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المؤلفون: Robert J. Ternansky, Patricia L. Gladstone, Zhuoqi Zhang, Graham Parry, Fernando Donate, Renzhong Fu, Jose Juarez, Amy L. Allan, Jinbao Xiang, Andrew P. Mazar, Xu Bai
المصدر: MedChemComm. 7:1946-1951
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, chemistry.chemical_classification, 010405 organic chemistry, Kinase Family, Drug discovery, Kinase, Stereochemistry, Organic Chemistry, Pharmaceutical Science, Biology, 01 natural sciences, Biochemistry, In vitro, 0104 chemical sciences, 03 medical and health sciences, 030104 developmental biology, Enzyme, chemistry, Drug Discovery, Molecular Medicine, Phosphorylation, IC50, Tricyclic
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::6d5f7ca18a4f4a40c7af850c56c2e9e9
https://doi.org/10.1039/c6md00351f -
2
المؤلفون: Kevin J. Tomaselli, Julia Herrmann, Robert O. Sayers, Joe C. Wu, Lalitha Kodandapani, Kathy G. Jahangiri, Craig D. Fisher, David T. Winn, Edward D. Robinson, Steven P. Meduna, Robert J. Ternansky, Pauline Yeo, Karen L. Valentino, Jose-Luis Diaz, Vincent J. Kalish, Steven D. Linton, Kristen Sebring, Robert A. Armstrong, Joseph F. Krebs, Niel C. Hoglen, Alfred P. Spada, Brad P. Hirakawa, Ning Chen, Brett R. Ullman, Brett Weylan Ching, Cheng-zhi Zhang, Xu Bai, Xin Gu, Kip Nalley, Long-Shiuh Chen, Patricia L. Gladstone, Jeff McQuiston, Teresa Aja, Todd Groessl, Donald S. Karanewsky, Suzanne Weeks, Lawrence C. Fritz, Patricia C. Contreras
المصدر: Journal of Medicinal Chemistry. 48:6779-6782
مصطلحات موضوعية: Adult, Biological Availability, Phases of clinical research, Apoptosis, Pharmacology, Jurkat Cells, Mice, Structure-Activity Relationship, Liver disease, Pharmacokinetics, In vivo, Drug Discovery, medicine, Animals, Humans, Aspartate Aminotransferases, Pentanoic Acids, Caspase, Liver injury, Cholestasis, Clinical Trials, Phase I as Topic, biology, Caspase 3, Chemistry, Liver Diseases, Alanine Transaminase, Hepatitis C, Chronic, medicine.disease, Caspase Inhibitors, In vitro, Rats, Liver, Biochemistry, Enzyme inhibitor, Hepatocytes, biology.protein, Molecular Medicine, Half-Life
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المؤلفون: Wayne C. Guida, Robert J. Ternansky, Fernando Donate, Jason A Nydick, Patricia L. Gladstone, Tara E. Jackson, Jose Juarez, Melissa L. P. Price
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:107-110
مصطلحات موضوعية: Models, Molecular, Molecular model, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Guanidines, Biochemistry, Chemical synthesis, Drug Discovery, Humans, Computer Simulation, Homology modeling, Enzyme Inhibitors, Thymidine phosphorylase, Molecular Biology, chemistry.chemical_classification, Thymidine Phosphorylase, Binding Sites, biology, Bicyclic molecule, Chemistry, Organic Chemistry, Enzyme, Structural Homology, Protein, Docking (molecular), Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Protein Binding
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المؤلفون: Edward Piers, James G. K. Yee, Patricia L. Gladstone
المصدر: Organic Letters. 2:481-484
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, chemistry, Aryl, Intramolecular force, Organic Chemistry, chemistry.chemical_element, Oxidative coupling of methane, Physical and Theoretical Chemistry, Biochemistry, Carbon, Medicinal chemistry, Tricyclic
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المصدر: Tetrahedron. 54:10609-10626
مصطلحات موضوعية: chemistry, Organic Chemistry, Drug Discovery, Intermolecular force, Polymer chemistry, Conjugated diene, chemistry.chemical_element, Organic chemistry, Biochemistry, Copper
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المؤلفون: Patricia L. Gladstone, Thomas G. Back
المصدر: ChemInform. 25
مصطلحات موضوعية: Stereochemistry, Chemistry, General Medicine, Radical cyclization
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المصدر: ChemInform. 29
مصطلحات موضوعية: Chemistry, Intermolecular force, Polymer chemistry, Conjugated diene, chemistry.chemical_element, General Medicine, Copper
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المؤلفون: James G. K. Yee, Edward Piers, Patricia L. Gladstone
المصدر: ChemInform. 31
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, chemistry, Intramolecular force, Aryl, Polymer chemistry, chemistry.chemical_element, Oxidative coupling of methane, General Medicine, Carbon, Tricyclic
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المؤلفون: David H. Jones, Aleksander W. Roszak, Penelope W. Codding, Joseph H.-L. Chau, Patricia L. Gladstone, Jacek W. Morzycki, Thomas G. Back
المصدر: The Journal of Organic Chemistry. 57:4110-4121
مصطلحات موضوعية: Azasteroids, chemistry.chemical_compound, Stereospecificity, Molecular model, Chemistry, Stereochemistry, Organic Chemistry, Leaving group, Lactam, Nucleofuge, Nuclear magnetic resonance spectroscopy, Enone
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::f43535372c3066aba2e66e4ddf3aa8fb
https://doi.org/10.1021/jo00041a013 -
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المؤلفون: Bruce Ganem, Fernando Donate, Amy L. Allan, Steven Ealick, Stephanie A. Hopkins, David E. Shaw, Yingbo Li, Weiru Wang, Melissa L. P. Price, Robert J. Ternansky, Jose C. Juarez, Patricia L. Gladstone
المصدر: Journal of medicinal chemistry. 49(26)
مصطلحات موضوعية: chemistry.chemical_classification, Models, Molecular, Thymidine Phosphorylase, Pyrimidine, Bicyclic molecule, Molecular Structure, Stereochemistry, Biological activity, Bridged Bicyclo Compounds, Heterocyclic, Pyrimidine Nucleosides, Phosphonate, chemistry.chemical_compound, Structure-Activity Relationship, Enzyme, chemistry, Biochemistry, Drug Discovery, Molecular Medicine, Structure–activity relationship, Humans, Thymidine phosphorylase, Enzyme Inhibitors, Nucleoside