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المؤلفون: Susan Boroski, David Gray, Lynne Denny, Wenjian Xu, Brian M. Campbell, Nancy C. Stratman, Al Probert, Amy B. Dounay, Lori M. Evans, Nancy Sue Barta
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:6604-6607
مصطلحات موضوعية: Stereochemistry, Dopamine, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Partial agonist, Piperazines, Reuptake, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Norepinephrine reuptake inhibitor, Drug Discovery, medicine, Neurotransmitter Uptake Inhibitors, Neurotransmitter, Molecular Biology, Serotonin Plasma Membrane Transport Proteins, Molecular Structure, Organic Chemistry, Diphenyl ether, Stereoisomerism, Serotonin 5-HT1 Receptor Agonists, Monoamine neurotransmitter, chemistry, Molecular Medicine, Reuptake inhibitor, Ethers, medicine.drug
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2
المؤلفون: Brian Nichelson, Mark G. Vartanian, Charles Taylor, Susan M. Lotarski, Nancy Sue Barta, Sean D. Donevan, Sian E. Gibbons, Norman L. Colbry, Zhu Zhijian, Melvin R. Dickerson, Paul Galatsis, Russell J. DeOrazio, Jacob Bradley Schwarz, Kristin Knapp Lin, Zheng Li, Andrew John Thorpe, Jack J. Kinsora, Raymond Andrew Hudack, David J. Wustrow, David D. Manning, Ayman El-Kattan
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:3559-3563
مصطلحات موضوعية: Cyclohexanecarboxylic Acids, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Carboxylic Acids, Drug Evaluation, Preclinical, Pregabalin, Pharmaceutical Science, Biochemistry, Chemical synthesis, Epilepsy, Reflex, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Animals, Tetrazole, Carboxylate, Amines, Molecular Biology, gamma-Aminobutyric Acid, Binding Sites, Molecular Structure, Organic Chemistry, Stereoisomerism, Biological activity, Disease Models, Animal, Protein Subunits, Anticonvulsant, chemistry, Mice, Inbred DBA, Molecular Medicine, Anticonvulsants, Bioisostere, Gabapentin, medicine.drug
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المؤلفون: Dong Liming, Xinjun Hou, Elizabeth A. Lunney, Corinne E. Augelli-Szafran, Deal Judith G, Christopher F. Bigge, Darin Vanderpool, Raymond Andrew Hudack, Nancy Sue Barta, Bradley William Caprathe, Chuangxing Guo, Steve Bender, Richard E. Showalter, Lorraine Kathleen Fay, Arindam Chatterjee
المصدر: Journal of Medicinal Chemistry. 49:1202-1206
مصطلحات موضوعية: Peptidylprolyl isomerase, Aza Compounds, Binding Sites, Neurite, Chemistry, Hydrogen Bonding, Biological activity, Tacrolimus Binding Protein 1A, Isoquinolines, Ligands, Amides, Heterocyclic Compounds, 4 or More Rings, Tacrolimus, Structure-Activity Relationship, Neuroprotective Agents, FKBP, Biochemistry, Cis-trans-Isomerases, Drug Discovery, Molecular Medicine, Structure–activity relationship, Binding site, Cognitive decline
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4
المؤلفون: Nancy Sue Barta, Steven A. Weissman, Paul J. Reider, Kara B. Somerville, Daniel R. Sidler, Robert D. Larsen
المصدر: Organic Letters. 2:2821-2824
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Yield (chemistry), Organic Chemistry, Hydantoin, Physical and Theoretical Chemistry, Ring (chemistry), Biochemistry, Combinatorial chemistry, Styrene
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المؤلفون: Alan E. Rowan, Jorge M. M. Verkade, Nancy Sue Barta, Sudip Malik, Brian Gibson, Floris L. van Delft, John Cooke Hodges, Anup M. Jawalekar
المصدر: Molecules, 18, 7, pp. 7346-7363
Molecules
Molecules, 18, 7346-7363
Molecules, Vol 18, Iss 7, Pp 7346-7363 (2013)
Volume 18
Issue 7
Pages: 7346-7363مصطلحات موضوعية: Azides, Oligonucleotides, Pharmaceutical Science, chemistry.chemical_element, Synthetic Organic Chemistry, 010402 general chemistry, 01 natural sciences, Catalysis, Article, Analytical Chemistry, copper-free click, lcsh:QD241-441, chemistry.chemical_compound, strain-promoted cycloaddition, lcsh:Organic chemistry, Drug Discovery, azide, Organic chemistry, bicyclononyne, Physical and Theoretical Chemistry, GeneralLiterature_REFERENCE(e.g.,dictionaries,encyclopedias,glossaries), oligonucleotide conjugation, Phosphoramidite, Bicyclic molecule, Molecular Structure, 010405 organic chemistry, Oligonucleotide, Organic Chemistry, Molecular Materials, Stereoisomerism, Combinatorial chemistry, Copper, 0104 chemical sciences, Fluorescent labelling, chemistry, Chemistry (miscellaneous), Biotinylation, Click chemistry, Molecular Medicine, Click Chemistry, Azide
