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المؤلفون: Saijian, Shi, Jian, Xu, LingLing, Feng, Xin, Fan, Zhen, Chen, Yajuan, Qin, Nga N, Chung, Tingyou, Li, Peter W, Schiller
المصدر: Chemical biologydrug designREFERENCES. 96(5)
مصطلحات موضوعية: Narcotic Antagonists, Receptors, Opioid, mu, Animals, Oligopeptides
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المؤلفون: Ding Yi, Zhen Chen, Tingyou Li, Peter W. Schiller, Cai Yunxin, Dandan Lu, Nga N. Chung
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:3629-3631
مصطلحات موضوعية: 0301 basic medicine, Antioxidant, Stereochemistry, DPPH, medicine.medical_treatment, Clinical Biochemistry, Receptors, Opioid, mu, Pharmaceutical Science, Peptide, Biochemistry, Article, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Opioid Receptor Binding, Drug Discovery, medicine, Humans, Tyrosine, Molecular Biology, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, 3. Good health, DAMGO, PyBOP, 030104 developmental biology, chemistry, Opioid, Molecular Medicine, Oligopeptides, medicine.drug
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المؤلفون: Wim Bert Griet Schepens, Peter W. Schiller, Steven Ballet, Emilie Eiselt, Nga N. Chung, Tom Willemse, Louis Gendron, Jean-Michel Longpré, Philippe Sarret, Karlijn Hollanders, Véronique Blais, Bert U. W. Maes, Herman van Vlijmen, Brain Holleran
المصدر: Bioorganic and medicinal chemistry letters
مصطلحات موضوعية: Male, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Guinea Pigs, Receptors, Opioid, mu, Pharmaceutical Science, Phenylalanine, 010402 general chemistry, Ligands, 01 natural sciences, Biochemistry, Article, Rats, Sprague-Dawley, Mice, Opioid receptor, Receptors, Opioid, delta, Drug Discovery, Side chain, Structural isomer, medicine, Moiety, Animals, Humans, Opioid peptide, Biology, Molecular Biology, Oligopeptide, Molecular Structure, 010405 organic chemistry, Chemistry, Pharmacology. Therapy, Organic Chemistry, Affinities, 0104 chemical sciences, Analgesics, Opioid, HEK293 Cells, Molecular Medicine, Oligopeptides
وصف الملف: pdf
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المؤلفون: Louis Gendron, Dirk Tourwé, Frédéric Bihel, Nga N. Chung, Peter W. Schiller, Olivier Van der Poorten, Cecilia Betti, Robin Van Den Hauwe, Karel Guillemyn, Emilie Eiselt, Steven Ballet, François Hallé, Philippe Sarret
المساهمون: Laboratoire d'Innovation Thérapeutique (LIT), Université de Strasbourg (UNISTRA)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS), Department of Organic Chemistry, Vrije Universiteit Brussel (VUB), Department of Physiology and Biophysics, Université de Sherbrooke (UdeS), Montreal Neurological Institute and Hospital, McGill University = Université McGill [Montréal, Canada], Centre National de la Recherche Scientifique (CNRS)-Université de Strasbourg (UNISTRA)-Institut de Chimie du CNRS (INC)
المصدر: ACS Medicinal Chemistry Letters
ACS Medicinal Chemistry Letters, American Chemical Society, 2017, 8 (11), pp.1177-1182. ⟨10.1021/acsmedchemlett.7b00347⟩مصطلحات موضوعية: 0301 basic medicine, chemistry.chemical_classification, Tetrapeptide, 010405 organic chemistry, Stereochemistry, Organic Chemistry, Peptide, Dermorphin, [CHIM.THER]Chemical Sciences/Medicinal Chemistry, 01 natural sciences, Biochemistry, Combinatorial chemistry, ANT, 0104 chemical sciences, Amino acid, 03 medical and health sciences, chemistry.chemical_compound, Residue (chemistry), 030104 developmental biology, chemistry, Drug Discovery, Receptor, Selectivity, ComputingMilieux_MISCELLANEOUS
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المؤلفون: Nga N. Chung, Peter W. Schiller, Jason J. Guo, Grazyna Weltrowska, Brian C. Wilkes, Carole Lemieux
المصدر: Bioorganic & Medicinal Chemistry. 22:4581-4586
مصطلحات موضوعية: Intrinsic activity, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Receptors, Opioid, mu, Pharmaceutical Science, Biochemistry, Partial agonist, Article, Carfentanil, Structure-Activity Relationship, Opioid receptor, Opioid Receptor Binding, mental disorders, Drug Discovery, medicine, Molecular Biology, Binding selectivity, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Stereoisomerism, 3. Good health, Fentanyl, Molecular Docking Simulation, nervous system, Opioid, Docking (molecular), Molecular Medicine, medicine.drug
