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المؤلفون: Mark P. Grillo
المصدر: Transporters and Drug-Metabolizing Enzymes in Drug Toxicity
مصطلحات موضوعية: chemistry.chemical_classification, Acyl-CoA formation, chemistry.chemical_compound, Transacylation, Chemistry, Stereochemistry, Carboxylic acid, Acyl glucuronidation, Covalent binding, Glutathione, Potential toxicity
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::7de6b2ee3dd362ab9e2042d5906c1de8
https://doi.org/10.1002/9781119171003.ch6 -
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المؤلفون: Mark P. Grillo, Svetlana Markova, Marc Evanchik, Marc Trellu, Patricia Moliner, Priscilla Brun, Anne Perreard-Dumaine, Pascale Vicat, Chun Yang, James P. Driscoll, Tim J. Carlson
المصدر: Xenobiotica. 51:222-238
مصطلحات موضوعية: medicine.medical_specialty, Health, Toxicology and Mutagenesis, Toxicology, Left ventricular enlargement, 030226 pharmacology & pharmacy, Biochemistry, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, In vivo, Internal medicine, Myosin, medicine, cardiovascular diseases, Pharmacology, business.industry, Activator (genetics), Dilated cardiomyopathy, General Medicine, medicine.disease, In vitro, 030220 oncology & carcinogenesis, Heart failure, cardiovascular system, Cardiology, business
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3
المؤلفون: Mark P, Grillo, Svetlana, Markova, Marc, Evanchik, Marc, Trellu, Patricia, Moliner, Priscilla, Brun, Anne, Perreard-Dumaine, Pascale, Vicat, James P, Driscoll, Tim J, Carlson
المصدر: Xenobiotica; the fate of foreign compounds in biological systems. 51(2)
مصطلحات موضوعية: Cardiomyopathy, Dilated, Male, Mice, Dogs, Hepatocytes, Microsomes, Liver, Animals, Biological Availability, Humans, Caco-2 Cells, Myosins, Protein Binding, Rats
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4
المؤلفون: Marc J. Evanchik, Priscilla Brun, John C L Erve, Nicole V Haste, Mark P. Grillo, Svetlana Markova, Ryan Dick, Timothy J. Carlson, James P Driscoll
المصدر: Xenobiotica; the fate of foreign compounds in biological systems. 49(6)
مصطلحات موضوعية: Male, Benzylamines, Allosteric modulator, Metabolic Clearance Rate, Health, Toxicology and Mutagenesis, Pharmacology, Toxicology, 030226 pharmacology & pharmacy, Biochemistry, Rats, Sprague-Dawley, 03 medical and health sciences, 0302 clinical medicine, Dogs, Pharmacokinetics, Cytochrome P-450 Enzyme System, In vivo, medicine, Animals, Humans, Drug Interactions, Beta (finance), Uracil, Mice, Inbred ICR, Chemistry, Hypertrophic cardiomyopathy, General Medicine, Cardiomyopathy, Hypertrophic, medicine.disease, Small molecule, In vitro, Macaca fascicularis, 030220 oncology & carcinogenesis, Hepatocytes, Microsomes, Liver, Caco-2 Cells, Cardiac Myosins, Drug metabolism
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5
المؤلفون: Mark P. Grillo
المصدر: Expert Opinion on Drug Metabolism & Toxicology. 11:1281-1302
مصطلحات موضوعية: Drug, Magnetic Resonance Spectroscopy, Drug-Related Side Effects and Adverse Reactions, media_common.quotation_subject, Reactive intermediate, Pharmacology, Toxicology, medicine.disease_cause, Pharmacokinetics, Tandem Mass Spectrometry, medicine, Animals, Humans, media_common, Drug discovery, Chemistry, DNA, General Medicine, In vitro, Pharmaceutical Preparations, Drug Design, Toxicity, Carcinogenesis, Drug metabolism, Chromatography, Liquid, Protein Binding
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6
المؤلفون: Karen Siegler, Bei Shan, Mark P. Grillo, Marion Conn, Jiang Zhu, Jian Ken Zhang, Yingcai Wang, Julio C. Medina, Ming Yu, Peter Coward, Frank Kayser, Jiwen Jim Liu