وصف الملف: application/pdf
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المؤلفون: Joanne Brodfuehrer, Cheryl Li, Christopher Lepsy, Amy B. Dounay, Brian M. Campbell, Nancy Sue Barta, David Gray, Liming Zhang, Taraneh Haske
المصدر: The AAPS journal. 14(2)
مصطلحات موضوعية: Male, medicine.medical_specialty, Dopamine, Pharmaceutical Science, Prefrontal Cortex, Pharmacology, Atomoxetine Hydrochloride, Partial agonist, Models, Biological, Buspirone, Rats, Sprague-Dawley, Norepinephrine, Norepinephrine reuptake inhibitor, Internal medicine, medicine, Animals, Humans, Drug Partial Agonism, Prefrontal cortex, Adrenergic Uptake Inhibitors, Dose-Response Relationship, Drug, Propylamines, Chemistry, Atomoxetine, Serotonin 5-HT1 Receptor Agonists, Rats, Endocrinology, Pharmacodynamics, medicine.drug, Research Article
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7
المؤلفون: Elizabeth M. Collantes, Kim Zoski, David Gray, Tammy Whisman, Nancy Sue Barta, Samarendra N. Maiti, Rajendra Subedi, Daniel F. Ortwine, Rathna Iyer, Lynne Denny, Satavisha Dutta, Al Probert, Corey Coleman, Nancy C. Stratman, Amy B. Dounay, Wenjian Xu, Brian M. Campbell, Dongfeng Hou
المصدر: Bioorganicmedicinal chemistry letters. 20(3)
مصطلحات موضوعية: medicine.medical_specialty, Pyridines, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Partial agonist, Cell Line, Norepinephrine (medication), chemistry.chemical_compound, Norepinephrine reuptake inhibitor, Phenols, Internal medicine, Drug Discovery, medicine, Humans, Neurotransmitter, Molecular Biology, Dopamine transporter, Norepinephrine Plasma Membrane Transport Proteins, biology, Adrenergic Uptake Inhibitors, Organic Chemistry, Serotonin 5-HT1 Receptor Agonists, Serotonin Receptor Agonists, Endocrinology, chemistry, Norepinephrine transporter, Drug Design, Receptor, Serotonin, 5-HT1A, Catecholamine, biology.protein, Microsomes, Liver, Molecular Medicine, Reuptake inhibitor, medicine.drug
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المؤلفون: Nancy Sue Barta, Shelly Ann Glase, Wenjian Xu, David Gray
المصدر: ChemInform. 40
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Reboxetine, Morpholine, medicine, General Medicine, Pharmacology, medicine.drug, Norepinephrine reuptake
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9
المؤلفون: Brian M. Campbell, Amy B. Dounay, Pil H. Lee, Nancy Sue Barta, Lori M. Evans, Terry Crawford, Susan A. Borosky, Wenjian Xu, David Gray, Lynne Denny, Jack A. Bikker, Edward A. Lenoir
المصدر: Bioorganicmedicinal chemistry letters. 19(4)
مصطلحات موضوعية: Agonist, Indoles, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Ether, Biochemistry, Partial agonist, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Potency, Structure–activity relationship, Combinatorial Chemistry Techniques, Humans, Molecular Biology, 5-HT receptor, Molecular Structure, Chemistry, Organic Chemistry, Buspirone, Serotonin Receptor Agonists, Pyrimidines, Drug Design, Lipophilicity, Receptor, Serotonin, 5-HT1A, Microsome, Microsomes, Liver, Molecular Medicine
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المؤلفون: Wenjian Xu, Nancy Sue Barta, Shelly Ann Glase, David Gray
المصدر: Bioorganicmedicinal chemistry letters. 18(20)
مصطلحات موضوعية: Stereochemistry, Chemistry, Pharmaceutical, Morpholines, Clinical Biochemistry, Pharmaceutical Science, Stereoisomerism, Biochemistry, Chemical synthesis, Reuptake, chemistry.chemical_compound, Norepinephrine, Reboxetine, Structure-Activity Relationship, Norepinephrine reuptake inhibitor, Morpholine, Drug Discovery, medicine, Structure–activity relationship, Humans, Molecular Biology, Adrenergic Uptake Inhibitors, Chemistry, Organic Chemistry, Ketones, Monoamine neurotransmitter, Models, Chemical, Drug Design, Molecular Medicine, medicine.drug, Central Nervous System Agents, Toluene