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المؤلفون: Mark A. Nagy, Robert Hilgraf, Deborah S. Mortensen, Jan Elsner, Stephen Norris, Jayashree Tikhe, Won Yoon, David Paisner, Mercedes Delgado, Paul Erdman, Jason Haelewyn, Godrej Khambatta, Li Xu, William J. Romanow, Kevin Condroski, Sogole Bahmanyar, Meg McCarrick, Brent Benish, Kate Blease, Laurie LeBrun, Mehran F. Moghaddam, Julius Apuy, Stacie S. Canan, Brydon L. Bennett, Yoshitaka Satoh
المصدر: Journal of Medicinal Chemistry. 64:18193-18208
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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المؤلفون: Leah Fung, Hans C. Lee, Richard J. Jones, Frank Mercurio, Robert W. Sullivan, Imelda Lam, David I. Stirling, Fazal Shirazi, Jianxuan Zou, Paul Erdman, David Hecht, Hua Wang, Normand Richard, Kyle W. H. Chan, Brooke McElwee, Aparajita Hoskote Chourasia, Elisabet E. Manasanch, Isere Kuiatse, Robert Z. Orlowski, Eduardo Torres
المصدر: Journal of Molecular Medicine. 98:1161-1173
مصطلحات موضوعية: Ubiquitin-Protein Ligases, Antineoplastic Agents, Apoptosis, Bortezomib, Mice, 03 medical and health sciences, 0302 clinical medicine, In vivo, Cell Line, Tumor, hemic and lymphatic diseases, Drug Discovery, Biomarkers, Tumor, medicine, Animals, Humans, Lenalidomide, Genetics (clinical), Multiple myeloma, Dexamethasone, Cell Proliferation, Chemistry, Cereblon, medicine.disease, Pomalidomide, Thalidomide, Disease Models, Animal, Drug Resistance, Neoplasm, Proteostasis, Cancer research, Molecular Medicine, Multiple Myeloma, 030215 immunology, medicine.drug
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المؤلفون: Aparajita Hoskote Chourasia, Hannah Majeski, Angela Pasis, Paul Erdman, Ashwini Oke, David Hecht, David Lonergan, Frank Mercurio, Kyle Chan, Dung Luong Thai, Leah Fung
المصدر: Journal of Clinical Oncology. 40:7025-7025
مصطلحات موضوعية: Cancer Research, Oncology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::8e1b6705c27eeba185d511f792b0eec0
https://doi.org/10.1200/jco.2022.40.16_suppl.7025 -
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المؤلفون: David Hecht, Kyle Chan, Paul Erdman, Eduardo Torres, yinon Ben-Neriah, Brooke McElwee, Frank Mercurio, Aparajita Chourasia, Leah Fung, Robert Sullivan, Imelda Calderon
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1cbce36130955bb33ebe35f3bdfe327d
https://doi.org/10.1021/scimeetings.0c07400 -
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المصدر: ACS Med Chem Lett
مصطلحات موضوعية: 010405 organic chemistry, Drug discovery, Chemistry, Organic Chemistry, 01 natural sciences, Biochemistry, Combinatorial chemistry, Pyrrolidine, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, 3d space, Drug Discovery, Lead compound
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المؤلفون: Guy Brachya, Yinon Ben-Neriah, Moshe Oren, Liran I. Shlush, Itay Omer, Amitai Rivlin, Robert W. Sullivan, Eli Pikarsky, Nathali Kaushansky, Li Dansu, Adar Zinger, Frank Mercurio, Ross L. Levine, Eitan Winter, Waleed Minzel, Ido Burstain, Avanthika Venkatachalam, Joseph Vacca, Leah Fung, Eric Hung, Maya Shaham, Irit Snir-Alkalay, Avner Fink, Paul Erdman, Shlomo Elias
مصطلحات موضوعية: 0301 basic medicine, Kinase, Myeloid leukemia, Biology, medicine.disease, General Biochemistry, Genetics and Molecular Biology, Article, 3. Good health, 03 medical and health sciences, Haematopoiesis, Leukemia, Leukemia, Myeloid, Acute, 030104 developmental biology, Apoptosis, hemic and lymphatic diseases, Cancer research, medicine, Humans, Cyclin-dependent kinase 9, Progenitor cell, Cyclin-dependent kinase 7, Tumor Suppressor Protein p53
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e2440625cc9c49007ec76bcf64decbae
https://europepmc.org/articles/PMC6701634/ -
9Discovery of N-substituted 7-azaindoles as Pan-PIM kinases inhibitors - Lead optimization - Part III
المؤلفون: Andrew Hebert, Paul Erdman, Maniar Sachin, Anlai Wang, Alexandre Gross, Elina Tserlin, Claude Barberis, Vinod F. Patel, Jiang John Z, Mark Czekaj, Mikhail Levit, James Pribish, Frank Sun, Matthieu Barrague, Luke Fire, Shih-Min A. Huang
المصدر: Bioorganicmedicinal chemistry letters. 29(3)
مصطلحات موضوعية: Indoles, Clinical Biochemistry, hERG, Compound 17, Pharmaceutical Science, Antineoplastic Agents, 01 natural sciences, Biochemistry, Part iii, Mice, Structure-Activity Relationship, Proto-Oncogene Proteins c-pim-1, Cell Line, Tumor, Drug Discovery, Animals, Humans, Molecular Biology, Protein Kinase Inhibitors, Cell Proliferation, biology, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Chemistry, Organic Chemistry, Neoplasms, Experimental, Combinatorial chemistry, 0104 chemical sciences, Rats, 010404 medicinal & biomolecular chemistry, Pim kinases, biology.protein, Molecular Medicine, Tumor growth inhibition, Drug Screening Assays, Antitumor
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المؤلفون: Sachin Maniar, Anlai Wang, James Pribish, Shih-Min A. Huang, Andrew Hebert, Mikhail Levit, Jinyu Liu, Claude Barberis, Luke Fire, Elina Tserlin, Paul Erdman, Vinod F. Patel, Mark Czekaj, Joseph D. Batchelor, Frank Sun
المصدر: Bioorganic & Medicinal Chemistry Letters. 30:127625
مصطلحات موضوعية: Indoles, Pyrrolidines, Clinical Biochemistry, hERG, Pharmaceutical Science, Antineoplastic Agents, Crystallography, X-Ray, 01 natural sciences, Biochemistry, Mice, Piperidines, Proto-Oncogene Proteins c-pim-1, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Tumor growth, Protein Kinase Inhibitors, Molecular Biology, PK/PD models, Aza Compounds, biology, 010405 organic chemistry, Chemistry, Kinase, Organic Chemistry, Cancer, Stereoisomerism, medicine.disease, Xenograft Model Antitumor Assays, Rats, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Permeability (electromagnetism), biology.protein, Cancer research, Molecular Medicine, Tumor growth inhibition, Protein Binding