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المؤلفون: Joanna Mika, Joost Van Duppen, Katarzyna Popiolek-Barczyk, Attila Keresztes, John M. Streicher, Peter W. Schiller, Karel Guillemyn, Steven Ballet, Adriano Mollica, Jozef Vanden Broeck, Joanna Starnowska, Carole Lemieux, Barbara Przewlocka, Roberto Costante, Dirk Tourwé, Nga N. Chung
مصطلحات موضوعية: 0301 basic medicine, NK1 antagonists, Physiology, medicine.drug_class, Cognitive Neuroscience, Analgesic, Receptors, Opioid, mu, Hybrid peptides, Substance P, Pharmacology, opioid agonism, Ligands, Biochemistry, Article, 03 medical and health sciences, chemistry.chemical_compound, Mice, 0302 clinical medicine, Receptors, Opioid, delta, medicine, Animals, Receptor, Spinal Cord Injuries, neuropathic pain, Analgesics, Chemistry, acute pain, Cell Biology, General Medicine, Receptors, Neurokinin-1, Receptor antagonist, Constriction, Analgesics, Opioid, 030104 developmental biology, Opioid, Spinal Cord, Neuropathic pain, Chronic Disease, Neuralgia, NK1 receptor antagonist, μ-opioid receptor, 030217 neurology & neurosurgery, medicine.drug
وصف الملف: Print-Electronic
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bbdd56be47ca77328f58848e3431857d
https://lirias.kuleuven.be/handle/123456789/632022 -
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المؤلفون: Patrycja Kleczkowska, Dirk Tourwé, Csaba Tömböly, Lipkowski Andrzej W, Steven Ballet, Carsten Uhd Nielsen, Anna Lesniak, Birger Brodin, Cecilia Betti, Nga N. Chung, Hans Christian Cederberg Helms, Peter W. Schiller, Alexandre Novoa
المصدر: ACS Medicinal Chemistry Letters. 5:352-357
مصطلحات موضوعية: chemistry.chemical_classification, Agonist, Glycosylation, medicine.drug_class, Organic Chemistry, Peptide, Pharmacology, Biochemistry, In vitro, chemistry.chemical_compound, chemistry, In vivo, Opioid receptor, Paracellular transport, Drug Discovery, medicine, Opioid peptide
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المؤلفون: Bert U. W. Maes, Emilie Eiselt, Tom Willemse, Jean-Michel Longpré, Wim Bert Griet Schepens, Philippe Sarret, Brian J. Holleran, Véronique Blais, Peter W. Schiller, Nga N. Chung, Karlijn Hollanders, Steven Ballet, Louis Gendron, Herman van Vlijmen
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:3418
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Agonism, Opioid peptide, Molecular Biology, Biochemistry, Chemical space
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المؤلفون: Ewa Gibula-Bruzda, Jan Izdebski, Jolanta Kotlinska, Ewa Witkowska, Nga N. Chung, Peter W. Schiller
المصدر: Peptides. 39:103-110
مصطلحات موضوعية: Male, Nociception, Agonist, Physiology, medicine.drug_class, Narcotic Antagonists, Analgesic, Pharmacology, Biochemistry, Article, Cellular and Molecular Neuroscience, chemistry.chemical_compound, Endocrinology, Drug tolerance, Naltrindole, Receptors, Opioid, delta, medicine, Animals, Rats, Wistar, Pain Measurement, Morphine, Receptors, Opioid, kappa, Antagonist, Drug Synergism, Drug Tolerance, Naltrexone, Rats, Analgesics, Opioid, Opioid, chemistry, Deltorphin, Oligopeptides, medicine.drug
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المؤلفون: Sofie Stalmans, Steven Ballet, Carole Lemieux, Dirk Tourwé, Nathalie Bracke, Mariana Spetea, Mark E. Cooper, Peter W. Schiller, Bart De Spiegeleer, Evelien Wynendaele, Sylvia Van Dorpe, Johannes Zuegg, Cecilia Betti, Alexandre Novoa, Nga N. Chung
المصدر: Journal of Medicinal Chemistry. 55:9549-9561
مصطلحات موضوعية: Nociception, Agonist, Biodistribution, Stereochemistry, medicine.drug_class, Peptide, Article, Mice, Structure-Activity Relationship, Drug Discovery, Side chain, medicine, Animals, Structure–activity relationship, Peptide bond, Tissue Distribution, Pain Measurement, chemistry.chemical_classification, Molecular Structure, Chemistry, digestive, oral, and skin physiology, Brain, Analgesics, Opioid, Opioid Peptides, Blood-Brain Barrier, Receptors, Opioid, Lipophilicity, Molecular Medicine, μ-opioid receptor, Oligopeptides