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المؤلفون: Tsuyoshi Nakamura, Mika Yokoyama, Mayuko Akiu, Takashi Tsuji, Kouki Iida, Ken Sakurai, Yoshitaka Sogawa, Koji Terayama, Tomohiro Honda, Jun Tanaka, Daigo Asano, Anthony B. Pinkerton
المصدر: Chemical and Pharmaceutical Bulletin. 69:1110-1122
مصطلحات موضوعية: Male, Nicotinamide phosphoribosyltransferase, Mice, Obese, Type 2 diabetes, Pharmacology, Nicotinamide adenine dinucleotide, Small Molecule Libraries, Structure-Activity Relationship, chemistry.chemical_compound, Pharmacokinetics, Oral administration, Drug Discovery, medicine, Animals, Humans, Urea, Obesity, Nicotinamide Phosphoribosyltransferase, Nucleotide salvage, Chemistry, Activator (genetics), Body Weight, General Chemistry, General Medicine, NAD, medicine.disease, Diabetes Mellitus, Type 2, Anti-Obesity Agents, NAD+ kinase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1559d4d089014d0c71e8a23a236697a9
https://doi.org/10.1248/cpb.c21-00700 -
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المؤلفون: Mayuko Akiu, Takashi Tsuji, Yoshitaka Sogawa, Koji Terayama, Mika Yokoyama, Daigo Asano, Tomohiro Honda, Tomomichi Ishizaka, Tomoko Hasegawa, Anthony B. Pinkerton, Tsuyoshi Nakamura
المصدر: HETEROCYCLES. 104:94
مصطلحات موضوعية: Pharmacology, Organic Chemistry, Analytical Chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::d04af8f16133d0aaef6c447d4bbfefd9
https://doi.org/10.3987/com-21-14559 -
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المؤلفون: Jun Tanaka, Daigo Asano, E. Hampton Sessions, Koji Terayama, Mika Yokoyama, Mayuko Akiu, Takashi Tsuji, Ken Sakurai, Stephen J. Gardell, Yoshitaka Sogawa, Anthony B. Pinkerton, Eduard Sergienko, Tsuyoshi Nakamura
المصدر: Bioorganic & Medicinal Chemistry Letters. 43:128048
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Nicotinamide phosphoribosyltransferase, Pharmaceutical Science, 01 natural sciences, Biochemistry, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, Drug Discovery, Animals, Humans, Urea, Enzyme Inhibitors, Nicotinamide Phosphoribosyltransferase, Molecular Biology, Nucleotide salvage, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Activator (genetics), Organic Chemistry, Metabolism, 0104 chemical sciences, Mice, Inbred C57BL, 010404 medicinal & biomolecular chemistry, chemistry, Lipophilicity, Cytokines, Molecular Medicine, Triazolopyridine, NAD+ kinase, Lead compound
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المؤلفون: Mayuko Akiu, Steven E. Cohen, Chen-Ting Ma, E. Hampton Sessions, Layton H. Smith, Michael R. Jackson, Paul Hershberger, Stephen J. Gardell, Patrick R. Maloney, Takashi Tsuji, Eduard Sergienko, Satyamaheshwar Peddibhotla, Jun Tanaka, Anthony B. Pinkerton, Tsuyoshi Nakamura, Meghan E. Hopf
المصدر: Bioorganic & Medicinal Chemistry Letters. 41:128007
مصطلحات موضوعية: Clinical Biochemistry, Nicotinamide phosphoribosyltransferase, Pharmaceutical Science, 01 natural sciences, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Humans, Urea, Nicotinamide Phosphoribosyltransferase, Molecular Biology, Nucleotide salvage, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Activator (genetics), Organic Chemistry, Neurodegeneration, medicine.disease, In vitro, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry, Cytokines, Molecular Medicine, NAD+ kinase
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المؤلفون: Yoshitaka Sogawa, Yasuyuki Abe, Mayuko Akiu, Kousei Shimada, Yoko Nagai, Masanori Izumi, Masahiro Konishi, Masanori Suzuki, Rie Abe-Ohya, Shozo Kobayashi, Hisashi Takahashi, Hideo Takamori, Kazuhiro Yoshida, Takashi Hara, Masayoshi Asano, Yohei Kiyotsuka
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:4205-4210
مصطلحات موضوعية: Central Nervous System, 0301 basic medicine, Carboxylic acid, Clinical Biochemistry, Central nervous system, Pharmaceutical Science, Blood Pressure, Acetates, Pharmacology, Heterocyclic Compounds, 2-Ring, 030226 pharmacology & pharmacy, Biochemistry, Eating, Mice, 03 medical and health sciences, chemistry.chemical_compound, Dogs, 0302 clinical medicine, Pharmacokinetics, Heart Rate, In vivo, Drug Discovery, medicine, Animals, Humans, Moiety, Adverse effect, Molecular Biology, chemistry.chemical_classification, Organic Chemistry, Imidazoles, Brain, Mice, Inbred C57BL, Receptors, Bombesin, 030104 developmental biology, medicine.anatomical_structure, chemistry, Injections, Intravenous, Molecular Medicine, Bombesin Receptor Subtype-3, Anti-Obesity Agents, Penetrant (biochemical), Half-Life
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