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1دورية أكاديمية
المؤلفون: Benjamin M. Vincent, Daniel F. Tardiff, Jeff S. Piotrowski, Rebecca Aron, Matthew C. Lucas, Chee Yeun Chung, Helene Bacherman, YiQun Chen, Michelle Pires, Radha Subramaniam, Dimple B. Doshi, Heather Sadlish, Waseem K. Raja, Eric J. Solís, Vikram Khurana, Bertrand Le Bourdonnec, Robert H. Scannevin, Kenneth J. Rhodes
المصدر: Cell Reports, Vol 25, Iss 10, Pp 2742-2754.e31 (2018)
مصطلحات موضوعية: Biology (General), QH301-705.5
وصف الملف: electronic resource
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2
المؤلفون: Matthew C. Lucas, Melinda S. Merchant, Matthew O'Connor, Carl Cook, Sherri Smith, Anthony Trombino, Wu-Yan Zhang, Irache Visiers, Kate Tith, Reza Foroughi, Nigel Waters, Iwona Wrona, Michael Pickard, Sudharshan Eathiraj, Karsten Witt, Christopher Roberts, Rachel Humphrey, Elizabeth Buck
المصدر: Molecular Cancer Therapeutics. 20:P02-04
مصطلحات موضوعية: Cancer Research, Oncology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ae653c049d0da4a11d8de415f56e2dfa
https://doi.org/10.1158/1535-7163.targ-21-p02-04 -
3
المؤلفون: Etienne Dardenne, Noboru Ishiyama, Tai-An Lin, Matthew C Lucas
المصدر: Bioorganic & Medicinal Chemistry. 87:117275
مصطلحات موضوعية: Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Molecular Biology, Biochemistry
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4
المؤلفون: Iwona Wrona, Matthew C. Lucas
المصدر: Medicinal Chemistry Reviews ISBN: 9780996293235
Medicinal Chemistry Reviewsمصطلحات موضوعية: chemistry.chemical_classification, Transient receptor potential channel, chemistry, Ankyrin, Biology, Cell biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::53a471c0b79f39633b625539d1decf78
https://doi.org/10.29200/acsmedchemrev-v51.ch8 -
5
المؤلفون: Heather Sadlish, Matthew C. Lucas, Vikram Khurana, Kenneth J. Rhodes, Waseem K. Raja, Yiqun Chen, Rebecca Aron, Daniel F. Tardiff, Radha Subramaniam, Bertrand Le Bourdonnec, Eric Solis, Dimple B. Doshi, Jeff S. Piotrowski, Benjamin Vincent, Chee Yeun Chung, Michelle Pires, Helene Bacherman, Robert H. Scannevin
المصدر: Cell Reports, Vol 25, Iss 10, Pp 2742-2754.e31 (2018)
مصطلحات موضوعية: 0301 basic medicine, Parkinson's disease, Phenotypic screening, Saccharomyces cerevisiae, Pharmacology, General Biochemistry, Genetics and Molecular Biology, Protein Aggregates, 03 medical and health sciences, 0302 clinical medicine, medicine, Animals, Humans, Cytotoxicity, Induced pluripotent stem cell, lcsh:QH301-705.5, Triglycerides, Neurons, Synucleinopathies, Oxadiazoles, Chemistry, Fatty Acids, Lipid Metabolism, medicine.disease, Rats, Stearoyl-CoA Desaturase, 030104 developmental biology, lcsh:Biology (General), Cytoprotection, Toxicity, alpha-Synuclein, Chemical genetics, 030217 neurology & neurosurgery
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6
المصدر: Pharmacology & Therapeutics. 138:294-309
مصطلحات موضوعية: Pharmacology, Innate immune system, Syk, hemic and immune systems, chemical and pharmacologic phenomena, Biology, medicine.disease_cause, Autoimmunity, Immune system, immune system diseases, hemic and lymphatic diseases, Immunology, Cancer research, biology.protein, medicine, Bruton's tyrosine kinase, Pharmacology (medical), Refractory Chronic Lymphocytic Leukemia, Tyrosine kinase, PI3K/AKT/mTOR pathway
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المؤلفون: Yonglin Ren, Ryan Craig Schoenfeld, Adrian J. Fretland, Maria E. Fuentes, Kung-Ching Chang, Yimin Qian, Rachid Hamid, Yun Chen, Achyutharao Sidduri, Matthew Michael Hamilton, Christopher S. Stevenson, Gabriel Stephen Deems, Lin Zhang, Terry Truitt, Dramane Ibrahim Laine, Arjun Narayanan, Ruoqi Peng, David C. Budd, Matthew C. Lucas, Rama K. Kondru, Ruben Alvarez Sanchez
