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1دورية أكاديمية
المصدر: F1000Research, Vol 6 (2017)
مصطلحات موضوعية: Cancer Therapeutics, Cell Growth & Division, Cellular Death & Stress Responses, Drug Discovery & Design, Molecular Pharmacology, Medicine, Science
وصف الملف: electronic resource
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المؤلفون: Kristiina Vuori, Nicholas D.P. Cosford, John C. Reed, Kate Welsh, Curt T. Hauser, Trina R. Cooley, Ying Su, Hongbin Yuan, Santhi Reddy Ganji, Robert J. Ardecky, Marcos González-López, Mitchell Vamos, Darren Finlay
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4f12185c74bb597eff8220a84448b54e
https://doi.org/10.1158/1535-7163.22503459.v1 -
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المؤلفون: Kristiina Vuori, Nicholas D.P. Cosford, John C. Reed, Kate Welsh, Curt T. Hauser, Trina R. Cooley, Ying Su, Hongbin Yuan, Santhi Reddy Ganji, Robert J. Ardecky, Marcos González-López, Mitchell Vamos, Darren Finlay
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0973df3f26c30eec6ca1ebd86e91a52b
https://doi.org/10.1158/1535-7163.22503462 -
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المؤلفون: Nicole A Bakas, Lester J. Lambert, Nicholas D. P. Cosford, Mitchell Vamos, Huiyu Ren, Apirat Chaikuad, Reuben J. Shaw, Carina Wimer, Maria Celeridad, Douglas J. Sheffler, Lutz Tautz, Sonja N. Brun, Allison S. Limpert, Stefan Knapp
المصدر: J Med Chem
مصطلحات موضوعية: Cell Survival, Poly ADP ribose polymerase, Antineoplastic Agents, Apoptosis, Triple Negative Breast Neoplasms, Poly(ADP-ribose) Polymerase Inhibitors, Protein Serine-Threonine Kinases, Article, Piperazines, Olaparib, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, Autophagy, Animals, Autophagy-Related Protein-1 Homolog, Humans, Protein Kinase Inhibitors, Triple-negative breast cancer, Cell Proliferation, Kinase, HEK 293 cells, Intracellular Signaling Peptides and Proteins, Drug Synergism, Mice, Inbred C57BL, HEK293 Cells, Pyrimidines, chemistry, Cell culture, PARP inhibitor, Cancer research, Molecular Medicine, Phthalazines, Female, Drug Screening Assays, Antitumor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::64e4b2f1d43e7a3f43e170153e08bf32
https://europepmc.org/articles/PMC8064294/ -
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المؤلفون: Laura J. Martins, Lars Pache, Peter Teriete, John M. Marlett, Ana M. Maestre, Viviana Simon, Miriam S. Dutra, Frederic D. Bushman, Young Hwang, Sumit K. Chanda, John A. T. Young, Lara Manganaro, Adam M. Spivak, Nicholas D. P. Cosford, Mitchell Vamos, Alberto Bosque, Ana Fernandez-Sesma, Vicente Planelles, Renate König, Jeffrey P. Murry
المصدر: Cell Host & Microbe. 18:345-353
مصطلحات موضوعية: Cancer Research, medicine.drug_class, Histone deacetylase inhibitor, Virus Activation, Repressor, Biology, medicine.disease, Microbiology, Virology, 3. Good health, Ubiquitin ligase, chemistry.chemical_compound, chemistry, Transcription (biology), Immunology and Microbiology(all), Panobinostat, Virus latency, medicine, biology.protein, Cancer research, Parasitology, Molecular Biology, Viral load
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المؤلفون: Reuben J. Shaw, Dhanya Raveendra-Panickar, Nicholas D. P. Cosford, Chih-Cheng Yang, Douglas J. Sheffler, Haixia Zou, Juan Rong, Daniel F. Egan, Peter Teriete, Benjamin E. Turk, Hua Jane Lou, Mitchell Vamos, Chad J. Miller, John M. Asara, Matthew G. H. Chun
المصدر: Molecular Cell. 59(2):285-297
