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المؤلفون: Suttipol Radomkit, Daniel R. Fandrick, Stefan Braith, Chris H. Senanayake, Arindom Chatterjee, Keith R. Fandrick, Carl A. Busacca, Nitinchandra D. Patel
المصدر: The Journal of Organic Chemistry. 86:4877-4882
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, chemistry, Base (chemistry), 010405 organic chemistry, Organic Chemistry, Organic chemistry, Phenols, 010402 general chemistry, 01 natural sciences, 0104 chemical sciences, Catalysis
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المؤلفون: Heewon Lee, Nelu Grinberg, Nitinchandra D. Patel, Andrew Ye, Azad Hossain, Carl A. Busacca, Jon C. Lorenz, Chris H. Senanayake, Anjan Saha, Denis Byrne, Nizar Haddad, Suresh R. Kapadia, Xudong Wei, Nathan K. Yee, Philomen DeCroos, Bikshandarkoil A. Narayanan, Max Sarvestani, Scott Pennino
المصدر: The Journal of Organic Chemistry. 85:8339-8351
مصطلحات موضوعية: Protease, 010405 organic chemistry, Chemistry, medicine.medical_treatment, Organic Chemistry, Convergent synthesis, Substrate (chemistry), Ether, 010402 general chemistry, 01 natural sciences, Combinatorial chemistry, Protease inhibitor (biology), 0104 chemical sciences, Sulfone, chemistry.chemical_compound, Nucleophilic aromatic substitution, Yield (chemistry), medicine, medicine.drug
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المؤلفون: Zhulin Tan, Nitinchandra D. Patel, Harald Engelhardt, Mark Petronczki, Georg Egger, Elisabeth Grondal, Lyne Lamarre, Joyce C. Leung, Bernadette Sharps, Nizar Haddad, Anke Baum, Andreas Bergner, Andreas Schrenk, Renate Schnitzer, Eugene Chong, Tobias Wunberg, Moriz Mayer, Thomas Gerstberger, Dietrich Böse, Andreas Zoephel, Darryl B. McConnell, Christian Engelhardt, Monika Kriz, Nina C. Gonnella, Mariusz Krawiec, Heinz Stadtmüller, Peter Ettmayer, Jonathan T. Reeves, Julian E. Fuchs, Barbara Hopfgartner, Dirk Scharn, Andreas Grimm, Biljana Peric Simov, Flavio Solca, Gerd Bader, Sandra Döbel, Roland Kousek
المصدر: Journal of Medicinal Chemistry. 62:10272-10293
مصطلحات موضوعية: Lung Neoplasms, Protein Conformation, Entropy, Transgene, Antineoplastic Agents, Mice, Transgenic, Crystallography, X-Ray, medicine.disease_cause, 01 natural sciences, Mice, Structure-Activity Relationship, 03 medical and health sciences, T790M, Carcinoma, Non-Small-Cell Lung, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Epidermal growth factor receptor, Protein Kinase Inhibitors, 030304 developmental biology, 0303 health sciences, Mutation, biology, Chemistry, Xenograft Model Antitumor Assays, respiratory tract diseases, 0104 chemical sciences, ErbB Receptors, 010404 medicinal & biomolecular chemistry, Protein kinase domain, Cyclization, Cell culture, Hepatocytes, Cancer research, biology.protein, Molecular Medicine, Benzimidazoles, Female, Tyrosine kinase
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المؤلفون: Keith R, Fandrick, Nitinchandra D, Patel, Suttipol, Radomkit, Arindom, Chatterjee, Stefan, Braith, Daniel R, Fandrick, Carl A, Busacca, Chris H, Senanayake
المصدر: The Journal of organic chemistry. 86(6)
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المؤلفون: Sergei Tcyrulnikov, Joshua D. Sieber, Nitinchandra D. Patel, Kendricks S. Lao, Marisa C. Kozlowski, Soumik Biswas, Chris H. Senanayake, Nelu Grinberg, Krishnaja Duvvuri, Neil K. Garg, B. Frank Gupton, Daniel Rivalti, Jinhua J. Song, Scott Pennino, Bo Qu, Heewon Lee, Donghong A. Gao, Yongda Zhang, Hari P. R. Mangunuru, Nizar Haddad, Bryan J. Simmons, Keith R. Fandrick
المصدر: ACS Catalysis. 8:10190-10209