المصدر: Journal of Medicinal Chemistry. 55:7920-7939
مصطلحات موضوعية: Gene isoform, Spectrometry, Mass, Electrospray Ionization, Magnetic Resonance Spectroscopy, Phospholipid, Antagonist, Administration, Oral, Stimulation, Fibroblasts, Pharmacology, Mice, Structure-Activity Relationship, chemistry.chemical_compound, chemistry, Drug Discovery, Lysophosphatidic acid, Knockout mouse, Animals, Humans, Pyrazoles, Molecular Medicine, Structure–activity relationship, lipids (amino acids, peptides, and proteins), Receptors, Lysophosphatidic Acid, Receptor, Lung
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8
المؤلفون: Laurent Salphati, Stewart J. Baker, Steve Price, Jim Nonomiya, Matthew C. Lucas, Timothy Hancox, David Knowles, Bohdan Waszkowycz, Neil Anthony Pegg, David Chantry, Bryan K. Chan, Paul Blaney, Anthony Brown, Steven T. Staben, Jodie Pang, Paul Depledge, Rama K. Kondru, Mark Ultsch, Paul Goldsmith, Karin Reif, Angelina Bisconte, Cristina Lewis, Eileen Mary Seward, Jeremy Murray, Brian Safina, Daniel P. Sutherlin, Zachary Kevin Sweeney, Georgette Castanedo, David Michael Goldstein, Jasmit Kaur, Sukhjit Sohal, Binqing Wei, John Lesnick, Stephen J. Shuttleworth, Alan Nadin
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:4296-4302
مصطلحات موضوعية: Male, Gene isoform, Stereochemistry, Clinical Biochemistry, Mutant, Pharmaceutical Science, Biochemistry, Rats, Sprague-Dawley, Mice, Phosphatidylinositol 3-Kinases, Structure-Activity Relationship, In vivo, Drug Discovery, Animals, Protein Isoforms, Computer Simulation, Protein Kinase Inhibitors, Molecular Biology, PI3K/AKT/mTOR pathway, Phosphoinositide-3 Kinase Inhibitors, Mice, Inbred BALB C, Binding Sites, Chemistry, Kinase, Organic Chemistry, Tryptophan, Protein Structure, Tertiary, Rats, Liver, Injections, Intravenous, Mutation, Molecular Medicine, Female, Selectivity
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9
المؤلفون: Robert Greenhouse, Hai-Ying Cai, Ryan Craig Schoenfeld, David S. Carter, Stephen M. Lynch, Ann Marie Madera, Sandra Steiner, Yansheng Zhai, Eun Kyung Lee, Robert James Weikert, Clara Jeou Jen Lin, Kerem Erol Ozboya, Amy Geraldine Moore, Pravin Iyer, Matthew C. Lucas
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:5559-5566
مصطلحات موضوعية: Serotonin, Pyrrolidines, Dopamine, Clinical Biochemistry, hERG, Pain, Pharmaceutical Science, Antidepressive Agents, Tricyclic, Biochemistry, Norepinephrine, chemistry.chemical_compound, Dopamine Uptake Inhibitors, In vivo, Drug Discovery, medicine, Animals, Humans, Neurotransmitter Uptake Inhibitors, Neurotransmitter, Molecular Biology, biology, Depression, Organic Chemistry, Rats, Monoamine neurotransmitter, chemistry, Drug Design, Catecholamine, biology.protein, Molecular Medicine, Caco-2 Cells, Reuptake inhibitor, Selective Serotonin Reuptake Inhibitors, medicine.drug
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المؤلفون: Matthew C. Lucas, Gisele A. Tavares, Deborah Carol Reuter, Nidhi Arora, Amy Fung, Sophie Le Pogam, Vincent Leveque, Hanbiao Yang, Yanli Yang, Dov Nitzan, Robert Than Hendricks, Calvin Yee, Julie Q. Hang, Sonal Rajyaguru, Seth F. Harris
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:4614-4619
مصطلحات موضوعية: Molecular model, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Hepacivirus, Thiophenes, Viral Nonstructural Proteins, Crystallography, X-Ray, Antiviral Agents, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Protein structure, Amide, Drug Discovery, Peptide bond, Structure–activity relationship, Enzyme Inhibitors, Binding site, Molecular Biology, NS5B, Binding Sites, Chemistry, Organic Chemistry, virus diseases, Amides, digestive system diseases, Protein Structure, Tertiary, Drug Design, Molecular Medicine, Bioisostere