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1دورية أكاديمية
المؤلفون: Jay M West, Nikolai Zvonok, Kyle M Whitten, Subramanian K Vadivel, Anna L Bowman, Alexandros Makriyannis
المصدر: PLoS ONE, Vol 7, Iss 8, p e43877 (2012)
وصف الملف: electronic resource
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المصدر: Biochemical and Biophysical Research Communications. 591:31-36
مصطلحات موضوعية: Hydrolysis, Biophysics, Arachidonic Acids, Cell Biology, Buffers, Ligands, Biochemistry, Monoacylglycerol Lipases, Amidohydrolases, Glycerides, Substrate Specificity, Kinetics, HEK293 Cells, Isomerism, Receptor, Cannabinoid, CB1, Cyclic AMP, Humans, Molecular Biology, Chromatography, High Pressure Liquid, Endocannabinoids
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3دورية أكاديمية
المؤلفون: Arman A. Sadybekov, Anastasiia V. Sadybekov, Yongfeng Liu, Christos Iliopoulos-Tsoutsouvas, Xi-Ping Huang, Julie Pickett, Blake Houser, Nilkanth Patel, Ngan K. Tran, Fei Tong, Nikolai Zvonok
المصدر: Nature, Nature. 601(7893):452-459
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المؤلفون: Yiran Wu, Keith A. Sharkey, Zhi-Jie Liu, Tian Hua, Alexandros Makriyannis, Catherine M. Keenan, Nikolai Zvonok, Ganesh A. Thakur, Christina A Brust, Travis W. Grim, Simiao Wu, Spyros P. Nikas, Shan Jiang, Fei Tong, Jimit Girish Raghav, Christos Iliopoulos-Tsoutsouvas, Laura M. Bohn, Jo-Hao Ho
المصدر: Journal of Medicinal Chemistry. 64:3870-3884
مصطلحات موضوعية: Male, Cannabinoid receptor, Stereochemistry, CHO Cells, Ligands, 01 natural sciences, Receptor, Cannabinoid, CB2, Mice, 03 medical and health sciences, Cricetulus, Receptor, Cannabinoid, CB1, In vivo, Drug Discovery, Animals, Humans, 030304 developmental biology, Binding affinities, Cannabinoid Receptor Agonists, Analgesics, 0303 health sciences, Cannabinoids, Chemistry, Extramural, Ligand (biochemistry), In vitro, Rats, 3. Good health, 0104 chemical sciences, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Electrophile, Molecular Medicine, Locomotion, Body Temperature Regulation
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المؤلفون: Arman A. Sadybekov, Anastasiia V. Sadybekov, Yongfeng Liu, Christos Iliopoulos-Tsoutsouvas, Xi-Ping Huang, Julie Pickett, Blake Houser, Nilkanth Patel, Ngan K. Tran, Fei Tong, Nikolai Zvonok, Manish K. Jain, Olena Savych, Dmytro S. Radchenko, Spyros P. Nikas, Nicos A. Petasis, Yurii S. Moroz, Bryan L. Roth, Alexandros Makriyannis, Vsevolod Katritch
المصدر: Nature
مصطلحات موضوعية: Multidisciplinary, Article
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b6cb628454a81cf54d8ee8f1bed3cf87
https://europepmc.org/articles/PMC9763054/ -
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المؤلفون: Ioannis P. Papanastasiou, Markos-Orestis Georgiadis, Christos Iliopoulos-Tsoutsouvas, Carol A. Paronis, Christina A. Brust, Ngan K. Tran, Lipin Ji, Xiaoyu Ma, JodiAnne T. Wood, Nikolai Zvonok, Fei Tong, Laura M. Bohn, Spyros P. Nikas, Alexandros Makriyannis
المصدر: European journal of medicinal chemistry. 230
مصطلحات موضوعية: Pharmacology, Structure-Activity Relationship, Receptor, Cannabinoid, CB1, Organic Chemistry, Drug Discovery, General Medicine, Dronabinol
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7
