kirk J. Nelson, Sergio E. Wong, Michael Trzoss, Jeff B. Locke, Jay C. Nix, Vickie Brown-Driver, Felice C. Lightstone, Zhiyong Chen, Toan B. Nguyen, Karen J. Shaw, Suzanne Akers-Rodriguez, Xiaoming Li, Suk Joong Lee, Amanda Castellano, Dean L. Shinabarger, Timothy M. Murphy, Junhu Zhang, Leslie W. Tari, Chris M. Pillar, Voon Ong, Grayson Hough, Thanh Lam, Daniel C. Bensen
المصدر: PLoS ONE, Vol 8, Iss 12, p e84409 (2013)
PLoS ONEمصطلحات موضوعية: DNA Topoisomerase IV, Models, Molecular, Indoles, Protein Conformation, Topoisomerase IV, medicine.drug_class, Antibiotics, lcsh:Medicine, Microbial Sensitivity Tests, DNA gyrase, Microbiology, Mice, chemistry.chemical_compound, Drug Resistance, Bacterial, medicine, Animals, Topoisomerase II Inhibitors, lcsh:Science, Multidisciplinary, Natural product, Bacteria, biology, Topoisomerase, lcsh:R, Anti-Bacterial Agents, Multiple drug resistance, chemistry, DNA Gyrase, Drug Design, biology.protein, Female, lcsh:Q, Topoisomerase-II Inhibitor, Antibacterial activity, Research Article
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المؤلفون: Mark Stidham, Thanh Lam, Bryan P. Kwan, Mark L. Cunningham, Zhiyong Chen, Felice C. Lightstone, Junhu Zhang, Karen J. Shaw, Leslie W. Tari, Toan B. Nguyen, Christopher J. Creighton, John T. Finn, Xiaoming Li, Michael Trzoss, Daniel C. Bensen, Sergio E. Wong, Jay C. Nix
المصدر: Bioorganicmedicinal chemistry letters. 23(5)
مصطلحات موضوعية: DNA Topoisomerase IV, Models, Molecular, Dual targeting, Topoisomerase IV, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, DNA gyrase, Broad spectrum, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Topoisomerase II Inhibitors, Pyrroles, Molecular Biology, chemistry.chemical_classification, biology, Chemistry, Topoisomerase, Organic Chemistry, biochemical phenomena, metabolism, and nutrition, Anti-Bacterial Agents, Enzyme, Pyrimidines, DNA Gyrase, Drug Design, biology.protein, Molecular Medicine, Pharmacophore, DNA
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المؤلفون: Vickie Brown-Driver, Christopher J. Creighton, John T. Finn, Toan B. Nguyen, Mark L. Cunningham, Zhiyong Chen, Amanda Castellano, Mark Stidham, Sergio E. Wong, Xiaoming Li, Karen J. Shaw, Thanh Lam, Junhu Zhang, Bryan P. Kwan, Kirk J. Nelson, Felice C. Lightstone, Leslie W. Tari, Daniel C. Bensen, Micheal Trzoss
المصدر: Bioorganicmedicinal chemistry letters. 23(5)
مصطلحات موضوعية: DNA Topoisomerase IV, Topoisomerase IV, Clinical Biochemistry, Pharmaceutical Science, medicine.disease_cause, Biochemistry, DNA gyrase, Microbiology, Structure-Activity Relationship, Drug Discovery, medicine, Structure–activity relationship, Humans, Topoisomerase II Inhibitors, Pyrroles, Molecular Biology, Escherichia coli, biology, Pseudomonas aeruginosa, Chemistry, Topoisomerase, Organic Chemistry, biochemical phenomena, metabolism, and nutrition, biology.organism_classification, Acinetobacter baumannii, Anti-Bacterial Agents, Pyrimidines, DNA Gyrase, Drug Design, biology.protein, bacteria, Molecular Medicine, Antibacterial activity