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1دورية أكاديمية
المؤلفون: Bayliss, Martin K., Butler, James, Feldman, Paul L., Green, Darren V.S., Leeson, Paul D., Palovich, Michael R., Taylor, Anthony J.
المصدر: In Drug Discovery Today October 2016 21(10):1719-1727
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2
المؤلفون: Peter T. Buckley, James J. Foley, Edward F. Webb, Roderick S. Davis, Dulcie B. Schmidt, Jakob Busch-Petersen, Michael Salmon, Jian Jin, Widdowson Katherine L, Kristen E. Belmonte, Henry M. Sarau, Yonghui Wang, Qi Jin, Palovich Michael R, Ann M. Bullion
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:7087-7091
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Bronchi, Muscarinic Antagonists, Biochemistry, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Solid-phase synthesis, In vivo, Drug Discovery, Muscarinic acetylcholine receptor, Animals, Urea, Structure–activity relationship, Moiety, Ammonium, Tyrosine, Molecular Biology, Chemistry, Organic Chemistry, Receptors, Muscarinic, Quaternary Ammonium Compounds, Molecular Medicine
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3
المؤلفون: Paul D. Leeson, Martin K. Bayliss, Anthony J. Taylor, Paul L. Feldman, Palovich Michael R, James Butler, Darren V. S. Green
المصدر: Drug discovery today. 21(10)
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Chemistry, media_common.quotation_subject, Property distribution, Administration, Oral, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Risk analysis (engineering), Pharmaceutical Preparations, Solubility, 030220 oncology & carcinogenesis, Lipophilicity, Drug Discovery, Animals, Humans, Quality (business), Drug pipeline, Hydrophobic and Hydrophilic Interactions, Oral retinoid, media_common
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4
المؤلفون: Henry M. Sarau, Sandra Umbrecht, Widdowson Katherine L, Palovich Michael R, Michael Salmon, Haibo Xie, Hongxing Yan, Jakob Busch-Petersen, Mark A. Luttmann, James J. Foley, Brian Peck, Jeremy Dufour, Zehong Wan, Gerald E. Hunsberger, Philip S. Landis, Dramane I. Laine, Alicia M. Bacon, Miriam Burman, Edward F. Webb, Roderick S. Davis, Dulcie B. Schmidt
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:3366-3369
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Muscarinic Antagonists, Biochemistry, Mice, Structure-Activity Relationship, DAROTROPIUM, chemistry.chemical_compound, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Structure–activity relationship, Molecular Biology, Bronchial Diseases, Organic Chemistry, Muscarinic antagonist, Tropane, Receptors, Muscarinic, chemistry, Design synthesis, Drug Design, Molecular Medicine, Tropanes, medicine.drug
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5
المؤلفون: Roderick S. Davis, Emilie Veronique Petitjean, Jessica L. Schneck, Alicia Bacon Davis, Palovich Michael R, Haibo Xie, Deng Jianghe, Jim Villa, David Bettoun, Baoguang Zhao, Brian Peck, Robert Midgett, Patrick McDevitt, Casey Kmett, Dramane I. Laine, Neysa Nevins, Brent W. Mccleland, Lin Guoliang, Anais Jolit, Sandra Umbrecht, Isabelle Delhom
المصدر: ACS Medicinal Chemistry Letters. 2:142-147
مصطلحات موضوعية: Cathepsin, Organic Chemistry, Pharmacology, Biochemistry, Cysteine protease, Cathepsin C, chemistry.chemical_compound, Cathepsin O, chemistry, In vivo, Drug Discovery, Cigarette smoke, Cyanamide, Selectivity
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6
المؤلفون: Yonghui Wang, Henry M. Sarau, Dongchuan Shi, Dwight M. Morrow, Miriam Burman, Michael L. Moore, Palovich Michael R, Ralph A. Rivero, Edward F. Webb, Dramane I. Laine, Jian Jin, Brian Budzik, Kristen E. Belmonte, Feng Wang, James J. Foley, Haibo Xie, Michael Salmon, Chongye Zhu, Manuela Berlanga, Zehong Wan
المصدر: Journal of Medicinal Chemistry. 51:5915-5918
