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1دورية أكاديمية
المؤلفون: Becker, Michael R., Ewing, William R., Davis, Roderick S., Pauls, Henry W., Ly, Cuong, Li, Aiwen, Mason, Helen J., Choi-Sledeski, Yong Mi, Spada, Alfred P., Chu, Valeria, Brown, Karen D., Colussi, Dennis J., Leadley, Robert J., Bentley, Ross, Bostwick, Jeff, Kasiewski, Charles, Morgan, Suzanne
المصدر: In Bioorganic & Medicinal Chemistry Letters 1999 9(18):2753-2758
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2دورية أكاديمية
المؤلفون: Roberts, Lee R., Corbett, Matthew S., Fussell, Steven J., Hitzel, Laure, Jessiman, Alan S., Mason, Helen J., Osborne, Rachel, Ralph, Michael J., Stennett, Adam S.D., Wheeler, Simon, Storer, R. Ian
المصدر: In Tetrahedron Letters 25 November 2015 56(47):6546-6550
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3
المؤلفون: Mason Helen J, Karen D. Brown, Valeria Chu, Guyan Liang, Daniel M. Green, Alfred P. Spada, Henry W. Pauls, Ross Bentley, Cuong Ly, Roderick S. Davis, Dennis J. Colussi, Daniel L. Cheney, Michael R. Becker, Y.M. Choi-Sledeski, Christopher T. Dunwiddie, Robert J. Leadley, Ewing William R, John H. Barton
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:2539-2544
مصطلحات موضوعية: Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, Isostere, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Administration, Oral, Pharmaceutical Science, Biochemistry, Chemical synthesis, Benzamidine, Amidine, Serine, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Drug Discovery, medicine, Animals, Structure–activity relationship, Molecular Biology, Binding Sites, Organic Chemistry, Isoquinolines, Benzamidines, chemistry, Molecular Medicine, Factor Xa Inhibitors
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4
المؤلفون: Alfred P. Spada, Robert J. Leadley, Jonathan S. Mason, Dennis J. Colussi, Ewing William R, Mark H. Perrone, Karen D. Brown, Michael R. Becker, Don D. Cha, Daniel M. Green, Ross Bentley, Henry W. Pauls, Christopher T. Dunwiddie, Jean-Pierre Guilloteau, Y.M. Choi-Sledeski, Sebastien Maignan, Mason Helen J, Vincent E. Manetta, Charles Kasiewski, Valeria Chu, Roderick S. Davis, Suzanne Morgan, Daniel L. Cheney, Jeff Bostwick
المصدر: Journal of Medicinal Chemistry. 42:3557-3571
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, medicine.drug_class, Factor Xa Inhibitor, Thiophenes, Crystallography, X-Ray, Amidine, Structure-Activity Relationship, chemistry.chemical_compound, Thrombin, In vivo, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Sulfonamides, Molecular Structure, biology, Chemistry, Anticoagulant, Anticoagulants, Stereoisomerism, Thrombosis, Trypsin, Pyrrolidinones, Rats, Biochemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Rabbits, Factor Xa Inhibitors, medicine.drug
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5دورية أكاديمية
المؤلفون: Johnson, Patrick S., Ryckmans, Thomas, Bryans, Justin, Beal, Dave M., Dack, Kevin N., Feeder, Neil, Harrison, Anthony, Lewis, Mark, Mason, Helen J., Mills, James, Newman, Julie, Pasquinet, Christelle, Rawson, Dave J., Roberts, Lee R., Russell, Rachel, Spark, Deborah, Stobie, Alan, Underwood, Toby J., Ward, Robin, Wheeler, Simon
المصدر: In Bioorganic & Medicinal Chemistry Letters 2011 21(19):5684-5687
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6دورية أكاديمية
المؤلفون: Watson, Christine, Owen, Dafydd R., Harding, Denise, Kon-I, Kana, Lewis, Mark L., Mason, Helen J., Matsumizu, Miyako, Mukaiyama, Takasuke, Rodriguez-Lens, Margarita, Shima, Akiko, Takeuchi, Mifune, Tran, Isabelle, Young, Tim
المصدر: In Bioorganic & Medicinal Chemistry Letters 2011 21(14):4284-4287
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7دورية أكاديمية
المؤلفون: Pryde, David C., Jones, Rhys, Middleton, Donald S., Laverty, Ben J., Fenwick, David R., Mason, Helen J., Corless, Martin, Smith, Nick N.
المصدر: In Bioorganic & Medicinal Chemistry Letters 15 November 2010 20(22):6400-6404
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8
المؤلفون: Orton E, Jane Kline, Amy Dodd, Gerald McGeehan, Mathew Morrisette, Christopher J. Burns, Mason Helen J, Salvino Joseph M, Richard Labaudininiere, Groneberg Robert D, Terence Kiesow, Rose Mathew, Sheng-Yuh Tang, Ramesh Narensingh
المصدر: Bioorganicmedicinal chemistry letters. 10(15)
مصطلحات موضوعية: Hydroxamic acid, Screening test, Chemistry, Organic Chemistry, Clinical Biochemistry, Phosphoric Diester Hydrolases, Pharmaceutical Science, Matrix Metalloproteinase Inhibitors, Hydroxamic Acids, Biochemistry, Combinatorial chemistry, Chemical synthesis, Cyclic Nucleotide Phosphodiesterases, Type 4, chemistry.chemical_compound, Structure-Activity Relationship, Solid-phase synthesis, 3',5'-Cyclic-AMP Phosphodiesterases, Drug Discovery, Molecular Medicine, Organic chemistry, Sulfones, Enzyme Inhibitors, Molecular Biology
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9دورية أكاديمية
المؤلفون: Pryde, David C., Corless, Martin, Fenwick, David R., Mason, Helen J., Stammen, Blanda C., Stephenson, Peter T., Ellis, David, Bachelor, David, Gordon, David, Barber, Christopher G., Wood, Anthony, Middleton, Donald S., Blakemore, David C., Parsons, Gemma C., Eastwood, Rachel, Platts, Michelle Y., Statham, Keith, Paradowski, Kerry A., Burt, Catherine, Klute, Wolfgang
المصدر: In Bioorganic & Medicinal Chemistry Letters 2009 19(4):1084-1088
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10
المؤلفون: Charles Kasiewski, Suzanne Morgan, Roderick S. Davis, Robert J. Leadley, Jeff Bostwick, Valeria Chu, Henry W. Pauls, Ewing William R, Karen D. Brown, Cuong Ly, Michael R. Becker, Mason Helen J, Ross Bentley, Y.M. Choi-Sledeski, Dennis J. Colussi, Alfred P. Spada, Aiwen Li
المصدر: Bioorganicmedicinal chemistry letters. 9(18)
مصطلحات موضوعية: Thienopyridine, medicine.drug_mechanism_of_action, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Pharmaceutical Science, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Dogs, In vivo, Drug Discovery, medicine, Structure–activity relationship, Animals, Pyrrolidinones, Molecular Biology, chemistry.chemical_classification, biology, Organic Chemistry, Thrombosis, Sulfonamide, Rats, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Factor Xa Inhibitors