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1
المؤلفون: Ching Kim Tye, Chunhong Yan, Sarah C. Traeger, Wayne Vaccaro, Yingru Zhang, Gerry Everlof, Jianqing Li, Henry Yip, Peng Li, John T. Hunt, Michael A. Poss, Gregory D. Vite, Mussari Christopher P, Steven Sheriff, Asoka Ranasinghe, Haiying Zhang, Richard A. Westhouse, Dharmpal S. Dodd, Richard Rampulla, Zheng Yang, Frank Marsilio, Derek J. Norris, Wen-Ching Han, Tram N. Huynh, Yufen Zhao, Patrice Gill, Nirmala Raghavan, Lalgudi S. Harikrishnan, Ashvinikumar V. Gavai, Susan Wee, John S. Tokarski, Dauh-Rurng Wu, Arvind Mathur, Mei-Li Wen, Huiping Zhang, David R. Tortolani, George V. Delucca, Krista Menard, Francis Y. Lee, Claude A. Quesnelle, Dawn Sun, Vijay T. Ahuja, Daniel O'malley, Christine Huang, Muthoni G. Kamau
المصدر: Journal of Medicinal Chemistry. 64:14247-14265
مصطلحات موضوعية: Drug, Proline, Phenylalanine, media_common.quotation_subject, Carbazoles, Administration, Oral, Antineoplastic Agents, Cell Cycle Proteins, Computational biology, BET inhibitor, Structure-Activity Relationship, Pharmacokinetics, In vivo, Drug Discovery, Transcriptional regulation, Humans, Potency, media_common, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Tryptophan, Signal transducing adaptor protein, Bromodomain, Molecular Medicine, Transcription Factors
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2
المؤلفون: Mei Li Wen Wu, Ming Chen, Fei Cao
المصدر: Applied Mechanics and Materials. 826:40-44
مصطلحات موضوعية: Engineering, business.industry, 010102 general mathematics, Particle swarm optimization, ComputerApplications_COMPUTERSINOTHERSYSTEMS, Control engineering, General Medicine, Aerodynamics, 01 natural sciences, Sizing, law.invention, Coaxial rotors, Conceptual design, Flight dynamics, law, Design process, 0101 mathematics, business, Intersection (aeronautics)
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3
المؤلفون: George L. Trainor, Jun Dai, Arvind Mathur, Francis Y. Lee, Sunilkumar Mandal, Yingru Zhang, Richard Rampulla, Kiran Babu Gona, Patrice Gill, Raja Thiruvenkadam, Victor R. Guarino, Wen-Ching Han, Ding Ren Shen, Aaron Balog, Mary Ellen Cvijic, Dauh-Rurng Wu, Gregory D. Vite, Krista Menard, Anne Rose, Sathiah Kandula, Ashvinikumar V. Gavai, Weifang Shan, John T. Hunt, Asoka Ranasinghe, Kelly McGlinchey, Richard A. Westhouse, Claude A. Quesnelle, Derek J. Norris, Mei-Li Wen, Ronald E. White, Kamalraj Thiyagarajan
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:1905-1909
مصطلحات موضوعية: Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Antineoplastic Agents, Pharmacology, Biochemistry, Mice, Structure-Activity Relationship, In vivo, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Receptor, Solid tumor, Molecular Biology, Cell Proliferation, Benzodiazepinones, Dose-Response Relationship, Drug, Molecular Structure, Receptors, Notch, Chemistry, Organic Chemistry, Biological activity, Neoplasms, Experimental, medicine.disease, Leukemia, Orally active, Microsomes, Liver, Molecular Medicine, Drug Screening Assays, Antitumor
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4
المؤلفون: Claude A. Quesnelle, Patrice Gill, Richard Rampulla, Ching Su, Gerry Everlof, George L. Trainor, Ke Chen, Vinod Arora, Richard A. Westhouse, Celia D’Arienzo, Andrew J. Tebben, Weifang Shan, John T. Hunt, Derek J. Norris, Louis J. Lombardo, Zheng Yang, Arvind Mathur, Mei-Li Wen, Yingru Zhang, Dauh-Rurng Wu, Wen-Ching Han, Krista Menard, Victor R. Guarino, Asoka Ranasinghe, Richard E. Olson, Ashvinikumar V. Gavai, Bruce S. Fischer, Phil S. Baran, Anne Rose, Lan Xiao, Ronald E. White, Mary Ellen Cvijic, Gregory D. Vite, Ding Ren Shen, Jere E. Meredith, Haiqing Wang, Francis Y. Lee, Aaron Balog
