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1دورية أكاديمية
المؤلفون: Jordi Doijen, Koen Temmerman, Christel Van den Eynde, Annick Diels, Nick Van den Broeck, Michiel Van Gool, Inha Heo, Steffen Jaensch, Marleen Zwaagstra, Mayra Diosa Toro, Winston Chiu, Steven De Jonghe, Pieter Leyssen, Denisa Bojkova, Sandra Ciesek, Jindrich Cinatl, Lore Verschueren, Christophe Buyck, Frank Van Kuppeveld, Johan Neyts, Marnix Van Loock, Ellen Van Damme
المصدر: Microorganisms, Vol 11, Iss 3, p 717 (2023)
مصطلحات موضوعية: cathepsin L inhibitor, coronavirus, in vitro, phenotypic screening, SARS-CoV-2, Biology (General), QH301-705.5
وصف الملف: electronic resource
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المؤلفون: Ann Vos, Frederik Jan Rita Rombouts, Andrés A. Trabanco, Daniel Oehlrich, Harrie J.M. Gijsen, Diederik Moechars, Sven Franciscus Anna Van Brandt, Aldo Peschiulli, Gregor James Macdonald, Michel Surkyn, Gary Tresadern, Michiel Van Gool, Nigel E. Austin, Michel Anna Jozef De Cleyn
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: animal structures, Amyloid β, biology, Chemistry, Organic Chemistry, hERG, Pharmacology, Biochemistry, Bioavailability, Piperazine, chemistry.chemical_compound, In vivo, mental disorders, Drug Discovery, biology.protein, Potency, Efflux, Penetrant (biochemical)
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المؤلفون: Sergio A. Alonso de Diego, Daniel Oehlrich, Harrie J.M. Gijsen, Andrés A. Trabanco, Hana Prokopcová, Nigel Austin, Michel Surkyn, Dries Van den Bossche, Frederik J. R. Rombouts, Deborah Dhuyvetter, Gregor James Macdonald, Sven Franciscus Anna Van Brandt, Herman Borghys, Michiel Van Gool, Diederik Moechars, Aránzazu García-Molina, Michel Anna Jozef De Cleyn, Carolina Martinez-Lamenca
المصدر: Journal of Medicinal Chemistry. 61:5292-5303
مصطلحات موضوعية: Male, 0301 basic medicine, ERG1 Potassium Channel, Guinea Pigs, hERG, Drug Evaluation, Preclinical, Administration, Oral, Biological Availability, Mice, Inbred Strains, Pharmacology, Rats, Sprague-Dawley, Amidine, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Dogs, 0302 clinical medicine, Drug Stability, In vivo, Oxazines, Drug Discovery, Animals, Aspartic Acid Endopeptidases, Humans, Structure–activity relationship, Protease Inhibitors, Amyloid beta-Peptides, Cardiovascular safety, biology, Peptide Fragments, Clinical trial, 030104 developmental biology, chemistry, Cardiovascular Diseases, Toxicity, β secretase, biology.protein, Molecular Medicine, Administration, Intravenous, Amyloid Precursor Protein Secretases, Chemical and Drug Induced Liver Injury, 030217 neurology & neurosurgery
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المؤلفون: Marijke Somers, Gregor James Macdonald, Oscar Delgado, Fabrice Jourdan, Sergio A. Alonso de Diego, Michiel Van Gool, Andrés A. Trabanco, Luc Ver Donck
المصدر: ChemMedChem. 12:905-912
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Allosteric modulator, Metabotropic glutamate receptor 5, Chemistry, Organic Chemistry, Allosteric regulation, Glutamate receptor, Biochemistry, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Metabotropic receptor, Drug Discovery, Molecular Medicine, Potency, Structure–activity relationship, General Pharmacology, Toxicology and Pharmaceutics, Metabotropic glutamate receptor 2, 030217 neurology & neurosurgery
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المؤلفون: Sven Franciscus Anna Van Brandt, Aldo Peschiulli, Andrés A. Trabanco, Ann Vos, Nigel Austin, Sergio A. Alonso de Diego, Michel Anna Jozef De Cleyn, Hana Prokopcová, Michel Surkyn, Dieder Moechars, Daniel Oehlrich, Gregor James Macdonald, Frederik J. R. Rombouts, Juan Antonio Vega, Michiel Van Gool, Ana Isabel de Lucas, Harrie J.M. Gijsen, Gary Tresadern
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: 010405 organic chemistry, Organic Chemistry, 01 natural sciences, Biochemistry, Combinatorial chemistry, 0104 chemical sciences, Amidine, Enzyme binding, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, Piperazine, chemistry, Drug Discovery, β secretase, Efflux, IC50
