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1
المؤلفون: Denton Hoyer, Mike Ran Zou, Lauren P. Blair, Jane S. Merkel, Alfonso Morales, Alan J. Tackett, Michael Norcia, Qin Yan, Jian Cao, Joyce Sayegh
المصدر: Journal of Biological Chemistry. 288:9408-9417
مصطلحات موضوعية: Jumonji Domain-Containing Histone Demethylases, Insecta, Chemistry, Pharmaceutical, Antineoplastic Agents, environment and public health, Biochemistry, Cell Line, Epigenesis, Genetic, Histones, Histone H3, Cell Line, Tumor, Neoplasms, Histone methylation, Animals, Humans, Gene Regulation, Molecular Biology, Cell Proliferation, Histone Demethylases, biology, Nuclear Proteins, Cell Biology, Small molecule, Recombinant Proteins, High-Throughput Screening Assays, Repressor Proteins, Thiazoles, Histone, Drug Design, biology.protein, Cancer research, H3K4me3, Demethylase, Peptides, JARID1B, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::87b57e6ade721fd9329802eb93248115
https://doi.org/10.1074/jbc.m112.419861 -
2
المؤلفون: Michael Norcia, Denton Hoyer, Molly Gale, Joyce Sayegh, Jian Cao, Peter C. Gareiss, Jane S. Merkel, Qin Yan
المصدر: Oncotarget
مصطلحات موضوعية: 0301 basic medicine, Luminescence, Breast Neoplasms, Pharmacology, medicine.disease_cause, Epigenesis, Genetic, Histones, 03 medical and health sciences, Inhibitory Concentration 50, 0302 clinical medicine, Drug tolerance, Demethylase activity, medicine, Humans, Neoplasm Metastasis, Cell Proliferation, drug resistance, biology, epigenetics, Cancer, Drug Tolerance, medicine.disease, 3. Good health, 030104 developmental biology, Treatment Outcome, Oncology, Drug Resistance, Neoplasm, histone demethylase inhibitor, anti-cancer drug, 030220 oncology & carcinogenesis, KDM5A, Cancer cell, biology.protein, MCF-7 Cells, Demethylase, JARID1B, Carcinogenesis, Peptides, Retinoblastoma-Binding Protein 2, HeLa Cells, Research Paper
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9aa03b5fdc213577f5d3c4afe7bf701a
https://pubmed.ncbi.nlm.nih.gov/27224921 -
3
المؤلفون: Michael Norcia, Shinichi Sakemi, Joyce A. Sutcliffe, Nakao Kojima, Etsuko Iwata, Taisuke Inagaki, Tatsuo Sakakibara, Yuji Yamauchi, Lillian M. Wondrack, Hideo Hirai, Keiji Kaneda
المصدر: ChemInform. 26
مصطلحات موضوعية: biology, Chemistry, Topoisomerase, General Medicine, biology.organism_classification, Cleavage (embryo), DNA gyrase, Biochemistry, biology.protein, DNA supercoil, Fermentation, Antibacterial activity, Selectivity, Bacteria
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المؤلفون: Thomas J. Dougherty, Kevin Daniel Freeman-Cook, Michael Norcia, Charlene R. Desbonnet, Hong Wang, Laura E. Zawadzke
المصدر: Assay and drug development technologies. 6(1)
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, Drug Evaluation, Preclinical, Microbial Sensitivity Tests, Peptidoglycan, Biology, Inhibitory postsynaptic potential, medicine.disease_cause, Pentapeptide repeat, Maltose-Binding Proteins, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Escherichia coli, Enzyme Inhibitors, Peptide Synthases, Proteus mirabilis, DNA Primers, chemistry.chemical_classification, DNA ligase, Receptors, Purinergic P2, Stereoisomerism, biology.organism_classification, Molecular biology, Enzyme assay, Anti-Bacterial Agents, Klebsiella pneumoniae, Enzyme, chemistry, Biochemistry, biology.protein, Molecular Medicine, Carrier Proteins, Bacteria
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::48833d584445e5f5fb637f2a45306e08
https://pubmed.ncbi.nlm.nih.gov/18315498 -
5
المؤلفون: Joyce A. Sutcliffe, J Bergeron, Christine A. Strick, Larry C. James, W G Su, James A. Retsema, L Wondrack, Dennis E. Danley, Mark Ammirati, Michael Norcia
مصطلحات موضوعية: Peptide Biosynthesis, Tetracycline, Biology, medicine.disease_cause, Glycylcycline, Ribosome, medicine, Escherichia coli, Pharmacology (medical), Antibacterial agent, Pharmacology, Doxycycline, Cell-Free System, Glycylglycine, Tetracycline Resistance, Ribosomal RNA, Molecular biology, Ribosomal binding site, Anti-Bacterial Agents, Infectious Diseases, Biochemistry, Biological Assay, Ribosomes, medicine.drug, Research Article
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8e8ff0851d0c8fc58e6c405aae3027ca
https://europepmc.org/articles/PMC163507/ -
6
المؤلفون: Shinichi Sakemi, Nakao Kojima, Hideo Hirai, Yuji Yamauchi, Taisuke Inagaki, Joyce A. Sutcliffe, Michael Norcia, Keiji Kaneda, Lillian M. Wondrack, Tatsuo Sakakibara, Etsuko Iwata
المصدر: The Journal of antibiotics. 48(2)
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, Stereochemistry, Naphthalenes, Gram-Positive Bacteria, DNA gyrase, Drug Discovery, Escherichia coli, Topoisomerase II Inhibitors, Antibacterial agent, Pharmacology, chemistry.chemical_classification, biology, Molecular Structure, Topoisomerase, Spectrum Analysis, Fungi, Biological activity, Stereoisomerism, biology.organism_classification, Anti-Bacterial Agents, Enzyme, Biochemistry, chemistry, Fermentation, biology.protein, DNA supercoil, Antibacterial activity, Bacteria
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a6c3e7a7c5b8df5b1e0e390e85e19b13
https://pubmed.ncbi.nlm.nih.gov/7706123 -
7دورية أكاديمية
المؤلفون: Laura E. Zawadzke, Michael Norcia, Charlene R. Desbonnet, Hong Wang, Kevin Freeman-Cook, Thomas J. Dougherty
المصدر: Assay & Drug Development Technologies; Feb2008, Vol. 6 Issue 1, p95-103, 9p
مصطلحات موضوعية: PEPTIDOGLYCANS, PEPTIDES, GRAM-positive bacteria, GRAM-negative bacteria, ENZYMES