المصدر: ACS Medicinal Chemistry Letters. 6:523-527
مصطلحات موضوعية: business.industry, Organic Chemistry, Pharmacology, medicine.disease, Biochemistry, T Acute Lymphoblastic Leukemia, Leukemia, In vivo, Drug Discovery, medicine, Receptor, business, Solid tumor, Clinical evaluation, Triple-negative breast cancer
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5
المؤلفون: Craig R. Fairchild, Francis Y. Lee, Anne Lewin, Kelly L. Covello, Rolf-Peter Ryseck, Mei-Li Wen, Donald R. Hawken, Robert A. Kramer, David Kan, Joseph Fargnoli, Stephen Castaneda
المصدر: Clinical Cancer Research. 14:8123-8131
مصطلحات موضوعية: Cancer Research, Indoles, Bevacizumab, Angiogenesis, medicine.medical_treatment, Angiogenesis Inhibitors, Antineoplastic Agents, Pharmacology, Antibodies, Monoclonal, Humanized, Mice, chemistry.chemical_compound, In vivo, Sunitinib, medicine, Animals, Humans, Pyrroles, ATP Binding Cassette Transporter, Subfamily B, Member 1, Mice, Inbred BALB C, Mice, Inbred C3H, Chemotherapy, business.industry, Ixabepilone, Antibodies, Monoclonal, Endothelial Cells, Drug Synergism, medicine.disease, Xenograft Model Antitumor Assays, Metastatic breast cancer, Oncology, chemistry, Paclitaxel, Epothilones, Female, business, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ebfaa4a117b00a2f221ecd8bf889097b
https://doi.org/10.1158/1078-0432.ccr-08-0025 -
6
المؤلفون: Dan You, Simone Oppenheimer, Brian E. Fink, Francis Y.F. Lee, Kristen A. Kellar, Bruce Rowley, Rolf P. Ryseck, Ching Ping Ho, David Bol, Chiang Yu, Mei-Li Wen, Matthew V. Lorenzi, Tai W. Wong, Gregory D. Vite
المصدر: Molecular Cancer Therapeutics. 5:1571-1576
مصطلحات موضوعية: Cancer Research, Receptor, ErbB-2, CD8 Antigens, Recombinant Fusion Proteins, Transgene, Blotting, Western, Cell, Mice, Nude, Mammary Neoplasms, Animal, Mice, Transgenic, Transfection, Receptor tyrosine kinase, Mice, medicine, Animals, Humans, Disulfides, Receptor, Mice, Inbred BALB C, biology, Kinase, Receptor Protein-Tyrosine Kinases, Epithelial Cells, Fibroblasts, Proto-Oncogene Proteins c-met, Salivary Gland Neoplasms, Fusion protein, Peptide Fragments, Rats, Cell biology, Gene Expression Regulation, Neoplastic, Disease Models, Animal, Cell Transformation, Neoplastic, medicine.anatomical_structure, Oncology, Cell culture, biology.protein, Female, Dimerization, Plasmids
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::39fb27ea3060c91c3d6561d069291438
https://doi.org/10.1158/1535-7163.mct-06-0078 -
7
المؤلفون: Cindy Wang, Joan M. Carboni, Marco M. Gottardis, Ann Greer, David Bol, Amy Camuso, Aixin Li, Bruce Rowley, Warren Hurlburt, Brent A. Rupnow, Francis Y.F. Lee, Darryl L. Hadsell, Mark D. Wittman, Saulnier Mark G, Upender Velaparthi, Tai W. Wong, Mei-Li Wen, Kurt Zimmermann, Richard A. Westhouse, Adrian V. Lee, Ching Ping Ho
المصدر: Cancer Research. 65:3781-3787
مصطلحات موضوعية: Cancer Research, medicine.medical_specialty, CD8 Antigens, Recombinant Fusion Proteins, Transplantation, Heterologous, Mice, Nude, Mice, Transgenic, Tropomyosin receptor kinase B, Adenocarcinoma, Biology, Transfection, Tropomyosin receptor kinase C, Receptor, IGF Type 1, Mice, Growth factor receptor, Pregnancy, Internal medicine, medicine, Animals, Humans, Transgenes, Protease-activated receptor 2, Insulin-like growth factor 1 receptor, Mice, Inbred BALB C, Mice, Inbred ICR, Mammary Neoplasms, Experimental, Salivary Gland Neoplasms, Cell biology, Cell Transformation, Neoplastic, Endocrinology, Oncology, Interleukin-21 receptor, ROR1, Female, Tyrosine kinase, Neoplasm Transplantation
