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1
المؤلفون: Palucki Brenda, Patrick G. Pollard, Liangqin Guo, Tung M. Fong, Matthew J. Wyvratt, Randy R. Miller, Shuwen He, Constantin Tamvakopoulos, Iyassu K. Sebhat, Qianping Peng, Ravi P. Nargund, Zhixiong Ye, Airu S. Chen, Doreen E. Cashen, David H. Weinberg, Min K. Park, Raman K. Bakshi, D. Euan MacIntyre, Howard Y. Chen, Rui Tang, Tanya MacNeil, Qingmei Hong, Alison M. Strack, Ralph A. Stearns, Jian Liu, William J. Martin
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2330-2334
مصطلحات موضوعية: medicine.drug_class, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Biological Availability, Pharmaceutical Science, Carboxamide, Pharmacology, Biochemistry, Partial agonist, Piperazines, Rats, Sprague-Dawley, Eating, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Oral administration, In vivo, Drug Discovery, medicine, Animals, Urea, Obesity, Receptor, Molecular Biology, Organic Chemistry, Haplorhini, Rats, Disease Models, Animal, Piperazine, chemistry, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
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2
المؤلفون: Doreen E. Cashen, Constantin Tamvakopoulos, Qianping Peng, William J. Martin, David H. Weinberg, Charles Rosenblum, Arthur A. Patchett, Tanya MacNeil, Patrick G. Pollard, Zhixiong Ye, Raman K. Bakshi, Ralph A. Stearns, Rubana N. Kalyani, Palucki Brenda, Joseph M. Metzger, Alison M. Strack, Lex H.T. Van der Ploeg, D. Euan MacIntyre, Iyassu K. Sebhat, Aurawan Vongs, Airu S. Chen, Ravi P. Nargund, Liangqin Guo, Matthew J. Wyvratt, Randy R. Miller, Rui Tang, Howard Y. Chen, Khaled J. Barakat
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:3501-3505
مصطلحات موضوعية: Male, Agonist, Quinuclidines, Time Factors, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Rodentia, Carboxamide, Biochemistry, Chemical synthesis, Piperazines, Rats, Sprague-Dawley, Eating, Structure-Activity Relationship, Piperidines, In vivo, Drug Discovery, medicine, Animals, Humans, Receptor, Molecular Biology, Aza Compounds, Bicyclic molecule, Chemistry, Penile Erection, digestive, oral, and skin physiology, Organic Chemistry, Small molecule, Rats, Microsomes, Liver, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin, Protein Binding
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3
المؤلفون: George A. Doss, Lex H.T. Van der Ploeg, Qianping Peng, Ravi P. Nargund, Charles Rosenblum, Randall R. Miller, Aurawan Vongs, Palucki Brenda, Tanya MacNeil, Ralph A. Stearns, Min K. Park, David H. Weinberg, Rui Tang, Arthur A. Patchett, Constantin Tamvakopoulos
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:1993-1996
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Piperazines, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Receptor, Molecular Biology, biology, Chemistry, Organic Chemistry, biology.organism_classification, In vitro, Piperazine, Microsoma, Microsome, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
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4
المؤلفون: William J. Martin, D. Euan MacIntyre, Ravi P. Nargund, Rubana N. Kalyani, Rui Tang, George A. Doss, Min K. Park, Alison M. Strack, Erin McGowan, Joseph M. Metzger, Charles Rosenblum, Randall R. Miller, Palucki Brenda, Qianping Peng, Arthur A. Patchett, Ralph A. Stearns, Patrick G. Pollard, Lex H.T. Van der Ploeg, Iyassu K. Sebhat, Constantin Tamvakopoulos, Cherrie Shepherd, Aurawan Vongs, Tanya MacNeil, David H. Weinberg, Zhixiong Ye
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:171-175
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Piperazines, Mice, Dogs, Erectile Dysfunction, Piperidines, In vivo, Drug Discovery, medicine, Animals, Obesity, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Haplorhini, In vitro, Rats, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
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5
