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1
المؤلفون: Mason Helen J, Karen D. Brown, Valeria Chu, Guyan Liang, Daniel M. Green, Alfred P. Spada, Henry W. Pauls, Ross Bentley, Cuong Ly, Roderick S. Davis, Dennis J. Colussi, Daniel L. Cheney, Michael R. Becker, Y.M. Choi-Sledeski, Christopher T. Dunwiddie, Robert J. Leadley, Ewing William R, John H. Barton
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:2539-2544
مصطلحات موضوعية: Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, Isostere, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Administration, Oral, Pharmaceutical Science, Biochemistry, Chemical synthesis, Benzamidine, Amidine, Serine, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Drug Discovery, medicine, Animals, Structure–activity relationship, Molecular Biology, Binding Sites, Organic Chemistry, Isoquinolines, Benzamidines, chemistry, Molecular Medicine, Factor Xa Inhibitors
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2
المؤلفون: Alfred P. Spada, Robert J. Leadley, Jonathan S. Mason, Dennis J. Colussi, Ewing William R, Mark H. Perrone, Karen D. Brown, Michael R. Becker, Don D. Cha, Daniel M. Green, Ross Bentley, Henry W. Pauls, Christopher T. Dunwiddie, Jean-Pierre Guilloteau, Y.M. Choi-Sledeski, Sebastien Maignan, Mason Helen J, Vincent E. Manetta, Charles Kasiewski, Valeria Chu, Roderick S. Davis, Suzanne Morgan, Daniel L. Cheney, Jeff Bostwick
المصدر: Journal of Medicinal Chemistry. 42:3557-3571
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, medicine.drug_class, Factor Xa Inhibitor, Thiophenes, Crystallography, X-Ray, Amidine, Structure-Activity Relationship, chemistry.chemical_compound, Thrombin, In vivo, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Sulfonamides, Molecular Structure, biology, Chemistry, Anticoagulant, Anticoagulants, Stereoisomerism, Thrombosis, Trypsin, Pyrrolidinones, Rats, Biochemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Rabbits, Factor Xa Inhibitors, medicine.drug
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3
المؤلفون: Michael R. Becker, et al. et al.
المصدر: ChemInform. 30
مصطلحات موضوعية: chemistry.chemical_classification, Thienopyridine, chemistry, medicine.drug_mechanism_of_action, In vivo, Factor Xa Inhibitor, medicine, General Medicine, Pyrrolidinones, Combinatorial chemistry, Pyrrole derivatives, Sulfonamide
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4
المؤلفون: Michael R. Becker, Frederick E. Ziegler
المصدر: The Journal of Organic Chemistry. 55:2800-2805
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, Hydrolysis, Ketone, Chemistry, Stereochemistry, Organic Chemistry, Hemiacetal, Total synthesis, Acid hydrolysis, Aldol condensation, Aldehyde, Derivative (chemistry)
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::83a41bf63b7c98e920a0fe32aae29918
https://doi.org/10.1021/jo00296a044 -
5
المؤلفون: Michael R. Becker, Simon D.P. Baugh, Michael Voronkov, Kunjian Gu
المصدر: ChemInform. 37
مصطلحات موضوعية: Pyrimidine, business.industry, Organic Chemistry, General Medicine, Modular design, Biochemistry, Combinatorial chemistry, Catalysis, chemistry.chemical_compound, chemistry, Transition metal, Yield (chemistry), Drug Discovery, Organic chemistry, business, Amination
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6
المؤلفون: Sébastien Maignan, Michael R. Becker, Spada Alfred P, Yong Mi Choi-Sledeski, Vincent Mikol, Jean-Pierre Guilloteau, William R. Ewing, Pauls Henry W
المصدر: Journal of medicinal chemistry. 46(5)
مصطلحات موضوعية: chemistry.chemical_classification, Sulfonyl, Models, Molecular, Binding Sites, Serine Proteinase Inhibitors, Molecular model, Molecular Structure, Hydrogen bond, Stereochemistry, Benzamidine, Piperazines, Sulfonamide, Amidine, Piperazine, chemistry.chemical_compound, chemistry, Drug Discovery, Factor Xa, Molecular Medicine, Moiety, Humans, Protein Binding
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7
المؤلفون: Spada Alfred P, Wei He, Stephen M. Condon, Dennis Colussi, Myers Michael R, Christopher J. Burns, Karen Brown, Michael R. Becker, Barbara Hanney, Valeria Chu
المصدر: Bioorganicmedicinal chemistry letters. 12(6)
مصطلحات موضوعية: medicine.drug_mechanism_of_action, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Coagulation Factor Xa, Pharmaceutical Science, Biochemistry, Chemical synthesis, Heterocyclic Compounds, 4 or More Rings, Structure-Activity Relationship, Drug Discovery, medicine, Structure–activity relationship, Animals, Humans, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Quinazoline derivatives, Bicyclic molecule, biology, Chemistry, Organic Chemistry, Kinetics, Enzyme, Enzyme inhibitor, Factor Xa, biology.protein, Molecular Medicine, Benzimidazoles, Factor Xa Inhibitors
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8
المؤلفون: Yong Mi Choi-Sledeski, Stéphanie Pouzieux, and Alfred P. Spada, Sébastien Maignan, Vincent Mikol, William R. Ewing, Pauls Henry W, Michael R. Becker, Klein Scott I, Jean-Pierre Guilloteau
المصدر: Journal of medicinal chemistry. 43(17)
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, Stereochemistry, Protein Conformation, Crystallography, X-Ray, Ligands, Benzamidine, Amidine, chemistry.chemical_compound, Thrombin, Fibrinolytic Agents, Drug Discovery, Hydrolase, medicine, Moiety, Humans, Trypsin, Serine protease, biology, Ligand (biochemistry), Benzamidines, chemistry, Coagulation, Factor Xa, biology.protein, Molecular Medicine, medicine.drug, Factor Xa Inhibitors, Protein Binding
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9
المؤلفون: Salvino Joseph M, Michael R. Becker, Yong Gong, Y.M. Choi-Sledeski, Roderick S. Davis, Henry W. Pauls, Karen D. Brown, Valeria Chu
المصدر: Bioorganicmedicinal chemistry letters. 10(10)
مصطلحات موضوعية: medicine.drug_mechanism_of_action, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Factor Xa Inhibitor, Pharmaceutical Science, Anticoagulants, Biochemistry, Combinatorial chemistry, Pyrrolidinones, chemistry.chemical_compound, Structure-Activity Relationship, Sulfonate, Phase (matter), Drug Discovery, medicine, Molecular Medicine, Combinatorial Chemistry Techniques, Molecular Biology, Polymer supported, Factor Xa Inhibitors
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10
المؤلفون: Charles Kasiewski, Suzanne Morgan, Roderick S. Davis, Robert J. Leadley, Jeff Bostwick, Valeria Chu, Henry W. Pauls, Ewing William R, Karen D. Brown, Cuong Ly, Michael R. Becker, Mason Helen J, Ross Bentley, Y.M. Choi-Sledeski, Dennis J. Colussi, Alfred P. Spada, Aiwen Li
المصدر: Bioorganicmedicinal chemistry letters. 9(18)
مصطلحات موضوعية: Thienopyridine, medicine.drug_mechanism_of_action, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Pharmaceutical Science, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Dogs, In vivo, Drug Discovery, medicine, Structure–activity relationship, Animals, Pyrrolidinones, Molecular Biology, chemistry.chemical_classification, biology, Organic Chemistry, Thrombosis, Sulfonamide, Rats, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Factor Xa Inhibitors