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1رسالة جامعية
المؤلفون: Cordón Barris, Lluís
المساهمون: University/Department: Universitat Autònoma de Barcelona. Departament de Bioquímica i Biologia Molecular
مرشدي الرسالة: llbarris@hotmail.com, Bayascas Ramírez, José Ramón
المصدر: TDX (Tesis Doctorals en Xarxa)
مصطلحات موضوعية: PDK1, PIF-pocket, Development neuronal, Desarrollo neuronal, Desenvolupament neuronal, Ciències Experimentals
وصف الملف: application/pdf
URL الوصول: http://hdl.handle.net/10803/308331
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2كتاب إلكتروني
المؤلفون: Leroux, Alejandro E.Aff5, Gross, Lissy Z. F.Aff5, Sacerdoti, MarianaAff5, Biondi, Ricardo M.Aff5, Aff6, Aff7, Aff8
المساهمون: LAMBRIS, JOHN D., Series EditorAff1, REZAEI, NIMA, Series EditorAff2, Zhang, Jian, editorAff3, Nussinov, Ruth, editorAff4
المصدر: Protein Allostery in Drug Discovery. 1163:279-311
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3دورية أكاديمية
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4دورية أكاديمية
المؤلفون: Guo, Gang, Yang, Cui, Li, Gao-Feng, Li, Heng, Ma, Qian-Li, Guo, Qi, Yang, Xiu-Mei
المصدر: Chemical Papers. September 2015 69(9):1253-1261
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5دورية أكاديمية
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المصدر: PLoS ONE
CONICET Digital (CONICET)
Consejo Nacional de Investigaciones Científicas y Técnicas
instacron:CONICET
PLoS ONE, Vol 15, Iss 11, p e0242819 (2020)مصطلحات موضوعية: Protein Extraction, Artificial Gene Amplification and Extension, Regulatory Sequences, Nucleic Acid, Biochemistry, Polymerase Chain Reaction, purl.org/becyt/ford/1 [https], Database and Informatics Methods, Phosphatidylinositol 3-Kinases, Protein Isoforms, PIF-pocket, PKB, Post-Translational Modification, Phosphorylation, Extraction Techniques, Messenger RNA, Precipitation Techniques, Nucleic acids, embryonic structures, Medicine, Sequence Analysis, Hydrophobic and Hydrophilic Interactions, Research Article, Signal Transduction, Bioinformatics, Science, Research and Analysis Methods, Transfection, splicing, Sequence Motif Analysis, Cell Line, Tumor, Genetics, Immunoprecipitation, Humans, ddc:610, Nucleotide Motifs, purl.org/becyt/ford/1.6 [https], Molecular Biology Techniques, Molecular Biology, Cell Proliferation, Akt, Biology and Life Sciences, Proteins, Alternative Splicing, HEK293 Cells, RNA processing, RNA, Gene expression, Proto-Oncogene Proteins c-akt
وصف الملف: application/octet-stream; application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::054dc5b232099dec17084413b56d3f8b
http://publikationen.ub.uni-frankfurt.de/frontdoor/index/index/docId/61113 -
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المؤلفون: Ricardo M. Biondi, Sonja Neimanis, Katrien Busschots, Pedro M. Alzari, Jörg O. Schulze, Evelyn Süß, Giorgio Saladino, Dalibor Odadzic, María-Natalia Lisa, Francesco Luigi Gervasio, Stefan Zeuzem, V. Hindie, Amanda K. Herbrand
المساهمون: Universitätsklinikum Frankfurt, University College of London [London] (UCL), Microbiologie structurale - Structural Microbiology (Microb. Struc. (UMR_3528 / U-Pasteur_5)), Institut Pasteur [Paris] (IP)-Université Paris Diderot - Paris 7 (UPD7)-Centre National de la Recherche Scientifique (CNRS), German Cancer Research Center - Deutsches Krebsforschungszentrum [Heidelberg] (DKFZ), The work was supported by BMBF GO-Bio (0315102), DFG BI 1044/2-3 and DFG BI 1044/12-1 (to R.M.B.) and in part by the Engineering and Physical Sciences Research Council (grant no. EP/M013898/1)., Université Paris Diderot - Paris 7 (UPD7)-Institut Pasteur [Paris]-Centre National de la Recherche Scientifique (CNRS)
المصدر: Cell Chemical Biology
Cell Chemical Biology, 2016, 23 (10), pp.1193-1205. ⟨10.1016/j.chembiol.2016.06.017⟩
