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1
المؤلفون: Yang Wen, Yang He, Nader Fotouhi, Sherif Daouti, Packman Kathryn E, Norman Kong, Wen-hui Li, Kenneth Kolinsky, David C. Heimbrook, Anthony Specian, Frank John Podlaski, Qing Xiang, Nicholas John Silvester Huby, Huisheng Wang, Brian Higgins, Huifeng Niu
المصدر: Cancer Research. 69:1924-1932
مصطلحات موضوعية: MAPK/ERK pathway, Cancer Research, MAP Kinase Signaling System, Angiogenesis, MAP Kinase Kinase 2, MAP Kinase Kinase 1, Antineoplastic Agents, Biology, Mitogen-activated protein kinase kinase, Cell Line, Mice, medicine, Animals, Humans, Phosphorylation, Extracellular Signal-Regulated MAP Kinases, Protein kinase A, Protein Kinase Inhibitors, Imidazoles, Macaca fascicularis, Thiazoles, Oncology, Mechanism of action, Biochemistry, Cancer cell, Cancer research, Female, medicine.symptom, Signal transduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::88d97f0577a8efa56ee33c335664b715
https://doi.org/10.1158/0008-5472.can-08-2627 -
2
المؤلفون: Louis M. Renzetti, Li Chen, Karen Rowan, Allen Sheffron, Tai-Nan Huang, Jian Ping Lou, Jefferson Wright Tilley, Kenneth G. Hull, Virginia Schwinge, Gerry Kaplan, Achyutharao Sidduri, Robert M. Campbell, Robert William Guthrie, Nicholas John Silvester Huby
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:2475-2478
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Phenylalanine, Clinical Biochemistry, Vascular Cell Adhesion Molecule-1, Pharmaceutical Science, Carboxamide, Integrin alpha4beta1, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Molecule, Molecular Biology, Alkyl, chemistry.chemical_classification, Molecular Structure, Organic Chemistry, Antagonist, Cycloparaffins, In vitro, Cycloalkane, chemistry, Molecular Medicine, Lead compound, Protein Binding
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3
المؤلفون: Gary L. Olson, Damir Vidovic, Ramakanth Sarabu, J. Hammer, Francesco Sinigaglia, Zoltan A. Nagy, Michael Steinmetz, Nicholas John Silvester Huby, Jeanmarie Guenot, Charles Belunis, Kouichi Ito, Robert K. Campbell, Paul Gillespie, David Robert Bolin, Steven Joseph Berthel, Vincent S. Madison, Fiorenza Falcioni
المصدر: Nature Biotechnology. 17:562-567
مصطلحات موضوعية: Peptidomimetic, T-Lymphocytes, Antigen presentation, Biomedical Engineering, Arthritis, Bioengineering, Plasma protein binding, Biology, medicine.disease_cause, Applied Microbiology and Biotechnology, Cell Line, Arthritis, Rheumatoid, medicine, Humans, Amino Acid Sequence, Peptide sequence, Autoimmune disease, Antigen Presentation, Molecular Mimicry, Hydrogen Bonding, HLA-DR Antigens, medicine.disease, Cathepsins, Molecular mimicry, Amino Acid Substitution, Cell culture, Immunology, Molecular Medicine, Oligopeptides, Protein Binding, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::70409305cc5fff290c510e7758273981
https://doi.org/10.1038/9865 -
4
المؤلفون: Huifeng Niu, Brian Higgins, Kenneth Kolinsky, Huisheng Wang, Jia Kui Li, Sherif Daouti, Harpreet K. Sandhu, Petra Goelzer, David C. Heimbrook, Mei Liu, Packman Kathryn E, Aruna Railkar, Nader Fotouhi, John Anthony Moliterni, Nicholas John Silvester Huby, Christine Rizzo
المصدر: Molecular cancer therapeutics. 9(1)
مصطلحات موضوعية: MAPK/ERK pathway, Cancer Research, MAP Kinase Kinase 2, MAP Kinase Kinase 1, Mice, Nude, Pharmacology, Biology, Imidazolidines, Mice, Pharmacokinetics, In vivo, Cell Line, Tumor, medicine, Animals, Humans, Protein kinase A, Protein Kinase Inhibitors, Kinase, Melanoma, medicine.disease, Phenylbutyrates, Xenograft Model Antitumor Assays, Macaca fascicularis, Oncology, Mechanism of action, Pharmacodynamics, medicine.symptom, Drug Screening Assays, Antitumor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1a10022a43f230d2596f5b4e8f29b8ef
https://pubmed.ncbi.nlm.nih.gov/20053779 -
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المؤلفون: Sherrie L. Pietranico, Ping Wang, Nicholas John Silvester Huby, Mary-Lou Gubler, Louise H. Foley, Weiya Yun, John Vermeulen, Stanley Wertheimer, Gwendolyn Ramsey, Pete William Dunten, Katherine Toth
المصدر: Bioorganicmedicinal chemistry letters. 17(14)
مصطلحات موضوعية: chemistry.chemical_classification, Models, Molecular, Bicyclic molecule, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Lyase, Biochemistry, Chemical synthesis, Sulfonamide, chemistry.chemical_compound, Cytosol, chemistry, Amide, Xanthines, Drug Discovery, Molecular Medicine, Humans, Phosphoenolpyruvate Carboxykinase (GTP), Enzyme Inhibitors, Phosphoenolpyruvate carboxykinase, Molecular Biology, Derivative (chemistry), Alkyl
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المؤلفون: Ramakanth Sarabu, Fiorenza Falcioni, Amy Swain, Lucja Orzechowski, Raymond Makofske, Ursula Kammlott, Xiaolei Zhang, Jeanmarie Guenot, Donald C. Cox, Damir Vidovic, Gary L. Olson, Nan Jiang, David Robert Bolin, Robert Crowther, Joel P. Cooper, Paul Gillespie, Diana Gaizband, Robert M. Campbell, Charles Belunis, David J. Weber, Kouichi Ito, Steven Joseph Berthel, Agostino Perrotta, Robert Palermo, Nicholas John Silvester Huby, Zoltan A. Nagy, Katherine Toth
المصدر: Journal of medicinal chemistry. 43(11)
مصطلحات موضوعية: Models, Molecular, Peptide Biosynthesis, Phage display, Stereochemistry, Protein Conformation, T-Lymphocytes, Antigen presentation, Carbohydrates, Peptide, Major histocompatibility complex, Crystallography, X-Ray, Binding, Competitive, Methylation, Cathepsin B, chemistry.chemical_compound, Structure-Activity Relationship, Antigen, Drug Discovery, HLA-DR, Humans, chemistry.chemical_classification, MHC class II, Antigen Presentation, Dipeptide, biology, Molecular Mimicry, Dipeptides, HLA-DR Antigens, chemistry, Biochemistry, biology.protein, Molecular Medicine, Cell Division
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المؤلفون: Sherif Daouti, Higgins Brian, Christine Rizzo, Huisheng Wang, Packman Kathryn E, Nicholas John Silvester Huby, Huifeng Niu, Kenneth Kolinsky
المصدر: Molecular Cancer Therapeutics. 8:A247-A247
مصطلحات موضوعية: MAPK/ERK pathway, Cancer Research, Chemistry, Melanoma, MEK inhibitor, Cancer, Gene mutation, Pharmacology, medicine.disease, In vitro, Gemcitabine, Oncology, Cell culture, medicine, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::10396dd8cb444c69daf82b4204ca5103
https://doi.org/10.1158/1535-7163.targ-09-a247