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1
المؤلفون: Jeremy S. Parker, Nash Ian Alun, Katherine M. P. Wheelhouse, Peter J. Lindsay-Scott, Paul Alan Glossop, Timothy J. Donohoe
مصطلحات موضوعية: Oxidative cyclization, Molecular Structure, Pyridines, chemistry.chemical_element, Pyridine-N-oxide, Stereoisomerism, Homogeneous catalysis, General Chemistry, General Medicine, Osmium, Amino Alcohols, Catalysis, Pyrrolidine, chemistry.chemical_compound, chemistry, Cyclization, Organic chemistry, Carbamates, Oxidation-Reduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6f1b0cff515eb3658cccc300c9e5da01
https://doi.org/10.1002/anie.200705425 -
2
المؤلفون: Paul A. Bethel, Kurt Gordon Pike, Alan C. Reid, Wendy L. Snelson, John G. Cumming, Stefan Gerhardt, Richard A. Pauptit, Dearg S. Brown, Thompson Caroline Rachel, Nash Ian Alun, Jonathan E. Finlayson, Steve Swallow
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:3879-3883
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Plasma protein binding, Crystallography, X-Ray, Biochemistry, Piperazines, Mitogen-Activated Protein Kinase 14, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Aniline, Drug Discovery, Animals, Humans, Structure–activity relationship, Transferase, Benzamide, Protein Kinase Inhibitors, Molecular Biology, Quinazolinone, Inflammation, biology, Chemistry, Drug discovery, Anti-Inflammatory Agents, Non-Steroidal, Organic Chemistry, Blood Proteins, Rats, Molecular Weight, Solubility, Mitogen-activated protein kinase, biology.protein, Molecular Medicine, Protein Binding
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3
المؤلفون: Andrew David Morley, Galith Karoutchi, Stefan Gerhardt, Attilla Ting, Chris De Savi, Nash Ian Alun, Ken Page
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:271-277
مصطلحات موضوعية: Models, Molecular, Zinc binding, Matrix metalloproteinase inhibitor, Chemistry, Pharmaceutical, Clinical Biochemistry, Pharmaceutical Science, Matrix Metalloproteinase Inhibitors, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, Dogs, Matrix Metalloproteinase 13, Osteoarthritis, Drug Discovery, Animals, Humans, Structure–activity relationship, Potency, Enzyme Inhibitors, Lead (electronics), Molecular Biology, Chemistry, Organic Chemistry, Dosing regimen, Combinatorial chemistry, Rats, Bioavailability, Zinc, Models, Chemical, Solubility, Drug Design, Molecular Medicine, Selectivity
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المؤلفون: Michael James, Gordon A. Hamlin, Stefan Gerhardt, David Ryan, Nash Ian Alun, Attilla Ting, Stephen J. Norris, Galith Karoutchi, Chris De Savi, Neil Rankine, David J. Hargreaves, Christine M. Wood, Sarah V. Baker, Philip A. MacFaul, Andrew David Morley, Kostas Karabelas
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:4215-4219
مصطلحات موضوعية: Molecular model, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Stereoisomerism, Carboxamide, Matrix Metalloproteinase Inhibitors, Crystallography, X-Ray, Biochemistry, Structure-Activity Relationship, Catalytic Domain, Matrix Metalloproteinase 13, Drug Discovery, Hydrolase, medicine, Structure–activity relationship, Protease Inhibitors, Binding site, Molecular Biology, Binding Sites, biology, Chemistry, Organic Chemistry, Zinc, Enzyme inhibitor, biology.protein, Molecular Medicine, Selectivity
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المؤلفون: Janet D. Culshaw, Jason Breed, M. Raymond V. Finlay, Julie A. Tucker, J.J. Stanway, Claire Brassington, Kate Byth, Andy Barker, Malcolm Anderson, Nash Ian Alun, Richard A. Pauptit, Andrew D. Roberts, Andrew Peter Thomas, Hazel M. Weir, Michael A. Walker, David M. Andrews, Nicholas John Newcombe, Eric Fisher, Dave W. Heaton, Helen H.J. McMiken, Clive Green, Sandra E. Oakes
المصدر: Bioorganicmedicinal chemistry letters. 18(20)
مصطلحات موضوعية: Chemistry, Pharmaceutical, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Cell Cycle Proteins, Crystallography, X-Ray, Biochemistry, Sulfone, chemistry.chemical_compound, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, Cyclin-dependent kinase, Drug Discovery, Transferase, Imidazole, Animals, Humans, Molecular Biology, chemistry.chemical_classification, Aniline Compounds, biology, Kinase, Organic Chemistry, Imidazoles, Hydrogen Bonding, Cyclin-Dependent Kinases, Enzyme, chemistry, Models, Chemical, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, CDK inhibitor