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1
المؤلفون: Minoru Tomida, Kosuke Anan, Shoichi Yamamoto, Shunji Shinohara, Aya Tazawa, Nobuyoshi Hasebe, Shigenori Yagi, Masaharu Kume, Shinji Shimada, Yoshihiro Haga, Moriyasu Masui, Hiroyuki Kai, Hiroki Tsuji
المصدر: Bioorganic & Medicinal Chemistry Letters. 29:1143-1147
مصطلحات موضوعية: Male, Clinical Biochemistry, Analgesic, Pharmaceutical Science, Pharmacology, Receptors, N-Methyl-D-Aspartate, 01 natural sciences, Biochemistry, Rats, Sprague-Dawley, Structure-Activity Relationship, chemistry.chemical_compound, Pharmacokinetics, Drug Discovery, Animals, Isoxazole, Molecular Biology, Analgesics, Molecular Structure, 010405 organic chemistry, Organic Chemistry, Antagonist, Rats, 0104 chemical sciences, Bioavailability, 010404 medicinal & biomolecular chemistry, chemistry, Drug Design, Neuropathic pain, Molecular Medicine, NMDA receptor, Derivative (chemistry)
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2
المؤلفون: Naoki Miyake, You Adachi, Yoshihide Sugata, Fumiya Ikarashi, Shin-Ichiro Hara, Yukihito Sumino, Kazuya Okamoto, Tatsuro Yasukata, Moriyasu Masui, Takanori Kurita, Masahiko Nagai
المصدر: Organic Process Research & Development. 23:565-570
مصطلحات موضوعية: chemistry.chemical_compound, Scale (ratio), 010405 organic chemistry, Chemistry, Organic Chemistry, food and beverages, Dolutegravir sodium, Physical and Theoretical Chemistry, 010402 general chemistry, 01 natural sciences, Combinatorial chemistry, Pyrone, 0104 chemical sciences
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3
المؤلفون: Shuhei Yoshida, Ken-ichi Kusakabe, Moriyasu Masui, Kouki Fuchino
المصدر: Tetrahedron Letters. 64:152684
مصطلحات موضوعية: Scaffold, 010405 organic chemistry, Chemistry, Organic Chemistry, Burgess reagent, 010402 general chemistry, 01 natural sciences, Biochemistry, 0104 chemical sciences, chemistry.chemical_compound, Acetoxy group, Reagent, Drug Discovery, Organic chemistry, Phosphorus pentoxide
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4
المؤلفون: Yasuyoshi Iso, Harrie J.M. Gijsen, Gaku Sakaguchi, Shuhei Yoshida, Deborah Dhuyvetter, Yasunori Mitsuoka, Shigeru Ando, Shuichi Hiroyama, Yoshinori Yamano, Kiyotaka Koyabu, Moriyasu Masui, Herman Borghys, Yasuto Kido, Noriyuki Kurose, Motoko Hosono, Masayoshi Ogawa, Hisanori Ito, Chie Unemura, Shuichi Ohnishi, Takahiko Yamamoto, Ken-ichi Kusakabe, Kazuo Komano, Hirofumi Miyajima, Tamio Fukushima, Kouki Fuchino
المصدر: Journal of medicinal chemistry. 61(12)
مصطلحات موضوعية: ERG1 Potassium Channel, ATP Binding Cassette Transporter, Subfamily B, hERG, Guinea Pigs, ATP-binding cassette transporter, Oxazines, Pharmacology, Crystallography, X-Ray, 01 natural sciences, Madin Darby Canine Kidney Cells, 03 medical and health sciences, Structure-Activity Relationship, 0302 clinical medicine, Dogs, Drug Discovery, Structure–activity relationship, Animals, Aspartic Acid Endopeptidases, Humans, Protease Inhibitors, ATP Binding Cassette Transporter, Subfamily B, Member 1, chemistry.chemical_classification, Mice, Knockout, Amyloid beta-Peptides, biology, 010405 organic chemistry, Rational design, Brain, Peptide Fragments, 0104 chemical sciences, Mice, Inbred C57BL, chemistry, Drug Design, Knockout mouse, biology.protein, Molecular Medicine, Efflux, Amyloid Precursor Protein Secretases, Amyloid precursor protein secretase, 030217 neurology & neurosurgery
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5
المؤلفون: Nobuyoshi Hasebe, Hiroyuki Kai, Kosuke Anan, Shigenori Yagi, Shunji Shinohara, Shinji Shimada, Miho Ohara, Moriyasu Masui, Masaharu Kume, Hiroki Tsuji, Shoichi Yamamoto, Shin-Ichiro Hara
المصدر: Bioorganicmedicinal chemistry letters. 27(17)
مصطلحات موضوعية: 0301 basic medicine, Clinical Biochemistry, Analgesic, Central nervous system, Cyclohexanol, Pharmaceutical Science, Administration, Oral, Pain, Pharmacology, 030226 pharmacology & pharmacy, Biochemistry, Receptors, N-Methyl-D-Aspartate, 03 medical and health sciences, chemistry.chemical_compound, Mice, Structure-Activity Relationship, 0302 clinical medicine, Pharmacokinetics, Formaldehyde, Drug Discovery, medicine, Distribution (pharmacology), Animals, Humans, Isoxazole, Receptor, Molecular Biology, Analgesics, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, Brain, Cyclohexanols, Rats, 030104 developmental biology, medicine.anatomical_structure, HEK293 Cells, nervous system, chemistry, Molecular Medicine, NMDA receptor
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6
المؤلفون: Moriyasu Masui, Marek P. Krzemiński
المصدر: e-EROS Encyclopedia of Reagents for Organic Synthesis
مصطلحات موضوعية: Hexane, chemistry.chemical_compound, Potassium permanganate, Hydroxylamine, Enantiopure drug, chemistry, Reagent, Organic chemistry, Stereoselectivity, Enantiomeric excess, Oxime, Medicinal chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::29461f595d0f9cee2e3f2e4a881f304a
https://doi.org/10.1002/047084289x.rn00063.pub2 -
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المؤلفون: Takayuki Shioiri, Moriyasu Masui
المصدر: Tetrahedron Letters. 39:5195-5198
مصطلحات موضوعية: Reduction (complexity), chemistry.chemical_compound, Chemistry, Trimethyl borate, Reagent, Organic Chemistry, Drug Discovery, Organic chemistry, Stereoselectivity, Borane, Biochemistry
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8
المؤلفون: Takayuki Shioiri, Moriyasu Masui
المصدر: Tetrahedron. 51:8363-8370
مصطلحات موضوعية: Pinene, chemistry.chemical_compound, chemistry, Stereochemistry, Yield (chemistry), Organic Chemistry, Drug Discovery, Organic chemistry, Biochemistry
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9
المؤلفون: Takayuki Shioiri, Moriyasu Masui
المصدر: ChemInform. 26
مصطلحات موضوعية: Terpene, Pinene, chemistry.chemical_compound, Chemistry, Yield (chemistry), Organic chemistry, General Medicine
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المؤلفون: Moriyasu Masui, Takayuki Shioiri
المصدر: ChemInform. 27
مصطلحات موضوعية: Reduction (complexity), Pinene, chemistry.chemical_compound, chemistry, Organic chemistry, General Medicine, Borane