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المؤلفون: Giorgio Ottaviani, Lin Gao, Simona M. Ceccarelli, Ulrike Obst-Sander, Rodolfo Gasser, Xiaolei Zhang, Michael Paul Myers, Sung-Sau So, Bernd Kuhn, Holger Kühne, Shirley Li, Werner Neidhart, Aurelia Conte, Markus G. Rudolph
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:5092-5097
مصطلحات موضوعية: 0301 basic medicine, Dual inhibition, Protein Conformation, Clinical Biochemistry, Pharmaceutical Science, Fatty Acid-Binding Proteins, Biochemistry, Fatty acid-binding protein, Mice, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, In vivo, Drug Discovery, Animals, Amino Acid Sequence, Molecular Biology, Beneficial effects, Mice, Knockout, Sequence Homology, Amino Acid, Chemistry, Organic Chemistry, Insulin sensitivity, Transport protein, 030104 developmental biology, Drug Design, 030220 oncology & carcinogenesis, Molecular Medicine, Selectivity
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2
المؤلفون: Rebecca Taub, Robert Alan Goodnow, Lida Qi, Joseph Anthony Bilotta, Sherrie Lynn Pietranico-Cole, Yonglin Ren, Cheryl Spence, Jefferson Wright Tilley, Baolian Liu, Sung-Sau So, Kevin Richard Guertin, Karin Conde-Knape, Matthew Michael Hamilton, Nancy-Ellen Haynes, Kshitij Chhabilbhai Thakkar, Catherine Zwingelstein, Nathan Robert Scott, Paul Gillespie, Michael Paul Myers, Nader Fotouhi
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:2707-2711
مصطلحات موضوعية: Hydrocortisone, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Inhibitory Concentration 50, Mice, Camphor, chemistry.chemical_compound, Pharmacokinetics, In vivo, 11β-hydroxysteroid dehydrogenase type 1, 11-beta-Hydroxysteroid Dehydrogenase Type 1, Drug Discovery, Animals, Potency, Enzyme Inhibitors, Pyrazolones, Molecular Biology, Molecular Structure, biology, Chemistry, Organic Chemistry, Hit to lead, Rats, Enzyme Activation, biology.protein, Molecular Medicine, Female
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3
المؤلفون: Robert Alan Goodnow, Sung-Sau So, Gopal Bose, Goutam Saha, Karin Conde-Knape, Sherrie Lynn Pietranico-Cole, Paul Gillespie, Michael Paul Myers, Kakali Moulik, Catherine Zwingelstein
المصدر: Bioorganicmedicinal chemistry letters. 24(3)
مصطلحات موضوعية: Agonist, Pyrimidine, Chemistry, Stereochemistry, medicine.drug_class, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Glucose excursion, Biochemistry, Receptors, G-Protein-Coupled, chemistry.chemical_compound, Mice, Structure-Activity Relationship, GPR119, Pyrimidines, Pharmacokinetics, Drug Discovery, medicine, Molecular Medicine, Potency, Animals, Humans, Pyrazoles, Molecular Biology