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::75c86c8d67f12be593606f26753f4d4c
https://doi.org/10.1158/0008-5472.can-04-4602 -
8
المؤلفون: John Wityak, Amrita Kamath, Louis J. Lombardo, Ping Chen, John T. Hunt, Ivan Inigo, Stephen Castaneda, Joel C. Barrish, Herbert E. Klei, Robert J. Schmidt, John S. Tokarski, Sidney Pitt, Derek J. Norris, Francis Y. Lee, Jagabandhu Das, Craig Fairchild, Kathy A. Johnston, Punit Marathe, Robert M. Borzilleri, Cornelius Lyndon A M, Suhong Pang, Mei-Li Wen, Russell Peterson, Gary L. Schieven, Kamelia Behnia, David Kan, Arthur M. Doweyko
المصدر: Journal of Medicinal Chemistry. 47:6658-6661
مصطلحات موضوعية: Stereochemistry, medicine.drug_class, Dasatinib, Antineoplastic Agents, Carboxamide, Pharmacology, Rats, Sprague-Dawley, Mice, chemistry.chemical_compound, Adenosine Triphosphate, hemic and lymphatic diseases, Drug Discovery, medicine, Animals, Humans, Enzyme Inhibitors, Proto-Oncogene Proteins c-abl, Thiazole, ABL, biology, Chemistry, medicine.disease, Rats, Thiazoles, Pyrimidines, src-Family Kinases, Enzyme inhibitor, biology.protein, Molecular Medicine, K562 Cells, Chronic myelogenous leukemia, Proto-oncogene tyrosine-protein kinase Src, K562 cells, medicine.drug
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9
المؤلفون: Feng Roger Luo, Robert A. Wild, Anne Blackwood-Chirchir, Francis Y. Lee, Holly Palme, Yu Chen Barrett, Amy Camuso, Richard Smykla, Zheng Yang, Susan Galbraith, Krista Fager, Mei-Li Wen, Kelly McGlinchey
المصدر: Cancer chemotherapy and pharmacology. 62(6)
مصطلحات موضوعية: Male, Cancer Research, medicine.drug_class, Dasatinib, Mice, Nude, Antineoplastic Agents, Biology, Adenocarcinoma, Toxicology, Peripheral blood mononuclear cell, Tyrosine-kinase inhibitor, Substrate Specificity, Mice, In vivo, hemic and lymphatic diseases, medicine, Animals, Humans, Pharmacology (medical), Phosphorylation, Protein Kinase Inhibitors, Pharmacology, Kinase, Prostatic Neoplasms, Biological activity, Phosphoproteins, Xenograft Model Antitumor Assays, Neoplasm Proteins, Specific Pathogen-Free Organisms, Thiazoles, Pyrimidines, src-Family Kinases, Oncology, Cancer research, Leukocytes, Mononuclear, Biomarker (medicine), Female, Drug Monitoring, Biomarkers, Cell Division, Proto-oncogene tyrosine-protein kinase Src, medicine.drug
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10
المؤلفون: Patrice Gill, Daniel O'malley, Mary Ellen Cvijic, George L. Trainor, Gregory D. Vite, Yingru Zhang, Richard Rampulla, Richard A. Westhouse, Celia D’Arienzo, Derek J. Norris, Wen-Ching Han, Ching Su, Mei-Li Wen, Libing Chen, Arvind Mathur, Andrew J. Tebben, Brian E. Fink, Bruce S. Fischer, Robin Moore, Francis Y. Lee, David Rodrigues, Qian Ruan, Gerry Everlof, Weifang Shan, John T. Hunt, Claude A. Quesnelle, Soong-Hoon Kim, Krista Menard, Dauh-Rurng Wu, Asoka Ranasinghe, Zheng Yang, Yufen Zhao, Ashvinikumar V. Gavai, Aaron Balog, Haiqing Wang, Ching Kim Tye, Melissa Yarde
المصدر: Cancer Research. 74:1643-1643
مصطلحات موضوعية: Gerontology, Cancer Research, Angiogenesis, Colorectal cancer, business.industry, Notch signaling pathway, medicine.disease, Metastasis, Breast cancer, Oncology, Cancer stem cell, Apoptosis, Cancer research, medicine, business, Transcription factor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::761271a037a354d0d93f3b39b4fca9c3
https://doi.org/10.1158/1538-7445.am2014-1643