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1دورية أكاديمية
المؤلفون: Fernando A. Batista, Soraya S. Bosch, Sabine Butzloff, Sergey Lunev, Kamila A. Meissner, Marleen Linzke, Atilio R. Romero, Chao Wang, Ingrid B. Müller, Alexander S. S. Dömling, Matthew R. Groves, Carsten Wrenger
المصدر: MicrobiologyOpen, Vol 8, Iss 7, Pp n/a-n/a (2019)
مصطلحات موضوعية: drug target validation, oligomeric state, phenotypic mapping, Plasmodium falciparum, structural biology, Microbiology, QR1-502
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2045-8827
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2دورية أكاديمية
المؤلفون: Sergey Lunev, Sabine Butzloff, Atilio R Romero, Marleen Linzke, Fernando A Batista, Kamila A Meissner, Ingrid B Müller, Alaa Adawy, Carsten Wrenger, Matthew R Groves
المصدر: PLoS ONE, Vol 13, Iss 4, p e0195011 (2018)
وصف الملف: electronic resource
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المؤلفون: Soraya S Bosch, Fernando de Assis Batista, Alexander Dömling, Sergey Lunev, Thales Kronenberger, Matthew Groves, Marleen Linzke, Carsten Wrenger
المساهمون: Drug Design, Medicinal Chemistry and Bioanalysis (MCB)
المصدر: ACS Infectious Diseases, 6(5), 986-999. TAYLOR & FRANCIS LTD
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USPمصطلحات موضوعية: 0301 basic medicine, chemistry.chemical_classification, biology, ANIMAIS PARASITOS, Transgene, 030106 microbiology, Mutant, Plasmodium falciparum, biology.organism_classification, In vitro, 3. Good health, 03 medical and health sciences, Aspartate carbamoyltransferase, 030104 developmental biology, Infectious Diseases, Enzyme, chemistry, Biochemistry, Cell culture, Pyrimidine metabolism
وصف الملف: application/vnd.openxmlformats-officedocument.wordprocessingml.document
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المؤلفون: Henning Ulrich, Attila Tárnok, Marleen Linzke, Matthew Groves, Sun Liu Rei Yan, Carsten Wrenger
المصدر: Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USPمصطلحات موضوعية: 0301 basic medicine, Histology, Aptamer, SUBCELLULAR COMPARTMENTS, Plasmodium falciparum, ENDOPLASMIC-RETICULUM, MICROSCOPIA DE FLUORESCÊNCIA, ACRIDINE-ORANGE, Computational biology, GFP, Plasmodium, Pathology and Forensic Medicine, RED-BLOOD-CELLS, 03 medical and health sciences, 0302 clinical medicine, Live cell imaging, PARASITOPHOROUS VACUOLE, parasitic diseases, medicine, Animals, Humans, Parasite hosting, Parasites, GREEN FLUORESCENT PROTEIN, OXIDATIVE STRESS, Dyes, Cellular compartment, Staining, Life Cycle Stages, biology, INFECTED ERYTHROCYTES, Cell Biology, Flow Cytometry, biology.organism_classification, medicine.disease, Protozoan parasite, Malaria, 030104 developmental biology, FLOW-CYTOMETRIC ENUMERATION, 030220 oncology & carcinogenesis, THIAZOLE ORANGE, Cytometry
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المؤلفون: Marleen Linzke
المساهمون: Dömling, Alex, Wrenger, Carsten, Groves, Matthew, Drug Design
مصطلحات موضوعية: Drug, Apicoplast, media_common.quotation_subject, Plasmodium falciparum, Disease, Drug resistance, Biology, biology.organism_classification, medicine.disease, Virology, Plasmodium, medicine, Parasite hosting, Malaria, media_common
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7e3fd2e39db0002f45a9a13b7b3f3656
https://doi.org/10.33612/diss.107482905 -
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المؤلفون: Alexander Dömling, Fernando de Assis Batista, Matthew Groves, George Chamoun, Carsten Wrenger, Soraya S Bosch, Chao Wang, Paul D Kruithof, Jingyao Li, Sergey Lunev, Marleen Linzke
المساهمون: Drug Design, Medicinal Chemistry and Bioanalysis (MCB)
المصدر: Biochemical and Biophysical Research Communications, 497(3), 835-842. ACADEMIC PRESS INC ELSEVIER SCIENCE
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USPمصطلحات موضوعية: 0301 basic medicine, Plasmodium falciparum, Allosteric regulation, Biophysics, Crystallography, X-Ray, Biochemistry, 03 medical and health sciences, Non-competitive inhibition, Catalytic Domain, Drug Discovery, Aspartate Carbamoyltransferase, Journal Article, Humans, Enzyme Inhibitors, Malaria, Falciparum, MALÁRIA, Molecular Biology, Antiparasitic Agents, 030102 biochemistry & molecular biology, biology, Drug discovery, Chemistry, Active site, Cell Biology, biology.organism_classification, Antiparasitic agent, Molecular Docking Simulation, Aspartate carbamoyltransferase, 030104 developmental biology, Pyrimidine metabolism, biology.protein
