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المؤلفون: Jian Sun, Jacques J. Kessl, Kaitlin A McNeely, Julie A. Pigza, Nicholas G. Jentsch, Chiyang Lama, Jared D. Hume, Alison P Hart, Matthew Garrett Donahue
المصدر: ACS Medicinal Chemistry Letters. 9:1007-1012
مصطلحات موضوعية: 0301 basic medicine, biology, Stereochemistry, Aryl, 030106 microbiology, Organic Chemistry, Quinoline, Biochemistry, In vitro, Integrase, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, ANTIRETROVIRAL AGENTS, chemistry, Viral replication, Drug Discovery, biology.protein, Hiv 1 integrase
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المصدر: Tetrahedron Letters. 58:3219-3222
مصطلحات موضوعية: Annulation, 010405 organic chemistry, Chemistry, Hydride, Organic Chemistry, chemistry.chemical_element, Decane, 010402 general chemistry, Ring (chemistry), 01 natural sciences, Biochemistry, Radical cyclization, 0104 chemical sciences, Terpene, chemistry.chemical_compound, Intramolecular force, Drug Discovery, Organic chemistry, Palladium
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المؤلفون: Julie A. Pigza, Jared D. Hume, Jacques J. Kessl, Matthew Garrett Donahue, Jian Sun, Krunal Patel
المصدر: The Journal of Biological Chemistry
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Integrase inhibitor, HIV Integrase, Virus Replication, Biochemistry, HIV-1, human immunodeficiency virus type 1, quinoline, HTRF, homogeneous time resolved fluorescence, human immunodeficiency virus, biology, Chemistry, CTD, C-terminal domain, DMSAO, dimethyl sulfoxide, Chromatin, Integrase, Cell biology, Quinolines, Intercellular Signaling Peptides and Proteins, CCD, catalytic core domain, I N, integrase, Research Article, Protein Binding, drug design, Virus Integration, Protein subunit, Allosteric regulation, ALLINI, allosteric IN inhibitors, Antiviral Agents, oligomerization, Protein–protein interaction, antiviral agent, 03 medical and health sciences, Allosteric Regulation, Humans, NTD, N-terminal domain, HIV Integrase Inhibitors, Binding site, Molecular Biology, RNP, ribonucleoprotein complex, 030102 biochemistry & molecular biology, Cell Biology, protein–protein interaction, HEK293 Cells, 030104 developmental biology, vDNA, viral cDNA, Viral replication, HIV-1, biology.protein, ALLINI, integrase, Protein Multimerization
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::812afed44ebca78da55c911ffeaba508
https://doi.org/10.1016/j.jbc.2021.100363 -
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المصدر: Tetrahedron Letters. 58:1692-1694
مصطلحات موضوعية: Benzimidazole, 010405 organic chemistry, Stable isotope ratio, Organic Chemistry, 010402 general chemistry, Ring (chemistry), Mass spectrometry, 01 natural sciences, Biochemistry, Medicinal chemistry, 0104 chemical sciences, Isotopomers, chemistry.chemical_compound, Aniline, chemistry, Drug Discovery, Ammonium formate, Nitro, Organic chemistry
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المؤلفون: Emily B. Crull, Samer M. Beauti, Jared D. Hume, Amy H. Pham, Jacques J. Kessl, Nicholas G. Jentsch, Matthew Garrett Donahue, Julie A. Pigza
المصدر: Beilstein Journal of Organic Chemistry
Beilstein Journal of Organic Chemistry, Vol 14, Iss 1, Pp 2529-2536 (2018)مصطلحات موضوعية: Sodium, chemistry.chemical_element, 010402 general chemistry, 01 natural sciences, Full Research Paper, lcsh:QD241-441, chemistry.chemical_compound, Residue (chemistry), lcsh:Organic chemistry, quinoline, Organic chemistry, isatoic anhydride, Carboxylate, lcsh:Science, HIV integrase, masked acyl cyanide, Triphosgene, 010405 organic chemistry, Quinoline, Organic Chemistry, 0104 chemical sciences, Chemistry, chemistry, Sodium hydroxide, Ethyl acetoacetate, Electrophile, cyclodehydration, lcsh:Q
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المصدر: The Journal of Organic Chemistry. 74:8726-8732
مصطلحات موضوعية: Cyclopropanes, Free Radicals, Allene, Organic Chemistry, Molecular Conformation, Free-radical reaction, Stereoisomerism, Photochemistry, Radical cyclization, Acceptor, Molecular conformation, chemistry.chemical_compound, chemistry, Fragmentation (mass spectrometry), Cyclization, Alkanes, Chemical reduction
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المؤلفون: David J. Hart, Matthew Garrett Donahue
المصدر: Canadian Journal of Chemistry. 82:314-317
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, chemistry, Aldol reaction, Organic Chemistry, Quassinoid, Titanium tetrachloride, Ketene, Organic chemistry, General Chemistry, Aldehyde, Radical cyclization, Catalysis
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المؤلفون: Matthew Garrett Donahue, Jeffrey N. Johnston, Ki Bum Hong
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:4971-4973
مصطلحات موضوعية: Mesylates, Oxazolidine, Proton, Nitrogen, Triazines, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Combinatorial chemistry, chemistry.chemical_compound, chemistry, Fragmentation (mass spectrometry), Drug Discovery, Solvents, Molecular Medicine, Organic chemistry, Azide, Protons, Brønsted–Lowry acid–base theory, Imide, Oxazoles, Molecular Biology, Trifluoromethanesulfonate
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المؤلفون: Jeffrey N. Johnston, Matthew Garrett Donahue
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:5602-5604
مصطلحات موضوعية: chemistry.chemical_classification, Dipeptide, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Phosphoramidon, Glycopeptides, Organophosphonates, Pharmaceutical Science, Peptide, respiratory system, Biochemistry, Chemical synthesis, Medicinal chemistry, Phosphonate, Coupling (electronics), chemistry.chemical_compound, chemistry, Drug Discovery, Molecular Medicine, Molecular Biology