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المؤلفون: Daigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe, Kouichi Yoshinari
المصدر: Drug Metabolism and Disposition. 50:235-242
مصطلحات موضوعية: Pharmacology, Pharmaceutical Science
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::70186cea69d28e89cf0b2a4873bd0d31
https://doi.org/10.1124/dmd.121.000665 -
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المؤلفون: Daisuke Nakai, Miho Kazui, Tomoko Ishizuka, Hidetaka Sakurai, Yumi Nishiya, Eiko Suzuki
المصدر: Drug Metabolism and Pharmacokinetics. 35:45-55
مصطلحات موضوعية: Pharmacology, Hydrolases, Chemistry, Valproic Acid, Alcohol Dehydrogenase, Phosphatidate Phosphatase, Pharmaceutical Science, Disposition, Metabolism, Prodrug, Drug interaction, Pyrrolidinones, Carbapenems, Quinolines, Animals, Humans, Drug Interactions, Prodrugs, Pharmacology (medical), Identification (biology), P450 Enzymes, Carboxylic Ester Hydrolases, Prasugrel Hydrochloride, Peptide Hydrolases
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3
المؤلفون: Daigo, Asano, Syoya, Hamaue, Hamim, Zahir, Hideyuki, Shiozawa, Yumi, Nishiya, Takako, Kimura, Miho, Kazui, Naotoshi, Yamamura, Marie, Ikeguchi, Takahiro, Shibayama, Shin-Ichi, Inoue, Tsuyoshi, Shinozuka, Toshiyuki, Watanabe, Chizuko, Yahara, Nobuaki, Watanabe, Kouichi, Yoshinari
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 50(3)
مصطلحات موضوعية: Aldehyde Oxidase, Cytochrome P-450 CYP2C8, Sulfonamides, Pyrimidines, Cytochrome P-450 Enzyme System, Microsomes, Liver, Animals, Humans, Pyrazoles
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::962904c1c9cdbb5aff75655771821958
https://pubmed.ncbi.nlm.nih.gov/34930785 -
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المؤلفون: Miho Kazui, Naoki Miyoshi, Ken Sakurai, Jun Kobayashi, Keisuke Motoyama, Tomoko Sakakura, Tsutomu Nagata, Akifumi Nakamura
المصدر: Bioorganicmedicinal chemistry letters. 28(12)
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Administration, Oral, Biological Availability, Biochemistry, TRPC6, 03 medical and health sciences, Transient receptor potential channel, chemistry.chemical_compound, Mice, Structure-Activity Relationship, 0302 clinical medicine, Drug Discovery, TRPC6 Cation Channel, Animals, Humans, Molecular Biology, IC50, biology, Bicyclic molecule, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, Calcium Channel Blockers, 030104 developmental biology, chemistry, Indans, biology.protein, Microsomes, Liver, Molecular Medicine, Nonane, Selectivity, 030217 neurology & neurosurgery, Derivative (chemistry)
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المؤلفون: Hidetaka Sakurai, Ryoko Sawamura, Takashi Izumi, Atsushi Kurihara, Naoya Wada, Akira Shinagawa, Miho Kazui, Tomoyo Honda, Yumi Nishiya
المصدر: Biopharmaceutics & Drug Disposition. 36:352-363
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Chemistry, Pharmaceutical Science, Human skin, General Medicine, Loxoprofen, In vitro, Enzyme, Biochemistry, Pharmacokinetics, Oral administration, medicine, Pharmacology (medical), Active metabolite, medicine.drug, Transdermal
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المؤلفون: Osamu Ando, Miho Kazui, Takashi Izumi, Katsunobu Hagihara, Toshihiko Ikeda, Atsushi Kurihara
المصدر: Drug Delivery System. 30:454-464