مصطلحات موضوعية: medicine.medical_specialty, Bronchoconstriction, Drug Evaluation, Preclinical, Pharmacology, Bronchial Provocation Tests, Piperazines, Bronchoconstrictor Agents, Mice, Structure-Activity Relationship, In vivo, Internal medicine, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Administration, Intranasal, Methacholine Chloride, Acetylcholine receptor, Molecular Structure, Chemistry, Antagonist, Muscarinic acetylcholine receptor M3, Stereoisomerism, Biological activity, Receptors, Muscarinic, Bronchodilator Agents, Disease Models, Animal, Endocrinology, Molecular Medicine, Nasal administration, medicine.symptom
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7
المؤلفون: Palovich Michael R, Miriam Burman, Edward F. Webb, Roderick S. Davis, Henry M. Sarau, Yonghui Wang, Wei Fu, Dwight M. Morrow, Jian Jin, Feng Wang, Qi Jin, Kristen E. Belmonte, Parvathi Rao, Michael L. Moore, Manuela Berlanga, James J. Foley, Chris J. Dehaas, Michael Salmon, Ralph A. Rivero, Lorena A. Kallal, Jakob Busch-Petersen, Dongchuan Shi
المصدر: Journal of Medicinal Chemistry. 51:4866-4869
مصطلحات موضوعية: medicine.drug_class, Bronchoconstriction, Guinea Pigs, Drug Evaluation, Preclinical, Muscarinic Antagonists, Pharmacology, Inhibitory postsynaptic potential, Mice, In vivo, Bronchodilator, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Acetylcholine receptor, Chemistry, Phenylurea Compounds, Antagonist, Bridged Bicyclo Compounds, Heterocyclic, Rats, Quaternary Ammonium Compounds, Biochemistry, Tyrosine, Molecular Medicine, Nasal administration, medicine.symptom
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المؤلفون: Widdowson Katherine L, Edward F. Webb, Palovich Michael R, James J. Foley, Kristen E. Belmonte, Haibo Xie, Peter T. Buckley, Noémie Buffet, Dramane I. Laine
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:6066-6069
مصطلحات موضوعية: Carbamate, medicine.medical_treatment, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Muscarinic Antagonists, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Mice, Pulmonary Disease, Chronic Obstructive, chemistry.chemical_compound, In vivo, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Receptor, Molecular Biology, Acetylcholine receptor, Molecular Structure, Chemistry, Organic Chemistry, Antagonist, Tropane, Bridged Bicyclo Compounds, Heterocyclic, Receptors, Muscarinic, Bronchodilator Agents, Molecular Medicine, Carbamates, Tropanes
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9
المؤلفون: Charles J. Kotzer, Palovich Michael R, Michael Salmon, Mark A. Luttmann, Victoria J. Barrett, Christopher J. DeHaas, Douglas W. P. Hay, Robert J. Slack, Dulcie B. Schmidt, Henry M. Sarau, Miriam Burman, Edward F. Webb, William L. Rumsey, James J. Foley, Dramane I. Laine, Peter T. Buckley
المصدر: The Journal of pharmacology and experimental therapeutics. 345(2)
مصطلحات موضوعية: Lung Diseases, Quinuclidines, Carbachol, Guinea Pigs, Scopolamine Derivatives, CHO Cells, Muscarinic Antagonists, Pharmacology, Umeclidinium bromide, Muscarinic Agonists, Cholinergic Antagonists, Mice, Cricetulus, Cricetinae, Muscarinic acetylcholine receptor, Administration, Inhalation, medicine, Animals, Tiotropium Bromide, Receptor, Lung, Receptor, Muscarinic M3, Mice, Inbred BALB C, Chemistry, Antagonist, Tiotropium bromide, Receptors, Muscarinic, Plethysmography, Kinetics, Molecular Medicine, Bronchoconstriction, Calcium, medicine.symptom, Acetylcholine, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b703d06aac0453f19e8ba31374b13055
https://pubmed.ncbi.nlm.nih.gov/23435542 -
10دورية أكاديمية
المؤلفون: Jin, Qi, Davis, Roderick S., Bullion, Ann M., Jin, Jian, Wang, Yonghui, Widdowson, Katherine L., Palovich, Michael R., Foley, James J., Schmidt, Dulcie B., Buckley, Peter T., Webb, Edward F., Salmon, Michael, Belmonte, Kristen E., Sarau, Henry M., Busch-Petersen, Jakob
المصدر: In Bioorganic & Medicinal Chemistry Letters 1 December 2012 22(23):7087-7091