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1دورية أكاديمية
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2دورية أكاديمية
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3دورية أكاديمية
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4دورية أكاديمية
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5دورية أكاديمية
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6دورية أكاديمية
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7دورية أكاديمية
المؤلفون: Lampe JW; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Alford JS; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Boriak-Sjodin PA; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Brach D; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Cosmopoulos K; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Duncan KW; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Eckley ST; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Foley MA; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Harvey DM; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Motwani V; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Munchhof MJ; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Raimondi A; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Riera TV; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Tang C; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Thomenius MJ; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Totman J; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States., Farrow NA; Epizyme Inc., 400 Technology Square, Fourth Floor, Cambridge, Massachusetts 02139, United States.
المصدر: ACS medicinal chemistry letters [ACS Med Chem Lett] 2021 Aug 24; Vol. 12 (10), pp. 1539-1545. Date of Electronic Publication: 2021 Aug 24 (Print Publication: 2021).
نوع المنشور: Journal Article
بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
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8دورية أكاديمية
المؤلفون: Rioux N, Duncan KW, Lantz RJ, Miao X, Chan-Penebre E, Moyer MP, Munchhof MJ, Copeland RA, Chesworth R, Waters NJ
المصدر: Xenobiotica; the fate of foreign compounds in biological systems [Xenobiotica] 2016; Vol. 46 (3), pp. 268-77.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Informa Healthcare Country of Publication: England NLM ID: 1306665 Publication Model: Print Cited Medium: Internet ISSN: 1366-5928 (Electronic) Linking ISSN: 00498254 NLM ISO Abbreviation: Xenobiotica Subsets: MEDLINE
مواضيع طبية MeSH: Enzyme Inhibitors/*pharmacokinetics , Ethers, Cyclic/*pharmacokinetics , Isoquinolines/*pharmacokinetics , Protein-Arginine N-Methyltransferases/*antagonists & inhibitors , Pyrimidines/*pharmacokinetics, Animals ; Cytochrome P-450 CYP2D6 Inhibitors/pharmacokinetics ; Cytochrome P-450 CYP3A Inhibitors/pharmacokinetics ; Dogs ; Hepatocytes/metabolism ; Humans ; Ketoconazole/pharmacokinetics ; Male ; Mice ; Microsomes, Liver/metabolism ; Quinidine/pharmacokinetics ; Rats ; Rats, Sprague-Dawley ; Species Specificity
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9دورية أكاديمية
المؤلفون: Duncan KW; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Rioux N; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Boriack-Sjodin PA; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Munchhof MJ; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Reiter LA; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Majer CR; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Jin L; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Johnston LD; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Chan-Penebre E; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Kuplast KG; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Porter Scott M; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Pollock RM; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Waters NJ; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Smith JJ; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Moyer MP; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Copeland RA; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States., Chesworth R; Epizyme, Inc. , 400 Technology Square, Cambridge, Massachusetts 02139, United States.
المصدر: ACS medicinal chemistry letters [ACS Med Chem Lett] 2015 Dec 02; Vol. 7 (2), pp. 162-6. Date of Electronic Publication: 2015 Dec 02 (Print Publication: 2016).
نوع المنشور: Journal Article
بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
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10دورية أكاديمية
المؤلفون: Chan-Penebre E; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Kuplast KG; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Majer CR; Warp Drive Bio, Cambridge, Massachusetts, USA., Boriack-Sjodin PA; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Wigle TJ; Warp Drive Bio, Cambridge, Massachusetts, USA., Johnston LD; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Rioux N; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Munchhof MJ; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Jin L; Agile Biostructure Solutions, Cambridge, Massachusetts, USA., Jacques SL; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., West KA; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Lingaraj T; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Stickland K; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Ribich SA; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Raimondi A; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Scott MP; Genentech, San Francisco, California, USA., Waters NJ; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Pollock RM; Warp Drive Bio, Cambridge, Massachusetts, USA., Smith JJ; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Barbash O; Cancer Epigenetics DPU, GlaxoSmithKline, Collegeville, Pennsylvania, USA., Pappalardi M; Cancer Epigenetics DPU, GlaxoSmithKline, Collegeville, Pennsylvania, USA., Ho TF; Department of Biological Reagents and Assay Development, GlaxoSmithKline, Collegeville, Pennsylvania, USA., Nurse K; Department of Biological Reagents and Assay Development, GlaxoSmithKline, Collegeville, Pennsylvania, USA., Oza KP; Department of Biological Reagents and Assay Development, GlaxoSmithKline, Collegeville, Pennsylvania, USA., Gallagher KT; Discovery Core Technologies and Capabilities, GlaxoSmithKline, Collegeville, Pennsylvania, USA., Kruger R; Cancer Epigenetics DPU, GlaxoSmithKline, Collegeville, Pennsylvania, USA., Moyer MP; Raze Therapeutics, Cambridge, Massachusetts, USA., Copeland RA; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Chesworth R; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA., Duncan KW; Departments of Biology and Molecular Discovery, Epizyme, Inc., Cambridge, Massachusetts, USA.
المصدر: Nature chemical biology [Nat Chem Biol] 2015 Jun; Vol. 11 (6), pp. 432-7. Date of Electronic Publication: 2015 Apr 27.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Nature Pub. Group Country of Publication: United States NLM ID: 101231976 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1552-4469 (Electronic) Linking ISSN: 15524450 NLM ISO Abbreviation: Nat Chem Biol Subsets: MEDLINE
مواضيع طبية MeSH: Antineoplastic Agents/*pharmacology , Isoquinolines/*pharmacology , Lymphoma, Mantle-Cell/*pathology , Protein-Arginine N-Methyltransferases/*antagonists & inhibitors , Pyrimidines/*pharmacology, Animals ; Antineoplastic Agents/chemistry ; Antineoplastic Agents/therapeutic use ; Cell Death/drug effects ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Crystallography, X-Ray ; Dose-Response Relationship, Drug ; Humans ; Inhibitory Concentration 50 ; Isoquinolines/chemistry ; Isoquinolines/therapeutic use ; Lymphoma, Mantle-Cell/drug therapy ; Lymphoma, Mantle-Cell/enzymology ; Male ; Methylation ; Mice, Inbred Strains ; Models, Molecular ; Molecular Structure ; Protein Binding ; Pyrimidines/chemistry ; Pyrimidines/therapeutic use ; Xenograft Model Antitumor Assays ; snRNP Core Proteins/metabolism