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المؤلفون: Manav Korpal, Nathalie Rioux, O'shea Morgan Welzel, Pete Smith, Sherri Smith, Markus Warmuth, Sudeep Prajapati, Zheng Guo Zhu
المصدر: Cancer Chemotherapy and Pharmacology. 83:151-160
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Indazoles, SERCA, Metabolic Clearance Rate, Pyridines, CYP3A, Drug Evaluation, Preclinical, Biological Availability, Estrogen receptor, Plasma protein binding, In Vitro Techniques, Pharmacology, Toxicology, Rats, Sprague-Dawley, 03 medical and health sciences, Dogs, 0302 clinical medicine, Cytochrome P-450 Enzyme System, Species Specificity, Pharmacokinetics, medicine, Animals, Cytochrome P-450 Enzyme Inhibitors, Humans, Tissue Distribution, Pharmacology (medical), Cells, Cultured, Chemistry, Estrogen Receptor alpha, In vitro, Macaca fascicularis, 030104 developmental biology, medicine.anatomical_structure, Oncology, 030220 oncology & carcinogenesis, Hepatocyte, Hepatocytes, Microsomes, Liver, Female, Estrogen Receptor Antagonists, Drug metabolism, Protein Binding
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المؤلفون: Sean Eckley, Markus Warmuth, Ping Zhu, Deepti Banka, Zhenhua J. Wu, Nicholas A. Larsen, Sudeep Prajapati, Ricardo Ribas, Ming-Hong Hao, Pavan Kumar, Pete Smith, Michael J. Wick, Kiran Aithal, Crystal Mackenzie, John D. Norris, Sasirekha Sivakumar, V. Subramanian, Tuong-Vi Nguyen, Lihua Yu, Sean Irwin, Andrew Hart, Craig Furman, Alyssa Moriarty, Amy Kim, Benjamin Caleb, O'shea Morgan Welzel, Craig Karr, Sunil Pancholi, Frédéric H. Vaillancourt, Silvia Buonamici, Manav Korpal, Namita Kumar, Weidong G. Lai, Diana Melchers, Peter Fekkes, René Houtman, Lesley-Ann Martin, Xiaoling Puyang, Victoria Rimkunas, Michael Thomas, Amy Siu, Reynolds Dominic, Sujatha Rajagopalan, Suzanne E. Wardell, John Wang, Jaya Julie Joshi, Zheng Guo Zhu, David M. Bolduc, Nathalie Rioux, Subhasree Das, Sergei Agoulnik, Shihua Yao, Galina Kuznetsov
المصدر: Cancer Discovery. 8:1176-1193
مصطلحات موضوعية: 0301 basic medicine, Fulvestrant, Cell growth, business.industry, Estrogen receptor, Cancer, medicine.disease, Estrogen Receptor Antagonists, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Breast cancer, Oncology, In vivo, 030220 oncology & carcinogenesis, Cancer research, medicine, business, Estrogen receptor alpha, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::0120259fcf7ad9215e86543a6ac089d0
https://doi.org/10.1158/2159-8290.cd-17-1229 -
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المؤلفون: Sean Irwin, Guo-Zhu Zheng, Sherri Smith, Craig Furman, Deepti Banka, Nathalie Rioux, Victoria Rimkunas, J Norris, Prashant Kumar, Nicholas A. Larsen, Y Yu, Anand Selvaraj, Sergei Agoulnik, Craig Karr, Andrew Hart, T Bowser, Lorna Helen Mitchell, Crystal MacKenzie, Huilan Yao, Pete Smith, Tarek Sahmoud, Peter Fekkes, Jiayi Wu, T-V Nguyen, Zhaojie Zhang, Frédéric H. Vaillancourt, Betty Chan, Mike Thomas, Benjamin Caleb, O'shea Morgan Welzel, Manav Korpal, Markus Warmuth, Ping Zhu, S Wardell, Amy K. Kim, Galina Kuznetsov, Sean Eckley, Allison Davis, Sudeep Prajapati, Jun Wang, Ming-Hong Hao, V. Subramanian, Naresh Kumar, Xiaoling Puyang, Lihua Yu, Jaya Julie Joshi, Reynolds Dominic, G W Lai
المصدر: Cancer Research. 78:P1-10
مصطلحات موضوعية: Cancer Research, Fulvestrant, Chemistry, Antagonist, Estrogen receptor, medicine.disease, Breast cancer, Oncology, Mechanism of action, Cancer research, medicine, medicine.symptom, Receptor, Estrogen receptor alpha, Tamoxifen, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::07d855e8c12d90a391ebb18e38827bdf
https://doi.org/10.1158/1538-7445.sabcs17-p1-10-08 -
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المؤلفون: Markus Warmuth, Manav Korpal, Deepti Banka, Peter Fekkes, Pavan Kumar, Andrew Hart, Lihua Yu, Ping Zhu, Lorna Helen Mitchell, Joyce Yang, W. George Lai, Amy Kim, Craig Karr, Pete Smith, Tarek Sahmoud, Xiaoling Puyang, Sherri Smith, Mike Thomas, Benjamin Caleb, O'shea Morgan Welzel, Victoria Rimkunas, Huilan Yao, Sean Eckley, Allison Davis, Silvia Buonamici, Crystal MacKenzie, V. Subramanian, Jeremy Wu, Zheng Guo Zhu, Christopher Rowbottom, Reynolds Dominic, Nicholas A. Larsen, Nathalie Rioux, Sean Irwin, Craig Furman
