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المؤلفون: Timo Heinrich, Jeyaprakashnarayanan Seenisamy, Beatrix Blume, Jörg Bomke, Michel Calderini, Uwe Eckert, Manja Friese-Hamim, Rainer Kohl, Martin Lehmann, Birgitta Leuthner, Djordje Musil, Felix Rohdich, Frank T. Zenke
المصدر: Journal of medicinal chemistry. 62(10)
مصطلحات موضوعية: Male, Molecular Conformation, Mice, Nude, Antineoplastic Agents, Structure-Activity Relationship, Methionine, Metals, Cell Line, Tumor, Drug Discovery, Human Umbilical Vein Endothelial Cells, Molecular Medicine, Animals, Humans, Methionyl Aminopeptidases, Female, Protease Inhibitors, Cell Proliferation
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المؤلفون: Eugen Merkul, Thorsten Knöchel, David Bruge, Dieter Dorsch, Margarita Wucherer-Plietker, Hans-Peter Buchstaller, Timo Heinrich, Dirk Finsinger, Thomas Müller, Hartmut Greiner, Christina Esdar, Ulrich Grädler, Michel Calderini
المصدر: Bioorganicmedicinal chemistry letters. 26(13)
مصطلحات موضوعية: Models, Molecular, animal structures, Indoles, Clinical Biochemistry, Pharmaceutical Science, Protein Serine-Threonine Kinases, Crystallography, X-Ray, 01 natural sciences, Biochemistry, Structure-Activity Relationship, Drug Discovery, Structure–activity relationship, Potency, Transferase, Humans, Molecular Biology, IC50, Protein Kinase Inhibitors, ADME, Virtual screening, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Kinase, Drug discovery, Chemistry, Organic Chemistry, Pyruvate Dehydrogenase Acetyl-Transferring Kinase, Combinatorial chemistry, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Molecular Medicine
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المؤلفون: Paul Czodrowski, Andree Blaukat, Frank Stieber, Julian Blagg, Djordje Musil, Felix Rohdich, Simon Crumpler, Rosemary Burke, Michael Busch, Kai Schiemann, Sharon Gowan, Michel Calderini, Stephanie Simon, Richard Schneider, Suzanne A. Eccles, Robert TePoele, Maria-Jesus Ortiz-Ruiz, Oliver Poeschke, Trevor Clive Dale, Florence I. Raynaud, Klaus Urbahns, Olajumoke Adeniji-Popoola, Wolfgang Kaufmann, Daniel Schwarz, Klaus Schneider, Aurélie Mallinger, Rahul S. Samant, Christian Rink, Christina Esdar, Mark Stubbs, Dennis Waalboer, Paul Workman, Paul A. Clarke, Dirk Wienke
المصدر: Cancer Research. 76:3025-3025
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Kinase, Wnt signaling pathway, Cancer, Context (language use), Pharmacology, Biology, medicine.disease, MED12, 03 medical and health sciences, 030104 developmental biology, Mediator, Oncology, In vivo, medicine, Cyclin-dependent kinase 8
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::205048a11978c437f58e8b431a90eeaa
https://doi.org/10.1158/1538-7445.am2016-3025