مصطلحات موضوعية: biology, 010405 organic chemistry, Negishi coupling, chemistry.chemical_element, General Chemistry, 010402 general chemistry, biology.organism_classification, 01 natural sciences, Combinatorial chemistry, Catalysis, Reductive elimination, Coupling reaction, 0104 chemical sciences, Transmetalation, chemistry, Catalytic cycle, Tetra, Palladium
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المؤلفون: Nitinchandra D, Patel, Xudong, Wei, Denis, Byrne, Bikshandarkoil A, Narayanan, Scott, Pennino, Max, Sarvestani, Anjan, Saha, Nizar, Haddad, Suresh, Kapadia, Jon C, Lorenz, Philomen, DeCroos, Andrew, Ye, Heewon, Lee, Nelu, Grinberg, Azad, Hossain, Carl A, Busacca, Nathan K, Yee, Chris H, Senanayake
المصدر: The Journal of organic chemistry. 85(13)
مصطلحات موضوعية: Humans, Protease Inhibitors, Hepacivirus, Sulfones, Viral Nonstructural Proteins, Antiviral Agents, Hepatitis C, Ethers
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المؤلفون: Nitinchandra D. Patel, Marisa C. Kozlowski, Osvaldo Gutierrez, Chris H. Senanayake, Carl A. Busacca, Keith R. Fandrick, C. Avery Sader, Daniel R. Fandrick, Yike Zou
المصدر: Organic Letters
مصطلحات موضوعية: Letter, Molecular Structure, 010405 organic chemistry, Ligand, Chemistry, Site selectivity, Organic Chemistry, Ketones, Ligands, 010402 general chemistry, 01 natural sciences, Biochemistry, Combinatorial chemistry, Catalysis, 0104 chemical sciences, Alkadienes, Site selective, Organic chemistry, Physical and Theoretical Chemistry, Copper
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المؤلفون: Zhidong Chen, Carl A. Busacca, Shengli Ma, Xingzhong Zeng, Peter Allen Nemoto, Paige E. Mahaney, Jason A. Mulder, Chris H. Senanayake, Jun Wang, Nitinchandra D. Patel, Zhibin Li, Todd Bosanac, Daniel R. Fandrick, Jean-Nicolas Desrosiers, Heewon Lee, Sonia Rodriguez, Jon C. Lorenz, Nathan K. Yee, Joe Gao, Nelu Grinberg, Hidenori Takahashi, Alessandra Bartolozzi, Jinhua J. Song, Keith R. Fandrick
المصدر: Organic Process Research & Development. 21:1427-1434
مصطلحات موضوعية: Chromatography, biology, 010405 organic chemistry, Chemistry, Organic Chemistry, Structural component, 010402 general chemistry, 01 natural sciences, Combinatorial chemistry, 0104 chemical sciences, Supercritical fluid chromatography, biology.protein, Physical and Theoretical Chemistry, 5-lipoxygenase-activating protein
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المؤلفون: Daniel Rivalti, Carl A. Busacca, Bo Qu, Arindom Chatterjee, Nathan K. Yee, Nitinchandra D. Patel, Nizar Haddad, Chris H. Senanayake, Joshua D. Sieber, Frederic G. Buono, Sonia Rodriguez, Jean-Nicolas Desrosiers, Stefan Braith, Keith R. Fandrick, Heewon Lee
المصدر: Asian Journal of Organic Chemistry. 6:1285-1291
مصطلحات موضوعية: Green chemistry, 010405 organic chemistry, Chemistry, Ligand, Organic Chemistry, chemistry.chemical_element, 010402 general chemistry, Photochemistry, 01 natural sciences, Micelle, Coupling reaction, 0104 chemical sciences, Palladium
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المؤلفون: Heewon Lee, Nelu Grinberg, Nizar Haddad, Chris H. Senanayake, Nathan K. Yee, Joshua D. Sieber, Dmitry Kurouski, Nitinchandra D. Patel, Keith R. Fandrick, Jinhua J. Song, Bo Qu, Jean-Nicolas Desrosiers, Sonia Rodriguez, Hari P. R. Mangunuru
المصدر: Advanced Synthesis & Catalysis. 358:3522-3527
مصطلحات موضوعية: Coupling, Atropisomer, biology, 010405 organic chemistry, Stereochemistry, Ligand, Quinoline, General Chemistry, 010402 general chemistry, 01 natural sciences, 0104 chemical sciences, Integrase, chemistry.chemical_compound, chemistry, Suzuki reaction, biology.protein, Selectivity