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المؤلفون: Ning Qin, Michael F.A. Finley, Christopher M. Flores, Michael P. Neeper, Michael P. Winters, Michael R. Brandt, Wall Mark, Nalin L. Subasinghe, Raymond W. Colburn, Zhihua Sui, Craig R. Schneider, Mary Lou Lubin
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:3780-3783
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Calcium channel, Organic Chemistry, Clinical Biochemistry, Patch clamp electrophysiology, Cell, Pharmaceutical Science, Pharmacology, N-type calcium channel, 010402 general chemistry, 01 natural sciences, Biochemistry, 0104 chemical sciences, medicine.anatomical_structure, Drug Discovery, Neuropathic pain, medicine, Molecular Medicine, Molecular Biology, Calcium influx
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المؤلفون: Mark J, Wall, Nalin L, Subasinghe, Michael P, Winters, Mary Lou, Lubin, Michael F A, Finley, Ning, Qin, Michael R, Brandt, Michael P, Neeper, Craig R, Schneider, Raymond W, Colburn, Christopher M, Flores, Zhihua, Sui
المصدر: Bioorganicmedicinal chemistry letters. 28(23-24)
مصطلحات موضوعية: Male, Analgesics, Patch-Clamp Techniques, Calcium Channel Blockers, Rats, Rats, Sprague-Dawley, Calcium Channels, N-Type, HEK293 Cells, Drug Discovery, Animals, Humans, Neuralgia, Pyrazoles, Calcium, Pyrans
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3
المؤلفون: Scott L. Dax, Mingde Xia, Dennis J. Stone, Xiaoqing Xu, Bin Zhu, Donald William Ludovici, Matthews Jay M, Mark A. Youngman, Tasha L. Hutchinson, Michael R. Brandt, Christopher M. Flores, Mary Lou Lubin, Mark J. Macielag, Raymond W. Colburn, Ning Qin, Manomi A. Tennakoon
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:2234-2237
مصطلحات موضوعية: Clinical Biochemistry, Cell, Glycine, TRPM Cation Channels, Pharmaceutical Science, Stereoisomerism, Pyrimidinones, Pharmacology, Biochemistry, Structure-Activity Relationship, Transient receptor potential channel, In vivo, Drug Discovery, TRPM8, medicine, Animals, Humans, Structure–activity relationship, Molecular Biology, Behavior, Animal, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, In vitro, Rats, HEK293 Cells, medicine.anatomical_structure, Molecular Medicine, Antagonism
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المؤلفون: Michael R. Brandt, Michael F.A. Finley, Ning Qin, Michael P. Winters, Craig R. Schneider, Mary Lou Lubin, Michael P. Neeper, Nalin L. Subasinghe, Zhihua Sui, Raymond W. Colburn, Christopher M. Flores, Wall Mark
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:4080-4083
مصطلحات موضوعية: Patch-Clamp Techniques, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, N-type calcium channel, Biochemistry, omega-Conotoxins, Cell Line, Structure-Activity Relationship, Calcium Channels, N-Type, Piperidines, In vivo, Drug Discovery, medicine, Animals, Humans, Potency, Molecular Biology, Analgesics, Ziconotide, Chemistry, Calcium channel, Organic Chemistry, Chronic pain, Metabolic stability, Calcium Channel Blockers, medicine.disease, High-Throughput Screening Assays, Rats, Neuropathic pain, Neuralgia, Pyrazoles, Molecular Medicine, Chronic Pain, medicine.drug
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المؤلفون: Shelley K. Ballentine, Mark R. Player, Mary Lou Lubin, Raul R. Calvo, Craig R. Schneider, William H. Parsons, Raymond W. Colburn, Parks Daniel J, Sanath K. Meegalla, Christopher M. Flores
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:1903-1907