وصف الملف: application/pdf
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المؤلفون: Atilio Reyes Romero, Carsten Wrenger, Sergey Lunev, Chao Wang, Marleen Linzke, Soraya S Bosch, Sabine Butzloff, Kamila Anna Meissner, Alexander Dömling, Fernando de Assis Batista, Matthew Groves, Ingrid B. Müller
المساهمون: Drug Design, Medicinal Chemistry and Bioanalysis (MCB)
المصدر: MicrobiologyOpen
MicrobiologyOpen, 8(7):e779. Wiley
MicrobiologyOpen, Vol 8, Iss 7, Pp n/a-n/a (2019)
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USPمصطلحات موضوعية: AMINOTRANSFERASE, Plasmodium falciparum, Mutant, lcsh:QR1-502, Druggability, PURINE, Computational biology, Biology, METABOLISM, Microbiology, lcsh:Microbiology, MECHANISMS, 03 medical and health sciences, 0302 clinical medicine, In vivo, structural biology, Gene, 030304 developmental biology, chemistry.chemical_classification, 0303 health sciences, oligomeric state, Original Articles, ANTIMALÁRICOS, biology.organism_classification, GENE, 3. Good health, Enzyme, chemistry, Structural biology, phenotypic mapping, Original Article, drug target validation, 030217 neurology & neurosurgery, Function (biology), INTERFACES
وصف الملف: application/pdf
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المؤلفون: Matthew Groves, Marleen Linzke, Carsten Wrenger, Yuanze Wang, Kamila Anna Meissner, Sergey Lunev, Fernando de Assis Batista
المساهمون: Drug Design, Medicinal Chemistry and Bioanalysis (MCB)
المصدر: CURRENT DRUG TARGETS, 18(9), 1069-1085. BENTHAM SCIENCE PUBL LTD
مصطلحات موضوعية: 0301 basic medicine, Plasmodium falciparum, Clinical Biochemistry, Druggability, Computational biology, Biology, Bioinformatics, Protein–protein interaction, Antimalarials, 03 medical and health sciences, Drug Delivery Systems, Protein structure, In vivo, Drug Discovery, Humans, Crossing Over, Genetic, Malaria, Falciparum, Pharmacology, Drug discovery, Proteins, Small molecule, 030104 developmental biology, Gene Knockdown Techniques, Molecular Medicine, Target protein, Function (biology)
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8c647bd33932f9bb528140b7a62e20cf
https://doi.org/10.2174/1389450117666160201115003 -
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المؤلفون: Sabine Butzloff, Atilio Reyes Romero, Alaa Adawy, Carsten Wrenger, Fernando de Assis Batista, Matthew Groves, Kamila Anna Meissner, Sergey Lunev, Marleen Linzke, Ingrid B. Müller
المساهمون: Drug Design, Medicinal Chemistry and Bioanalysis (MCB)
المصدر: 'PloS One ', vol: 13, pages: e0195011-1-e0195011-22 (2018)
PLOS ONE 13(4), e0195011-(2018). doi:10.1371/journal.pone.0195011
PLoS ONE, 13(4). PUBLIC LIBRARY SCIENCE
PLoS ONE, Vol 13, Iss 4, p e0195011 (2018)
PLOS ONE
PLoS ONE
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USPمصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Light, Mutant, Molecular Conformation, Thermal Stability, Druggability, Gene Expression, lcsh:Medicine, Plasma protein binding, Biochemistry, Substrate Specificity, Scattering, Malate Dehydrogenase, Drug Discovery, Medicine and Health Sciences, MALÁRIA, lcsh:Science, Conserved Sequence, Crystallography, Multidisciplinary, biology, Chemistry, Drug discovery, Physics, Electromagnetic Radiation, Condensed Matter Physics, Recombinant Proteins, 3. Good health, Physical Sciences, Crystal Structure, Thermodynamics, Protein Binding, Research Article, Drug Research and Development, Chemical physics, Plasmodium falciparum, Malate dehydrogenase, Antimalarials, 03 medical and health sciences, In vivo, Genetics, Parasitic Diseases, Humans, Point Mutation, Solid State Physics, Amino Acid Sequence, ddc:610, Pharmacology, Binding Sites, lcsh:R, Light Scattering, Wild type, Biology and Life Sciences, Proteins, Dimers (Chemical physics), Tropical Diseases, biology.organism_classification, Malaria, 030104 developmental biology, Mutation, lcsh:Q
وصف الملف: application/pdf