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المؤلفون: Helene Sahri, Julie Christie, Neil John Press, Mark Keenan, Sandra Haberthuer, Morris Tweed, Andrew R. Tuffnell, Mark Mercer, Joseph D. Fullerton, John R. Fozard, Thomas H. Keller, Nicola Elaine Press, Lyndon Nigel Brown, Roger J. Taylor, Clive Mccarthy, Julia Hatto, Robert Cheung, Pamela Tranter
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:3081-3085
مصطلحات موضوعية: medicine.drug_class, Clinical Biochemistry, Adenosine A3 Receptor Antagonists, Pharmaceutical Science, Pharmacology, Receptor, Adenosine A2B, Adenosine receptor antagonist, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Aminothiazole, Heterocyclic Compounds, Drug Discovery, medicine, Animals, Rats, Wistar, Receptor, Molecular Biology, ADME, Chemistry, Receptor, Adenosine A3, Organic Chemistry, Antagonist, Receptor antagonist, Adenosine, Adenosine receptor, Adenosine A2 Receptor Antagonists, Rats, Thiazoles, Molecular Medicine, medicine.drug
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المؤلفون: Nicola Elaine Press, Clive Mccarthy, Ian N. Bruce, Lewis Whitehead, Lilya Sviridenko, Mrinalini Sachin Oza, Gaynor Elizabeth Pilgrim, Darren Le Grand, Charles Owen, Louise Kirman, Graham Charles Bloomfield, Thomas H. Keller, Peter Finan, Judy Hayler, Mohammed Akhlaq, Denise Head, Emma Budd, Julia Hatto, Bernard Cuenoud, Peter Gedeck, Desmond O'Connor, Brian Cox, Catherine Leblanc
المصدر: Bioorganicmedicinal chemistry letters. 22(17)
مصطلحات موضوعية: Gene isoform, Models, Molecular, Cellular activity, Clinical Biochemistry, Pharmaceutical Science, Alpha (ethology), Bioinformatics, Biochemistry, Mice, Phosphatidylinositol 3-Kinases, Catalytic Domain, Drug Discovery, Animals, Humans, Protein Isoforms, PI3-Kinase Inhibitors, Molecular Biology, Protein Kinase Inhibitors, PI3K/AKT/mTOR pathway, Phosphoinositide-3 Kinase Inhibitors, Kinase, Chemistry, Organic Chemistry, SUPERFAMILY, Rats, Thiazoles, Molecular Medicine, Female, Signal Transduction