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1
المؤلفون: Miyako Masubuchi, Tatsuya Ito
المصدر: The Journal of Antibiotics. 67:353-360
مصطلحات موضوعية: DNA Replication, Pharmacology, Biological Products, Magnetic Resonance Spectroscopy, Natural product, Chromatography, Bacteria, Fungi, Biology, Mass Spectrometry, Anti-Bacterial Agents, High-Throughput Screening Assays, chemistry.chemical_compound, chemistry, Fermentation, Drug Discovery, Biologically active substances, Ultra high performance, Chromatography, High Pressure Liquid, Gene Library
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2
المؤلفون: Yasuhiko Shiratori, Hirosato Ebiike, Takaaki A. Fukami, Masahiro Sakaitani, Toshiyuki Tsukaguchi, Yuko Aoki, Nobuya Ishii, Kohsuke Asoh, Kenichi Kawasaki, Tatsuo Ohtsuka, Miyako Masubuchi, Nobuo Shimma, Osamu Kondoh, Ikumi Hyoudoh, Masami Kohchi
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:1753-1757
مصطلحات موضوعية: Chemistry, Pharmaceutical, Farnesyltransferase, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Quinolones, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Animals, Farnesyltranstransferase, Humans, Enzyme Inhibitors, Benzofuran, Molecular Biology, Benzofurans, chemistry.chemical_classification, Farnesyl-diphosphate farnesyltransferase, biology, Chemistry, Organic Chemistry, In vitro, Enzyme, Drug Design, biology.protein, Molecular Medicine, Tipifarnib, Drug Screening Assays, Antitumor, Neoplasm Transplantation, medicine.drug
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3
المؤلفون: Hidetoshi Shindoh, Michiko Hayase, Yuko Aoki, Shinji Tsujii, Hirosato Ebiike, Kenichi Kawasaki, Miyako Masubuchi, Tatsuo Ohtsuka, Yasuhiko Shiratori, Kenji Morikami, Kiyoaki Sakata, Satoshi Sogabe, Nobuo Shimma, Toshihiko Fujii
المصدر: Bioorganic & Medicinal Chemistry. 11:4463-4478
مصطلحات موضوعية: Male, Antifungal Agents, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Fungal Proteins, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Drug Resistance, Fungal, In vivo, Candida albicans, Drug Discovery, Animals, Structure–activity relationship, Enzyme Inhibitors, Benzofuran, Molecular Biology, Benzofurans, Fungal protein, biology, Organic Chemistry, Candidiasis, Fungal genetics, biology.organism_classification, Rats, Inbred F344, Rats, chemistry, Drug Design, Molecular Medicine, Lead compound, Acyltransferases, Protein Binding
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4
المؤلفون: Kenji Morikami, Kenichi Kawasaki, Satoshi Sogabe, Nobuo Shimma, Pingli Liu, Toshihiko Fujii, Yuko Aoki, Miyako Masubuchi, Tatsuo Ohtsuka, Yasuhiko Shiratori, Kiyoaki Sakata, Michiko Hayase, Hirosato Ebiike, Hidetoshi Shindoh
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:607-610
مصطلحات موضوعية: Drug, Antifungal Agents, media_common.quotation_subject, Clinical Biochemistry, Pharmaceutical Science, Computational biology, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Candida albicans, Drug Discovery, medicine, Animals, Humans, Benzofuran, Molecular Biology, Benzofurans, media_common, biology, Organic Chemistry, Candidiasis, medicine.disease, biology.organism_classification, Rats, Inbred F344, In vitro, Rats, Disease Models, Animal, chemistry, Area Under Curve, Drug Design, Molecular Medicine, Systemic candidiasis, Acyltransferases, Fluconazole, Protein Binding, medicine.drug
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5
المؤلفون: Hans Senn, Kiyoaki Sakata, Miyako Masubuchi, Alfred Ross, Werner Klaus, Takaaki Miura
المصدر: European Journal of Biochemistry. 268:4833-4841
مصطلحات موضوعية: biology, Ligand, Chemistry, Stereochemistry, Active site, Plasma protein binding, Nuclear magnetic resonance spectroscopy, Biochemistry, Crystallography, biology.protein, Molecule, Enantiomer, Bovine serum albumin, Ternary complex
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6