مصطلحات موضوعية: Benzimidazole, Clinical Biochemistry, TRPM Cation Channels, Pharmaceutical Science, Pharmacology, Biochemistry, chemistry.chemical_compound, Transient receptor potential channel, Dogs, In vivo, Drug Discovery, TRPM8, medicine, Animals, Humans, Molecular Biology, Ion channel, Analgesics, Organic Chemistry, Rats, Cold Temperature, HEK293 Cells, Allodynia, chemistry, Hyperalgesia, Cold Hypersensitivity, Neuropathic pain, Neuralgia, Molecular Medicine, Benzimidazoles, medicine.symptom
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المؤلفون: Yi Liu, Michael F.A. Finley, Mary Lou Lubin, Ning Qin, Michael P. Neeper, Christopher M. Flores, Edward J. Beck
المصدر: ASSAY and Drug Development Technologies. 8:685-694
مصطلحات موضوعية: Patch-Clamp Techniques, Calcitonin Gene-Related Peptide, Presynaptic Terminals, Pain, Pharmacology, omega-Conotoxins, Cell Line, Small Molecule Libraries, Calcium Channels, N-Type, Dorsal root ganglion, Ganglia, Spinal, Drug Discovery, Calcium flux, medicine, Animals, Humans, Patch clamp, Ion channel, Neurons, Analgesics, Ziconotide, Voltage-dependent calcium channel, Chemistry, Calcium channel, Calcium Channel Blockers, High-Throughput Screening Assays, Rats, Electrophysiology, HEK293 Cells, medicine.anatomical_structure, Spinal Cord, Luminescent Measurements, Molecular Medicine, Neuroscience, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::021e926842b8366d4a8742a010cc48f2
https://doi.org/10.1089/adt.2010.0311 -
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المؤلفون: Mary Lou Lubin, Danielle Lawrence, Ning Qin, Yi Liu, Michael R. D'Andrea, Michael R. Brandt, Dennis J. Stone, Yan Wang, Christopher M. Flores, Raymond W. Colburn
المصدر: Neuron. 54(3):379-386
مصطلحات موضوعية: Chemistry, General Neuroscience, Neuroscience(all), Icilin, Sensory system, In vitro, Cell biology, chemistry.chemical_compound, Transient receptor potential channel, In vivo, medicine, TRPM8, Cold sensitivity, medicine.symptom, SYSNEURO, Ion channel
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المؤلفون: Ellen E. Codd, Ning Qin, Navid Shafaee, Mary-Lou Lubin, Michael R. D'Andrea, Ana M. Correa
المصدر: European Journal of Biochemistry. 270:4762-4770
مصطلحات موضوعية: SCN3A, Open reading frame, Protein subunit, Specificity factor, Interleukin 5 receptor alpha subunit, RNA splicing, Biology, Biochemistry, Molecular biology, Gamma-aminobutyric acid receptor subunit alpha-1, Interleukin 10 receptor, alpha subunit
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9
المؤلفون: Ning Qin, Mary Lou Lubin, Michael R. Brandt, Edward J. Beck, Zhihua Sui, Christopher M. Flores, Michael P. Winters, Yi Liu, Michael P. Neeper, Michael F.A. Finley, Wall Mark, Nalin L. Subasinghe
المصدر: Bioorganicmedicinal chemistry letters. 24(9)
مصطلحات موضوعية: Chemistry, Stereochemistry, Calcium channel, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, N-type calcium channel, Calcium Channel Blockers, Biochemistry, Rats, Structure-Activity Relationship, Calcium Channels, N-Type, Drug Discovery, Microsomes, Liver, Molecular Medicine, Animals, Humans, Pyrazoles, Chronic Pain, Molecular Biology
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المؤلفون: Yi Liu, Mary Lou Lubin, Christopher M. Flores, Michael P. Winters, Michael F.A. Finley, Wall Mark, Ning Qin, Nalin L. Subasinghe, Michael R. Brandt, Michael P. Neeper, Zhihua Sui, Edward J. Beck
المصدر: Bioorganicmedicinal chemistry letters. 24(9)
مصطلحات موضوعية: Analgesics, Series (mathematics), Chemistry, Stereochemistry, Calcium channel, Organic Chemistry, Clinical Biochemistry, Chronic pain, Pharmaceutical Science, Pain, N-type calcium channel, medicine.disease, Calcium Channel Blockers, Biochemistry, Combinatorial chemistry, Rats, Calcium Channels, N-Type, In vivo, Drug Discovery, medicine, Microsomes, Liver, Molecular Medicine, Animals, Pyrazoles, Molecular Biology