المؤلفون: Ralph A. Stearns, Randy R. Miller, William J. Martin, Ravi P. Nargund, Erin McGowan, Lex H.T. Van der Ploeg, and Arthur A. Patchett, Andrew D. Howard, David B. R. Johnston, D. Euan MacIntyre, Rubana N. Kalyani, Khaled Barakat, Raman K. Bakshi, Ralph T. Mosley, Jennifer E. Drisko, Constantin Tamvakopoulos, Rui Tang, Alison M. Strack, Zhixiong Ye, Doreen E. Cashen, Tanya MacNeil, David H. Weinberg, Palucki Brenda, Gary J Hom, Iyassu K. Sebhat
المصدر: Journal of Medicinal Chemistry. 45:4589-4593
مصطلحات موضوعية: Agonist, Chemistry, medicine.drug_class, Biological activity, Pharmacology, Melanocortin receptor, THIQ, Drug Discovery, medicine, Anorectic, Molecular Medicine, Structure–activity relationship, Melanocortin, Receptor, medicine.drug
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6
المؤلفون: Ravi P. Nargund, Ralph A. Stearns, Constantin Tamvakopoulos, Palucki Brenda, Patrick R. Griffin, Xiaolan Shen, Judy Fenyk-Melody, Lawrence F. Colwell, Iyassu K. Sebhat, Khaled J. Barakat
المصدر: Rapid Communications in Mass Spectrometry. 14:1729-1735
مصطلحات موضوعية: Drug, Analyte, Chromatography, Drug discovery, Chemistry, media_common.quotation_subject, Organic Chemistry, Penetration (firestop), Plasma, Tandem mass spectrometry, Analytical Chemistry, Liquid chromatography–mass spectrometry, Dosing, Spectroscopy, media_common
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::4a381ac391dae1705c2296fdc228755d
https://doi.org/10.1002/1097-0231(20001015)14:19<1729::aid-rcm85>3.0.co;2-5 -
7دورية أكاديمية
المؤلفون: Hong, Qingmei, Bakshi, Raman K., Palucki, Brenda L., Park, Min K., Ye, Zhixiong, He, Shuwen, Pollard, Patrick G., Sebhat, Iyassu K., Liu, Jian, Guo, Liangqin, Cashen, Doreen E., Martin, William J., Weinberg, David H., MacNeil, Tanya, Tang, Rui, Tamvakopoulos, Constantin, Peng, Qianping, Miller, Randy R., Stearns, Ralph A., Chen, Howard Y., Chen, Airu S., Strack, Alison M., Fong, Tung M., MacIntyre, D. Euan, Wyvratt, Matthew J., Nargund, Ravi P.
المصدر: In Bioorganic & Medicinal Chemistry Letters 2011 21(8):2330-2334
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8
المؤلفون: Sheng-Shung Pong, Arthur A. Patchett, Carina P. Tan, Karen K. McKee, Lex H.Y. Van der Ploeg, Palucki Brenda, Donna L. Hreniuk, Ravi P. Nargund, Scott D. Feighner, Andrew D. Howard
المصدر: Bioorganicmedicinal chemistry letters. 11(14)
مصطلحات موضوعية: Indoles, Luminescence, Stereochemistry, Peptide Hormones, Clinical Biochemistry, Pharmaceutical Science, Peptide, Receptors, Cell Surface, Tripeptide, Peptide hormone, Biochemistry, Receptors, G-Protein-Coupled, chemistry.chemical_compound, Inhibitory Concentration 50, Piperidines, Drug Discovery, Humans, Spiro Compounds, Receptors, Ghrelin, Molecular Biology, Cells, Cultured, chemistry.chemical_classification, Binding Sites, Tetrapeptide, Chemistry, Organic Chemistry, Molecular Mimicry, In vitro, Ghrelin, Indoline, Molecular Medicine, Calcium, Piperidine, Peptides, hormones, hormone substitutes, and hormone antagonists, Protein Binding
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9دورية أكاديمية
المؤلفون: Palucki, Brenda L. *, Park, Min K., Nargund, Ravi P., Ye, Zhixiong, Sebhat, Iyassu K., Pollard, Patrick G., Kalyani, Rubana N., Tang, Rui, MacNeil, Tanya, Weinberg, David H., Vongs, Aurawan, Rosenblum, Charles I., Doss, George A., Miller, Randall R., Stearns, Ralph A., Peng, Qianping, Tamvakopoulos, Constantin, McGowan, Erin, Martin, William J., Metzger, Joseph M., Shepherd, Cherrie A., Strack, Alison M., MacIntyre, D. Euan, Van der Ploeg, Lex H.T., Patchett, Arthur A.
المصدر: In Bioorganic & Medicinal Chemistry Letters 2005 15(1):171-175
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10دورية أكاديمية
المؤلفون: Ye, Zhixiong, Guo, Liangqin, Barakat, Khaled J., Pollard, Patrick G., Palucki, Brenda L., Sebhat, Iyassu K., Bakshi, Raman K., Tang, Rui, Kalyani, Rubana N., Vongs, Aurawan, Chen, Airu S., Chen, Howard Y., Rosenblum, Charles I., MacNeil, Tanya, Weinberg, David H., Peng, Qianping, Tamvakopoulos, Constantin, Miller, Randy R., Stearns, Ralph A., Cashen, Doreen E., Martin, William J., Metzger, Joseph M., Strack, Alison M., MacIntyre, D. Euan, Van der Ploeg, Lex H.T., Patchett, Arthur A., Wyvratt, Matthew J., Nargund, Ravi P.
المصدر: In Bioorganic & Medicinal Chemistry Letters 2005 15(15):3501-3505