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1دورية أكاديمية
المؤلفون: Bharate, Jaideep B, McConnell, Nicholas, Naresh, Gunaganti, Zhang, Lingtian, Lakkaniga, Naga Rajiv, Ding, Lucky, Shah, Neil P, Frett, Brendan, Li, Hong-Yu
المصدر: Scientific reports. 8(1)
مصطلحات موضوعية: Cell Line, Tumor, Humans, Pyrimidines, Antineoplastic Agents, Protein Kinase Inhibitors, Enzyme Activation, Structure-Activity Relationship, Proto-Oncogene Proteins c-kit, fms-Like Tyrosine Kinase 3, Cell Line, Tumor
وصف الملف: application/pdf
URL الوصول: https://escholarship.org/uc/item/2294d0x7
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2
المؤلفون: Baljinder Singh, Amrita Sharma, Naresh Gunaganti, Mitch Rivers, Pradip K. Gadekar, Brady Greene, Michael Chichioco, Carlos E. Sanz-Rodriguez, Courtney Fu, Catherine LeBlanc, Erin Burchfield, Nyle Sharif, Benjamin Hoffman, Gaurav Kumar, Andrei Purmal, Kojo Mensa-Wilmot, Michael P. Pollastri
المصدر: Journal of Medicinal Chemistry. 66:1972-1989
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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3دورية أكاديمية
المؤلفون: Frett, Brendan, McConnell, Nicholas, Kharbanda, Anupreet, Naresh, Gunaganti, Rounseville, Benjamin, Warner, Christina, Chang, John, Debolske, Natalie, Li, Hong-yu
المصدر: In Tetrahedron 30 August 2018 74(35):4592-4600
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4
المؤلفون: Pilar Manzano, Maria Santos Martinez-Martinez, Miguel Navarro, Michael P. Pollastri, Naresh Gunaganti, Gloria Ceballos-Pérez, Kirsten Gillingwater, Domingo I. Rojas-Barros, Rosario Diaz-Gonzalez, Baljinder Singh
المساهمون: Tres Cantos Open Lab Foundation, National Institute of Allergy and Infectious Diseases (US), National Institutes of Health (US)
المصدر: Digital.CSIC. Repositorio Institucional del CSIC
instname
J Med Chemمصطلحات موضوعية: Antiparasitic, medicine.drug_class, Trypanosoma brucei brucei, Trypanosoma brucei, Proof of Concept Study, Medicinal chemistry, Article, Mice, Structure-Activity Relationship, Parasitic Sensitivity Tests, In vivo, parasitic diseases, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, African trypanosomiasis, ADME, Molecular Structure, Chemotype, biology, Chemistry, Hep G2 Cells, biology.organism_classification, medicine.disease, Trypanocidal Agents, In vitro, Rats, Purines, Microsomes, Liver, Molecular Medicine
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5
المؤلفون: Naresh Gunaganti, Yuet-Kin Leung, Lingtian Zhang, Naga Rajiv Lakkaniga, Brendan Frett, Hong-yu Li, Binyam Belachew
المصدر: European journal of medicinal chemistry. 206
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, endocrine system, endocrine system diseases, Pyrimidine, Antineoplastic Agents, Chemistry Techniques, Synthetic, 01 natural sciences, 03 medical and health sciences, chemistry.chemical_compound, Cell Movement, Cell Line, Tumor, Drug Discovery, Structure–activity relationship, Humans, Pyrroles, neoplasms, Protein Kinase Inhibitors, 030304 developmental biology, Cell Proliferation, Pharmacology, 0303 health sciences, 010405 organic chemistry, Kinase, Point mutation, Organic Chemistry, Proto-Oncogene Proteins c-ret, General Medicine, 0104 chemical sciences, Pyrimidines, chemistry, Biochemistry, Cell culture, Drug Design, Bioisostere, Growth inhibition, Lead compound
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6
المؤلفون: Lingtian Zhang, Naresh Gunaganti, Naga Rajiv Lakkaniga, Brendan Frett, Anupreet Kharbanda, Rose Cooper, Hong-yu Li
المصدر: Chemical Communications. 54:12954-12957
مصطلحات موضوعية: Pyridines, Decarboxylation, Antineoplastic Agents, 010402 general chemistry, 01 natural sciences, Article, Catalysis, Small Molecule Libraries, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, Pyridine, Materials Chemistry, Humans, Molecule, Molecular Structure, 010405 organic chemistry, Chemistry, Drug discovery, Imidazoles, Metals and Alloys, General Chemistry, Boronic Acids, Combinatorial chemistry, Chemical space, 0104 chemical sciences, Surfaces, Coatings and Films, Electronic, Optical and Magnetic Materials, Models, Chemical, Ceramics and Composites, Boronic acid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2bb956c535be6ad7842b4b160938bea3