Cell Chemical Biology, Cell Press, 2016, 23 (10), pp.1193-1205. ⟨10.1016/j.chembiol.2016.06.017⟩مصطلحات موضوعية: 0301 basic medicine, Clinical Biochemistry, PIF pocket, MESH: Allosteric Regulation, Biochemistry, MAP2K7, Adenosine Triphosphate, 0302 clinical medicine, Aurora Kinases, MESH: Adenosine Triphosphate, Drug Discovery, MESH: Protein Kinase Inhibitors, MESH: Allosteric Site, Aurora, [SDV.BBM.BS]Life Sciences [q-bio]/Biochemistry, Molecular Biology/Structural Biology [q-bio.BM], protein kinase, MESH: Pyruvate Dehydrogenase Acetyl-Transferring Kinase, MESH: Indazoles, ADENOSINE, Cell biology, Molecular Docking Simulation, ALLOSTERIC REGULATION, PDK1, adenosine, MESH: HEK293 Cells, 030220 oncology & carcinogenesis, Molecular Medicine, PIF POCKET, CIENCIAS NATURALES Y EXACTAS, Allosteric Site, AURORA, Indazoles, PROTEIN KINASE, Otras Ciencias Biológicas, [PHYS.PHYS.PHYS-BIO-PH]Physics [physics]/Physics [physics]/Biological Physics [physics.bio-ph], Allosteric regulation, [SDV.BC]Life Sciences [q-bio]/Cellular Biology, Protein Serine-Threonine Kinases, Biology, MESH: Protein-Serine-Threonine Kinases, Ciencias Biológicas, MESH: Aurora Kinases, 03 medical and health sciences, GSK2334470, MESH: Molecular Docking Simulation, [CHIM.CRIS]Chemical Sciences/Cristallography, Humans, [SDV.BBM]Life Sciences [q-bio]/Biochemistry, Molecular Biology, ddc:610, c-Raf, Binding site, Protein kinase A, Protein Kinase Inhibitors, Molecular Biology, Pharmacology, Binding Sites, MESH: Humans, small compounds, Cyclin-dependent kinase 2, Pyruvate Dehydrogenase Acetyl-Transferring Kinase, AGC kinase, SMALL COMPOUNDS, allosteric regulation, molecular dynamics, HEK293 Cells, Pyrimidines, 030104 developmental biology, MESH: Binding Sites, Allosteric enzyme, MESH: Pyrimidines, biology.protein, AGC KINASE, MOLECULAR DYNAMICS, Cyclin-dependent kinase 9, [INFO.INFO-BI]Computer Science [cs]/Bioinformatics [q-bio.QM]
وصف الملف: application/octet-stream; application/pdf
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المؤلفون: Alejandro E. Leroux, Ricardo M. Biondi, Jörg O. Schulze
المصدر: Seminars in Cancer Biology. 48:1-17
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, CIENCIAS MÉDICAS Y DE LA SALUD, PIF-POCKET, Allosteric regulation, Inmunología, Regulatory site, Protein Serine-Threonine Kinases, Biology, Serine, 03 medical and health sciences, Drug Discovery, Humans, AGC PROTEIN KINASE, Phosphorylation, Protein Kinase Inhibitors, Protein kinase B, Protein kinase C, rho-Associated Kinases, Drug discovery, Kinase, ALLOSTERIC, Pyruvate Dehydrogenase Acetyl-Transferring Kinase, DRUG DISCOVERY, Medicina Básica, 030104 developmental biology, Protein kinase domain, Biochemistry, REGULATION, Proto-Oncogene Proteins c-akt
وصف الملف: application/pdf
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المؤلفون: Simona Rapposelli, Simona Sestito
مصطلحات موضوعية: animal structures, Allosteric regulation, Antineoplastic Agents, Ligands, Metastasis, drug discovery, 3-Phosphoinositide-Dependent Protein Kinases, Patents as Topic, Adenosine Triphosphate, Drug Development, Neoplasms, medicine, metastasis, PH-domain inhibitor, Humans, Protein kinase A, Protein Kinase Inhibitors, Pharmacology, PDK1 inhibitor, Binding Sites, Drug discovery, business.industry, Kinase, Disease progression, chemoresistance, General Medicine, PI3K/PDK1/Akt pathway, medicine.disease, PIF-pocket inhibitor, 3-phosphoinositide-dependent kinase 1, Allosteric inhibitors, DFG-out inhibitor, Disease Progression, stomatognathic diseases, Drug development, Cancer research, Cancer development, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::41e2214e22dc68a772836660840c28b9
http://hdl.handle.net/11568/993542 -
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