مصطلحات موضوعية: Prasugrel, Thienopyridine, P2Y12 Receptor Antagonists, Chemistry, medicine, Pharmaceutical Science, Prodrug, Pharmacology, Clopidogrel, Active metabolite, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::be2a275a62e8484c34041d0fbc402750
https://doi.org/10.2745/dds.30.454 -
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المؤلفون: Hidenori Ikenaga, Toshihiko Ikeda, Toshihiko Nanba, Atsushi Kurihara, Katsunobu Hagihara, Miho Kazui, Kiichi Fusegawa, Takashi Izumi
المصدر: Drug Metabolism and Disposition. 39:565-570
مصطلحات موضوعية: Male, Prasugrel, Metabolite, Pharmaceutical Science, Thiophenes, Pharmacology, Piperazines, Acetic acid, chemistry.chemical_compound, Dogs, Cytochrome P-450 Enzyme System, In vivo, Microsomes, medicine, Thiolactone, Animals, Humans, Intestinal Mucosa, Active metabolite, Prasugrel Hydrochloride, Hydrolysis, Liver, chemistry, Area Under Curve, Microsomes, Liver, Microsome, Oxidation-Reduction, Platelet Aggregation Inhibitors, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cc041e08e9f05ceb736a75db196b2d5b
https://doi.org/10.1124/dmd.110.035956 -
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المصدر: Drug Metabolism and Disposition. 39:208-214
مصطلحات موضوعية: Thienopyridine, Stereochemistry, Metabolite, Blotting, Western, Pharmaceutical Science, Thiophenes, In Vitro Techniques, Piperazines, chemistry.chemical_compound, Cytosol, Thioredoxins, Tandem Mass Spectrometry, Glutaredoxin, Humans, Biotransformation, Glutaredoxins, Active metabolite, Pharmacology, Antibodies, Monoclonal, Glutathione, Thienopyridine Antiplatelet Agent, Liver, chemistry, Biochemistry, Chromatography, Gel, Microsomes, Liver, Platelet aggregation inhibitor, Thioredoxin, Prasugrel Hydrochloride, Platelet Aggregation Inhibitors
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1ba52932bcf2069747dee8efe9cff0e9
https://doi.org/10.1124/dmd.110.035196 -
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المؤلفون: Miho Kazui, Osamu Okazaki, Nagy A. Farid, Katsunobu Hagihara, Atsushi Kurihara, Kokichi Honda, Toshihiko Ikeda, Michiharu Yoshiike
المصدر: Drug Metabolism and Disposition. 37:2145-2152
مصطلحات موضوعية: Ticlopidine, Prasugrel, Thienopyridine, Pyridines, Metabolite, Pharmaceutical Science, Thiophenes, CYP2C19, Pharmacology, Piperazines, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, medicine, Thiolactone, Humans, cardiovascular diseases, Active metabolite, Prasugrel Hydrochloride, Chemistry, Genetic Variation, Clopidogrel, Microsomes, Liver, Platelet Aggregation Inhibitors, circulatory and respiratory physiology, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1afbba98628c128595467d1ff1fbcc86
https://doi.org/10.1124/dmd.109.028498 -
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المؤلفون: Hidenori Ikenaga, T. Nanba, T. Ikeda, Miho Kazui, Katsunobu Hagihara, Atsushi Kurihara, Osamu Okazaki, Masayuki Takahashi, Keiichi Fusegawa, N. A Farid
المصدر: Xenobiotica. 39:218-226
مصطلحات موضوعية: Male, Ticlopidine, Prasugrel, Thienopyridine, Health, Toxicology and Mutagenesis, Thiophenes, Pharmacology, Toxicology, Biochemistry, Piperazines, Rats, Sprague-Dawley, chemistry.chemical_compound, Dogs, Cytochrome P-450 Enzyme System, Oral administration, medicine, Thiolactone, Animals, cardiovascular diseases, Active metabolite, Molecular Structure, Hydrolysis, General Medicine, Prodrug, Clopidogrel, Rats, chemistry, Area Under Curve, Platelet aggregation inhibitor, Oxidation-Reduction, Prasugrel Hydrochloride, Platelet Aggregation Inhibitors, medicine.drug