https://doi.org/10.1039/c8cc07063f -
7
المؤلفون: Naga Rajiv Lakkaniga, Wei Yan, Naresh Gunaganti, Francesca Carlomagno, Neil Q. McDonald, Massimo Santoro, Fengping Lv, Hong-yu Li, Brendan Frett
المساهمون: Yan, Wei, Lakkaniga, Naga Rajiv, Carlomagno, Francesca, Santoro, Massimo, Mcdonald, Neil Q., Lv, Fengping, Gunaganti, Naresh, Frett, Brendan, Li, Hong-Yu
المصدر: J Med Chem
Journal of medicinal chemistry (Online) 62 (2019): 1731–1760. doi:10.1021/acs.jmedchem.8b01092
info:cnr-pdr/source/autori:Yan W.; Lakkaniga N.R.; Carlomagno F.; Santoro M.; McDonald N.Q.; Lv F.; Gunaganti N.; Frett B.; Li H.-Y./titolo:Insights into Current Tropomyosin Receptor Kinase (TRK) Inhibitors: Development and Clinical Application/doi:10.1021%2Facs.jmedchem.8b01092/rivista:Journal of medicinal chemistry (Online)/anno:2019/pagina_da:1731/pagina_a:1760/intervallo_pagine:1731–1760/volume:62مصطلحات موضوعية: animal structures, Antineoplastic Agents, 01 natural sciences, Article, Rats, Sprague-Dawley, 03 medical and health sciences, Catalytic Domain, Cell Line, Tumor, Neoplasms, Drug Discovery, medicine, Animals, Humans, Receptor, trkB, Receptor, trkC, Precision Medicine, Receptor, trkA, Receptor, Protein Kinase Inhibitors, 030304 developmental biology, 0303 health sciences, Mice, Inbred BALB C, Chemistry, Drug discovery, Kinase Family, Kinase, Drug Discovery3003 Pharmaceutical Science, Imatinib, Tropomyosin, Receptor Kinase, (TRK) Inhibitors, Precision medicine, 0104 chemical sciences, enzymes and coenzymes (carbohydrates), 010404 medicinal & biomolecular chemistry, nervous system, Trk receptor, embryonic structures, Cancer research, Molecular Medicine, medicine.drug
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8
المؤلفون: Neil Q. McDonald, Naresh Gunaganti, Massimo Santoro, Wei Yan, Naga Rajiv Lakkaniga, Brendan Frett, Hong-yu Li, Francesca Carlomagno, Fengping Lv
المصدر: Journal of Medicinal Chemistry. 63:10089-10089
مصطلحات موضوعية: Chemistry, Kinase, Trk receptor, Drug Discovery, Cancer research, Molecular Medicine, Receptor, Tropomyosin
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9
المؤلفون: Brendan Frett, David Jayabalan, Eloisi Caldas Lopes, Jorge Contreras, Morton Coleman, Jorge Monge, Monica L. Guzman, Naresh Gunaganti, Hong-yu Li, Ruben Niesvizky
المصدر: Cancer Research. 80:5155-5155
مصطلحات موضوعية: Cancer Research, business.industry, Bortezomib, Cell, Cancer, medicine.disease, Carfilzomib, chemistry.chemical_compound, medicine.anatomical_structure, Histone phosphorylation, Oncology, chemistry, Toxicity, medicine, Cancer research, business, Multiple myeloma, Lenalidomide, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::e7172fea2c76f464b6305f336744262c
https://doi.org/10.1158/1538-7445.am2020-5155 -
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المؤلفون: Naresh Gunaganti, Tadigopula Narender, Sandeep Kumar Singh, Naveen Parmar, Muhammad Wahajuddin, Ashok Kumar, Mamunur Rashid, Susanta Kar, Kalyan Mitra, Pragya Chandrakar
المصدر: European Journal of Medicinal Chemistry. 182:111632
مصطلحات موضوعية: Cell Survival, Antiprotozoal Agents, Pharmacology, Electron Transport Complex III, Mice, Structure-Activity Relationship, Parasitic Sensitivity Tests, Cricetinae, Chlorocebus aethiops, Drug Discovery, Extracellular, medicine, Animals, Amino Acids, Amastigote, Vero Cells, IC50, chemistry.chemical_classification, Mice, Inbred BALB C, Dose-Response Relationship, Drug, Molecular Structure, ATP synthase, biology, Chemistry, Organic Chemistry, General Medicine, medicine.disease, Mitochondria, Amino acid, Visceral leishmaniasis, biology.protein, Vero cell, Leishmaniasis, Visceral, Intracellular, Leishmania donovani