المؤلفون: Kiyoaki Sakata, Yoshihiko Ikeda, Nobuo Shimma, Shinji Tsujii, Yasuhiko Shiratori, Toshihiko Fujii, Kenichi Kawasaki, Hirosato Ebiike, Miyako Masubuchi, Tatsuo Ohtsuka, Satoshi Sogabe, Yuko Aoki
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:1833-1837
مصطلحات موضوعية: Antifungal Agents, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Species Specificity, Candida albicans, Receptors, Adrenergic, beta, Drug Discovery, Humans, Molecular Biology, Benzofurans, chemistry.chemical_classification, Bicyclic molecule, biology, Organic Chemistry, biology.organism_classification, Corpus albicans, In vitro, Enzyme, chemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Lead compound, Acyltransferases
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7
المؤلفون: Mikako Fujimori, Junko Watanabe, Miyako Masubuchi, Aya Nishio, Yumiko Nakamura, Fumiko Kawahara, Naoki Nakada, Shoko Matsukuma, Tsutomu Kamiyama, Kayoko Yamaji
المصدر: The Journal of Antibiotics. 50:402-411
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Molecular Structure, biology, Tetrapeptide, Stereochemistry, Stereoisomerism, Peptide, Isomerase, biology.organism_classification, Peptides, Cyclic, DNA gyrase, Streptomyces, Structure-Activity Relationship, Enzyme, chemistry, Biochemistry, Enzyme inhibitor, Drug Discovery, biology.protein, Topoisomerase II Inhibitors, Actinomycetales, Enzyme Inhibitors, Chromatography, High Pressure Liquid, Antibacterial agent
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a4a1c7d048215a6fed0a7c0c94da9b0f
https://doi.org/10.7164/antibiotics.50.402 -
8
المؤلفون: Kohichi Okamato, Miyako Masubuchi, Nobuo Shimma, Fumio Watanabe, Tadakatsu Hayase, Takeshi Murata, Takuo Tsukuda, Masahiro Aoki, Hiroshi Fukuda, Hidetoshi Shindoh, Susumu Komiyama, Kenichi Kawasaki, Masayuki Sudoh, Hiroshi Sakamoto, Kouhei Koyama, Atsunori Ohta, Asao Katsume, Yasuaki Matsubara, Yuko Aoki
المصدر: Bioorganicmedicinal chemistry letters. 23(1)
مصطلحات موضوعية: Cell Survival, Hepatitis C virus, Hepacivirus, Clinical Biochemistry, Pharmaceutical Science, medicine.disease_cause, Virus Replication, Biochemistry, Antiviral Agents, Cell Line, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Structure–activity relationship, Animals, Humans, Citrates, Molecular Biology, Natural product, biology, Phenylpropionates, Chemistry, Organic Chemistry, Enantioselective synthesis, Total synthesis, Stereoisomerism, biology.organism_classification, Virology, Rats, Viral replication, Cell culture, Molecular Medicine, Half-Life
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9
المؤلفون: Tsutomu Kamiyama, K. Yamaji, Miyako Masubuchi, J. Watanabe, F. Kawahara, Naoki Nakada, Shoko Matsukuma, A. Nishio, M. Fujimori, Yumiko Nakamura
المصدر: ChemInform. 28
مصطلحات موضوعية: Biochemistry, Chemistry, medicine.drug_class, Antibiotics, medicine, General Medicine, DNA Gyrase Inhibitors, Cyclothialidine
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10
المؤلفون: Kiyoaki Sakata, Kenichi Kawasaki, Michiko Hayase, Hirosato Ebiike, Hidetoshi Shindoh, Tsunehisa Aoyama, Satoshi Sogabe, Kenji Morikami, Nobuo Shimma, Toshihiko Fujii, Yasuhiko Shiratori, Miyako Masubuchi, Tatsuo Ohtsuka, Satoshi Niizuma, Yuko Aoki
المصدر: Bioorganicmedicinal chemistry letters. 13(1)
مصطلحات موضوعية: Models, Molecular, Antifungal Agents, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Ether, Biochemistry, Chemical synthesis, Fungal Proteins, chemistry.chemical_compound, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, Drug Stability, Drug Discovery, Candida albicans, medicine, Structure–activity relationship, Animals, Enzyme Inhibitors, Molecular Biology, Benzofurans, biology, Aryl, Organic Chemistry, Biological activity, medicine.disease, biology.organism_classification, Disease Models, Animal, chemistry, Drug Design, Molecular Medicine, Systemic candidiasis, Derivative (chemistry), Acyltransferases