المصدر: Cancer Research. 77:DDT01-04
مصطلحات موضوعية: Cancer Research, Fulvestrant, business.industry, 010401 analytical chemistry, Cancer, Estrogen receptor, Pharmacology, medicine.disease, 01 natural sciences, 0104 chemical sciences, 03 medical and health sciences, 0302 clinical medicine, Breast cancer, Oncology, Nuclear receptor, Selective estrogen receptor modulator, 030220 oncology & carcinogenesis, Medicine, business, Estrogen receptor beta, Tamoxifen, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::71b5b0fa7e9d8e6795b2dcf66171548d
https://doi.org/10.1158/1538-7445.am2017-ddt01-04 -
5
المؤلفون: Huiming Zhang, Linda Lee, Sudeep Prajapati, Betty Chan, Kazunobu Kira, Mingde Shan, Laura Corson, Ming-Hong Hao, Kuo-Ming Wu, O'shea Morgan Welzel, Yoshiharu Mizui, Samantha Perino, John Wang, Eun Sun Park, Lisa A. Marcaurelle, Marta Nevalainen, Arai Kenzo, Guo-Zhu Zheng, Markus Warmuth, Lihua Yu, Atsushi Endo, Jason T. Lowe, Xiang Liu, Baudouin Gerard, Pete Smith, Tivitmahaisoon Parcharee, Craig Karr, Silvia Buonamici, Keaney Gregg F, Tuoping Luo
المصدر: Organic Letters. 16:5560-5563
مصطلحات موضوعية: RNA Splicing Factors, Stereochemistry, RNA Splicing, Mutant, Antineoplastic Agents, Biochemistry, chemistry.chemical_compound, Cell Line, Tumor, Humans, Physical and Theoretical Chemistry, Cell Proliferation, Binding Sites, Natural product, Drug discovery, Cell growth, Organic Chemistry, Total synthesis, Ribonucleoprotein, U2 Small Nuclear, Phosphoproteins, chemistry, RNA splicing, Epoxy Compounds, Macrolides, Growth inhibition
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المؤلفون: Sherri Smith, Pete Smith, Ming-Hung Hao, John Wang, Nathalie Rioux, Sudeep Prajapati, Federico Colombo, O'shea Morgan Welzel, Darrel Nix, Markus Warmuth, Manav Korpal
المصدر: Drug Metabolism and Pharmacokinetics. 34:S22
مصطلحات موضوعية: Pharmacology, SERCA, Covalent bond, Chemistry, Antagonist, Biophysics, Pharmaceutical Science, Pharmacology (medical), In vitro in vivo
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7
المؤلفون: Lakshmi B. Akella, Eric N. Jacobsen, Etienne J. Donckele, O'shea Morgan Welzel, Baudouin Gerard, Sarathy Kesavan, Lisa A. Marcaurelle, Hao Xu
المصدر: ACS Combinatorial Science. 14:621-630
مصطلحات موضوعية: Chemistry, Stereoisomerism, General Chemistry, General Medicine, Quinolones, Combinatorial chemistry, Article, Catalysis, Stereocenter, Structure-Activity Relationship, Feasibility Studies, Urea, Organic chemistry, Povarov reaction
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المؤلفون: Jeremy R. Duvall, Sarathy Kesavan, Michael Foley, Byung-Chul Suh, O'shea Morgan Welzel, Jean-Charles Marie, Bérénice C. Lemercier, Bhaumik A. Pandya, Sivaraman Dandapani, Baudouin Gerard, Tiffanie Murillo, Lisa A. Marcaurelle, Mark E. Fitzgerald, Lakshmi B. Akella, Michael Dombrowski, Diane Hamann, Jason T. Lowe, Maurice D. Lee
المصدر: The Journal of organic chemistry. 78(11)
مصطلحات موضوعية: chemistry.chemical_classification, Scaffold, Stereochemistry, Organic Chemistry, Molecular Conformation, Glycoside, Stereoisomerism, respiratory system, Ring (chemistry), Article, chemistry.chemical_compound, chemistry, Pyran, Amide, Moiety, Amine gas treating, Glycosides, human activities, Pyrans
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9
المؤلفون: Mingde Shan, Samantha Perino, Zheng Guo Zhu, Linda Lee, Pete Smith, Eun Sun Park, Marta Nevalainen, Huiming Zhang, Kazunobu Kira, Markus Warmuth, Arai Kenzo, Atsushi Endo, Baudouin Gerard, Xiang Liu, Tivitmahaisoon Parcharee, Keaney Gregg F, Silvia Buonamici, Lihua Yu, Jason T. Lowe, John Wang, Craig Karr, Tuoping Luo, Laura Corson, Kuo-Ming Wu, Betty Chan, Lisa A. Marcaurelle, Sudeep Prajapati, Ming-Hong Hao, Yoshiharu Mizui, O'shea Morgan Welzel
المصدر: Cancer Research. 75:5564-5564
مصطلحات موضوعية: Genetics, Cancer Research, Spliceosome, Natural product, Mutant, Total synthesis, Biology, Inhibitory postsynaptic potential, chemistry.chemical_compound, Oncology, chemistry, RNA splicing, snRNP, Growth inhibition
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::d4b3f513df548c8caf875d85523e2a8a
https://doi.org/10.1158/1538-7445.am2015-5564 -
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