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المؤلفون: Robert H. Scannevin, Kenneth J. Rhodes, Mi Young Jung, Matvey E. Lukashev, Sowmya Chollate, Melanie N. Shackett, Masayuki Yamamoto, Weike Zeng, Sarah Ryan, Hiral Patel, Pradeep Bista
المصدر: Journal of Pharmacology and Experimental Therapeutics. 341:274-284
مصطلحات موضوعية: Central Nervous System, Antioxidant, NF-E2-Related Factor 2, medicine.medical_treatment, Oxidative phosphorylation, Biology, Pharmacology, medicine.disease_cause, Neuroprotection, Mice, chemistry.chemical_compound, Fumarates, medicine, Animals, Humans, Viability assay, Cells, Cultured, Mice, Knockout, Neurons, Dimethyl fumarate, Glutathione, Cytoprotection, Mice, Inbred C57BL, Oxidative Stress, Neuroprotective Agents, chemistry, Molecular Medicine, Oxidative stress, Signal Transduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::726689985fd6f8b86aa0a8ad08c76553
https://doi.org/10.1124/jpet.111.190132 -
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المؤلفون: Robert H. Scannevin, Tina Talreja, Lin Xu, Gnanasambandam Kumaravel, David Kocisko, Arthur G. Taveras, Anthone W. Dunah, Hairuo Peng, Kenneth J. Rhodes, Ellen Rohde, H. Moore Arnold, Sowmya Chollate, Pamela A. Snodgrass-Belt, Mi-yong Jung, Andrew Zhang, Zhili Xin, Melanie N. Shackett
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:7277-7280
مصطلحات موضوعية: Scaffold, Carboxylic acid, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Pharmaceutical Science, Pharmacology, Biochemistry, Mice, chemistry.chemical_compound, Piperidines, Oral administration, Drug Discovery, Animals, γ secretase, Enzyme Inhibitors, Molecular Biology, Phenylacetates, chemistry.chemical_classification, Amyloid beta-Peptides, Nonsteroidal, Anti-Inflammatory Agents, Non-Steroidal, Organic Chemistry, Brain, Combinatorial chemistry, Peptide Fragments, Rats, chemistry, Drug Design, Molecular Medicine, Amyloid Precursor Protein Secretases
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المؤلفون: Tina Talreja, Arthur G. Taveras, Michael Humora, Lawrence Gan, J. Hernan Cuervo, Kenneth J. Rhodes, Hairuo Peng, Lin Xu, Anthone W. Dunah, Gnanasambandam Kumaravel, Pamela A. Snodgrass-Belt, Mi-young Jung, Zhili Xin, Sowmya Chollate, Melanie N. Shackett, Ellen Rohde, H. Moore Arnold, Robert H. Scannevin
المصدر: ACS Medicinal Chemistry Letters. 2:786-791
مصطلحات موضوعية: biology, business.industry, Organic Chemistry, Notch signaling pathway, Pharmacology, Biochemistry, In vitro, Pharmacokinetics, In vivo, Oral administration, Pharmacodynamics, Drug Discovery, biology.protein, Medicine, Potency, business, Amyloid precursor protein secretase