مصطلحات موضوعية: Atg1, Cell Survival, Molecular Sequence Data, Protein Serine-Threonine Kinases, Substrate Specificity, Gene Knockout Techniques, Mice, Catalytic Domain, Consensus Sequence, Autophagy, Animals, Autophagy-Related Protein-1 Homolog, Humans, Amino Acid Sequence, Phosphorylation, RNA, Small Interfering, Mechanistic target of rapamycin, Protein Kinase Inhibitors, Molecular Biology, PI3K/AKT/mTOR pathway, Cells, Cultured, biology, Intracellular Signaling Peptides and Proteins, ULK2, Cell Biology, ULK1, Recombinant Proteins, HEK293 Cells, Pyrimidines, Benzamides, Cancer research, biology.protein
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المؤلفون: Nicholas D. P. Cosford, Mitchell Vamos
المصدر: The Journal of Organic Chemistry. 79:2274-2280
مصطلحات موضوعية: In situ, Cyanides, Molecular Structure, Pyridines, Chemistry, Organic Chemistry, Aminopyridines, Combinatorial chemistry, Article, chemistry.chemical_compound, Pyridine, Molecule, Organic chemistry
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المؤلفون: John C. Reed, Curt T. Hauser, Marcos González-López, Robert Ardecky, Kate Welsh, Nicholas D. P. Cosford, Hongbin Yuan, Darren Finlay, Trina R. Cooley, Kristiina Vuori, Ying Su, Mitchell Vamos, Santhi Ganji
المصدر: Molecular Cancer Therapeutics. 13:5-15
مصطلحات موضوعية: Cancer Research, Ubiquitin-Protein Ligases, Antineoplastic Agents, Apoptosis, X-Linked Inhibitor of Apoptosis Protein, Biology, Inhibitor of apoptosis, Article, Inhibitor of Apoptosis Proteins, Small Molecule Libraries, TNF-Related Apoptosis-Inducing Ligand, Cell Line, Tumor, Neoplasms, Baculoviral IAP Repeat-Containing 3 Protein, Humans, Molecular Targeted Therapy, Cytotoxicity, Inhibitor of apoptosis domain, Caspase 8, Cell biology, XIAP, Oncology, Drug Resistance, Neoplasm, Cancer cell, Tumor necrosis factor alpha, Signal Transduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dbf4fab71c8beb7ad98221a86a40df06
https://doi.org/10.1158/1535-7163.mct-13-0153 -
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المؤلفون: Sheridan J. S. Carrington, Nicholas D. P. Cosford, P. Jeffrey Conn, Colleen M. Niswender, Ryan D. Morrison, Douglas J. Sheffler, Anna L. Blobaum, Kiran Gogi, Shaun R. Stauffer, Joshua A. Bruner, Paige N. Vinson, J. Scott Daniels, Cody J. Wenthur, Mitchell Vamos, Craig W. Lindsley
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:3921-3925
مصطلحات موضوعية: Central Nervous System, animal structures, Allosteric modulator, Receptor, Metabotropic Glutamate 5, Clinical Biochemistry, Allosteric regulation, Glutamic Acid, Pharmaceutical Science, Pharmacology, Receptors, Metabotropic Glutamate, Sensitivity and Specificity, Biochemistry, Article, Permeability, Cell Line, Structure-Activity Relationship, chemistry.chemical_compound, Allosteric Regulation, Piperidines, Drug Discovery, Humans, Structure–activity relationship, Receptor, Molecular Biology, health care economics and organizations, Chemistry, Drug discovery, Organic Chemistry, food and beverages, Liver metabolism, Molecular Probes, Microsomes, Liver, Molecular Medicine, Metabotropic glutamate receptor 3, Penetrant (biochemical)
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المؤلفون: Mitchell Vamos, Yoshihisa Kobayashi
المصدر: Tetrahedron. 65:5899-5903
مصطلحات موضوعية: chemistry.chemical_classification, Stereochemistry, Organic Chemistry, Biochemistry, Chemical synthesis, Propellane, chemistry.chemical_compound, chemistry, Drug Discovery, Ugi reaction, Stereoselectivity, Pyroglutamic acid, Salinosporamide A, Derivative (chemistry), Lactone