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:156-160
مصطلحات موضوعية: Agonist, Sulfonamides, Dose-Response Relationship, Drug, Molecular Structure, Pyridines, medicine.drug_class, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Rats, Receptors, G-Protein-Coupled, Structure-Activity Relationship, GPR119, Drug Discovery, Microsomes, Liver, medicine, Animals, Humans, Molecular Medicine, Molecule, Molecular Biology
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7
المؤلفون: Pierre Deprez, Paul M. Wehn, Jeff D. Reagan, Minghan Wang, Paul E. Harrington, Mark P. Grillo, Kanaka Pattabiraman, James Davis, Charles Henley, Sean Morony, Taoues Temal, Christopher H. Fotsch, Steve F. Poon, Timothy J. Carlson, David J. St. Jean, Sarah E. Lively, Yuhua Yang, Jenny Ying-Lin Lu
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:6625-6628
مصطلحات موضوعية: Male, Calcimimetic, Metabolite, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Rats, Sprague-Dawley, chemistry.chemical_compound, Pharmacokinetics, In vivo, Drug Discovery, medicine, Animals, Urea, Potency, Molecular Biology, CYP3A4, Organic Chemistry, medicine.disease, Rats, Bioavailability, Thiazoles, chemistry, Parathyroid Hormone, Molecular Medicine, Hyperparathyroidism, Secondary, Secondary hyperparathyroidism, Receptors, Calcium-Sensing, Half-Life, Protein Binding
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8
المؤلفون: Mark P. Grillo, Michelle Tadano Lohr, Smriti Khera
المصدر: Drug Metabolism and Disposition. 41:111-121
مصطلحات موضوعية: Dipeptidase, Magnetic Resonance Spectroscopy, Stereochemistry, Pharmaceutical Science, Ibuprofen, In Vitro Techniques, Thioester, chemistry.chemical_compound, Tandem Mass Spectrometry, In vivo, Animals, Humans, Mercapturic acid, Pharmacology, chemistry.chemical_classification, Chromatography, biology, organic chemicals, gamma-Glutamyltransferase, Glutathione, In vitro, Enzyme, chemistry, Glycine, biology.protein, Cattle, Chromatography, Liquid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4a002dec87f47888e712a348a43ea541
https://doi.org/10.1124/dmd.112.048645 -
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المؤلفون: Mark P. Grillo, Michelle Tadano Lohr, Jill C. M. Wait
المصدر: Drug Metabolism and Disposition. 40:1515-1526
مصطلحات موضوعية: Mefenamic acid, Carboxylic acid, Acyl glucuronidation, Pharmaceutical Science, In Vitro Techniques, Thioester, Mefenamic Acid, chemistry.chemical_compound, Tandem Mass Spectrometry, In vivo, medicine, Animals, Humans, Biotransformation, Pharmacology, chemistry.chemical_classification, Chemistry, Metabolism, Glutathione, Rats, Biochemistry, Hepatocytes, Glucuronide, Chromatography, Liquid, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cde80e7dbf2a7269556d1b58e97c1f36
https://doi.org/10.1124/dmd.112.046102 -
10
المؤلفون: Mark P. Grillo, Jessica S. Houghton, Eskouhie Tchaparian, Craig Uyeda, Lixia Jin
المصدر: Drug Metabolism and Disposition. 39:2387-2394
مصطلحات موضوعية: Male, Pharmacology, Abcg2, Organic anion transporter 1, Reverse Transcriptase Polymerase Chain Reaction, Multidrug resistance-associated protein 2, Pharmaceutical Science, Transporter, Articles, Biology, Molecular biology, In vitro, Rats, Rats, Sprague-Dawley, Pharmaceutical Preparations, In vivo, Cell culture, Gene expression, Hepatocytes, biology.protein, Animals, Carrier Proteins, Cells, Cultured
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ddb10b8849cc9c354476165ec83df0bf
https://doi.org/10.1124/dmd.111.039545