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المؤلفون: Myriam Ciordia, Andrés A. Trabanco, María Sánchez-Roselló, Gary Tresadern, Michiel Van Gool, Natalia Mateu, Laura Pérez-Benito, Santos Fustero, Oscar Delgado
المصدر: Chemistry - A European Journal. 21:11719-11726
مصطلحات موضوعية: Hydrocarbons, Fluorinated, Molecular Structure, Tandem, Amino esters, Drug discovery, Stereochemistry, Organic Chemistry, Amidines, Stereoisomerism, Sequence (biology), General Chemistry, Combinatorial chemistry, Pyrrolidinones, Catalysis, Stereocenter, Amidine, chemistry.chemical_compound, chemistry, Cyclization, Biological property, Drug Discovery, Michael reaction, Aspartic Acid Endopeptidases, Amyloid Precursor Protein Secretases
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المؤلفون: Andrés A. Trabanco, Natalia Mateu, Laura Pérez-Benito, Oscar Delgado, María Sánchez-Roselló, Gary Tresadern, Santos Fustero, Michiel Van Gool, Myriam Ciordia
المصدر: ChemInform. 47
مصطلحات موضوعية: Amidine, chemistry.chemical_compound, Tandem, chemistry, Amino esters, Drug discovery, Biological property, Michael reaction, Sequence (biology), General Medicine, Combinatorial chemistry, Stereocenter
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المؤلفون: Michiel Van Gool, Michel Surkyn, Aránzazu García-Molina, Ann Vos, Nigel Austin, Gary Tresadern, Michel Anna Jozef De Cleyn, Dieder Moechars, Carolina Martinez-Lamenca, Herman Borghys, Daniel Oehlrich, Oscar Delgado, Hana Prokopcová, Gregor James Macdonald, José Manuel Alonso, Sergio A. Alonso de Diego, Harrie J.M. Gijsen, Sven Franciscus Anna Van Brandt, Richard Alexander, Frederik J. R. Rombouts, Andrés A. Trabanco
المصدر: Journal of medicinal chemistry. 58(20)
مصطلحات موضوعية: Male, Models, Molecular, Amyloid, Biological Availability, Pharmacology, Blood–brain barrier, Mice, Dogs, Alzheimer Disease, Cell Line, Tumor, mental disorders, Drug Discovery, Oxazines, medicine, Animals, Aspartic Acid Endopeptidases, Cytochrome P-450 Enzyme Inhibitors, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, P-glycoprotein, chemistry.chemical_classification, Amyloid beta-Peptides, biology, Brain, Blood Proteins, In vitro, Enzyme, medicine.anatomical_structure, chemistry, Biochemistry, Blood-Brain Barrier, Drug Design, biology.protein, Molecular Medicine, Female, Efflux, Amyloid Precursor Protein Secretases, Amyloid precursor protein secretase, Protein Binding
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المؤلفون: Harrie J.M. Gijsen, Richard Alexander, Frederik J. R. Rombouts, Juan Antonio Vega, Oscar Delgado, Gregor James Macdonald, John Spurlino, Andrés A. Trabanco, Michiel Van Gool, Gary Tresadern, Dieder Moechars, Francisca Delgado
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:7255-7260
مصطلحات موضوعية: Prioritization, Amyloid, Amyloid beta, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Crystal structure, Biochemistry, Piperazines, chemistry.chemical_compound, In vivo, Amide, Drug Discovery, Computer Simulation, Enzyme Inhibitors, Molecular Biology, Binding Sites, biology, Chemistry, Organic Chemistry, Rational design, Stereoisomerism, Combinatorial chemistry, Protein Structure, Tertiary, Enzyme Activation, Drug Design, biology.protein, β secretase, Molecular Medicine, Amyloid Precursor Protein Secretases
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المؤلفون: Michiel Van Gool, Francisca Delgado, Oscar Delgado, Carlos M. Martínez-Viturro, Miguel Ángel Pena, Sergio A. Alonso de Diego, Greet Vanhoof, Marta Artola, Gregor James Macdonald, José Manuel Bartolomé-Nebreda, María Luz Martín-Martín, Xavier Langlois, José Manuel Alonso, Han Min Tong, Susana Conde-Ceide, Anton Megens, Marijke Somers, Alberto Fontana
مصطلحات موضوعية: Chemistry, Phosphodiesterase Inhibitors, Phosphoric Diester Hydrolases, Phosphodiesterase, Administration, Oral, Biological Availability, Pharmacology, Bioavailability, Rats, Disease Models, Animal, Structure-Activity Relationship, Pharmacokinetics, In vivo, Drug Discovery, Animal models of schizophrenia, Schizophrenia, Molecular Medicine, Animals, PDE10A, Rats, Wistar
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::752a138a2d02674e482528380d513b5e
https://hdl.handle.net/1887/3203217