المؤلفون: Arman A, Sadybekov, Anastasiia V, Sadybekov, Yongfeng, Liu, Christos, Iliopoulos-Tsoutsouvas, Xi-Ping, Huang, Julie, Pickett, Blake, Houser, Nilkanth, Patel, Ngan K, Tran, Fei, Tong, Nikolai, Zvonok, Manish K, Jain, Olena, Savych, Dmytro S, Radchenko, Spyros P, Nikas, Nicos A, Petasis, Yurii S, Moroz, Bryan L, Roth, Alexandros, Makriyannis, Vsevolod, Katritch
المصدر: Nature. 601(7893)
مصطلحات موضوعية: Molecular Docking Simulation, rho-Associated Kinases, Drug Discovery, Libraries, Digital, Combinatorial Chemistry Techniques, Ligands, Algorithms
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8
المؤلفون: Nikolai Zvonok, Ken Mackie, Han Zhou, Spyros P. Nikas, Demetris P. Papahatjis, Andrea G. Hohmann, JodiAnne T. Wood, Shu Xu, Simiao Wu, Lipin Ji, Patricia H. Reggio, Marsha R. Eno, Lawrence J. Marnett, Khadijah A. Mohammad, Paula Morales, Yingpeng Liu, Ai-Ling Li, Dow P. Hurst, Shalley N. Kudalkar, Alexandros Makriyannis, Chandrashekhar Honrao, Othman Benchama, Marion Schimpgen
المصدر: Journal of Medicinal Chemistry. 61:8639-8657
مصطلحات موضوعية: Male, Nociception, 0301 basic medicine, Agonist, Cannabinoid receptor, medicine.drug_class, Stereochemistry, Freund's Adjuvant, Anti-Inflammatory Agents, Amidohydrolases, Mice, 03 medical and health sciences, chemistry.chemical_compound, Receptor, Cannabinoid, CB1, In vivo, Enzyme Stability, Drug Discovery, medicine, Animals, Humans, Ethanolamide, Lectins, C-Type, Inflammation, Mice, Knockout, chemistry.chemical_classification, Analgesics, Ligand (biochemistry), Endocannabinoid system, Monoacylglycerol Lipases, In vitro, Rats, HEK293 Cells, 030104 developmental biology, Enzyme, chemistry, Cyclooxygenase 2, Hyperalgesia, Molecular Medicine, lipids (amino acids, peptides, and proteins)
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المؤلفون: Alex Straiker, Shrouq I. Farah, Khadijah A. Mohammad, Alexandros Makriyannis, Catherine M. Weerts, Michael Speziale, Samantha Hilston, Nikolai Zvonok, Manjunath Lamani, Michael S. Malamas, Honrao Chandrashekhar, Christina Yume Miyabe, Maya Ploss
المصدر: Bioorganic & Medicinal Chemistry. :116244
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, DUAL (cognitive architecture), ABHD6, 01 natural sciences, Biochemistry, Combinatorial chemistry, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Drug Discovery, Molecular Medicine, Molecular Biology
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المؤلفون: Han Zhou, Ngan K. Tran, Nikolai Zvonok, Spyros P. Nikas, Alexandros Makriyannis, Marcus A. Tius, Fei Tong, Thanh C. Ho
المصدر: Bioorganic & Medicinal Chemistry Letters. 38:127882
مصطلحات موضوعية: Cannabinoid receptor, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, 01 natural sciences, Biochemistry, Cyclase, Receptor, Cannabinoid, CB2, Structure-Activity Relationship, chemistry.chemical_compound, Receptor, Cannabinoid, CB1, Drug Discovery, medicine, Cannabinoid receptor type 2, Humans, Molecular Biology, chemistry.chemical_classification, Nucleophilic addition, Dose-Response Relationship, Drug, Molecular Structure, Cannabinoids, 010405 organic chemistry, Organic Chemistry, Combinatorial chemistry, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry, Isothiocyanate, Molecular Medicine, lipids (amino acids, peptides, and proteins), Stereoselectivity, Cannabinoid, Tricyclic