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1
المؤلفون: Ujjini H. Manjunatha, Christel Brunschwig, Mathew Njoroge, Srinivasa P. S. Rao, Nina Lawrence, Dale Taylor, Rudolf Müller, Kelly Chibale, Paul M. Njaria, Renier van der Westhuyzen, Vinayak Singh, Leslie J. Street, Amanda Mabhula, Atica Moosa, Digby F. Warner, Denis Ngumbu Muhunga, Paul W. Smith
المصدر: Journal of Medicinal Chemistry. 64:9444-9457
مصطلحات موضوعية: 0303 health sciences, Carbamate, biology, Chemistry, medicine.medical_treatment, hERG, Prodrug, biology.organism_classification, Oxime, 01 natural sciences, 0104 chemical sciences, Mycobacterium tuberculosis, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, Mechanism of action, Biochemistry, Drug Discovery, medicine, biology.protein, Molecular Medicine, Structure–activity relationship, medicine.symptom, Mode of action, 030304 developmental biology
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2
المؤلفون: Anthony J. Smith, Dale Taylor, Anne J. Lenaerts, Thomas R. Ioerger, Nina Lawrence, Kelly Chibale, Rudolf Mueller, Vinayak Singh, Claire Le Manach, Aloysius T. Nchinda, Alissa Myrick, Mathew Njoroge, Paul M. Njaria, Elizabeth J. Brooks, Atica Moosa, Jessica N. Akester, Gregory T. Robertson
المصدر: ACS Infectious Diseases
مصطلحات موضوعية: 0301 basic medicine, medicine.drug_class, 030106 microbiology, Mutant, Antitubercular Agents, Antimycobacterial, Article, Sulfone, drug discovery, 03 medical and health sciences, chemistry.chemical_compound, Mice, Structure-Activity Relationship, In vivo, medicine, Glycerol, Structure–activity relationship, Animals, 2-aminoquinazolinones, Mycobacterium tuberculosis, In vitro, 030104 developmental biology, Infectious Diseases, chemistry, Biochemistry, Mechanism of action, tuberculosis, Drug Design, medicine.symptom
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3
المؤلفون: Renier, van der Westhuyzen, Amanda, Mabhula, Paul M, Njaria, Rudolf, Müller, Denis, Ngumbu Muhunga, Dale, Taylor, Nina, Lawrence, Mathew, Njoroge, Christel, Brunschwig, Atica, Moosa, Vinayak, Singh, Srinivasa P S, Rao, Ujjini H, Manjunatha, Paul W, Smith, Digby F, Warner, Leslie J, Street, Kelly, Chibale
المصدر: Journal of medicinal chemistry. 64(13)
مصطلحات موضوعية: Structure-Activity Relationship, Dose-Response Relationship, Drug, Molecular Structure, Heterocyclic Compounds, Oximes, Antitubercular Agents, Carbamates, Microbial Sensitivity Tests, Mycobacterium tuberculosis
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4
المؤلفون: Agnes W. Mathenge, Paul M. Njaria, Alex Njoroge Mwangi, Shital M. Maru, Geoffrey Kabue Kiriiri, Nicholas M. Njuguna, Peter M. Njogu
المصدر: Saudi Pharmaceutical Journal : SPJ
مصطلحات موضوعية: Product optimization, Pharmacology, Drug, Chromatography, media_common.quotation_subject, Pharmaceutical Science, Factorial experiment, In vivo anti-inflammatory, medicine.disease, Alternative treatment, Carrageenan, chemistry.chemical_compound, Meloxicam, chemistry, Formulation design, In vivo, medicine, Original Article, Meloxicam emulgels, Capsaicin fixed-dose combination, Menthol, Rheumatism, media_common, medicine.drug
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المؤلفون: Paul M. Njaria, Kennedy O. Abuga, FN Kamau, HK Chepkwony
المصدر: Chromatographia. 79:1507-1514
مصطلحات موضوعية: Guaifenesin, Chromatography, Chemistry, Bromhexine, 010401 analytical chemistry, Organic Chemistry, Clinical Biochemistry, Terbutaline, Ambroxol, Pseudoephedrine, 030226 pharmacology & pharmacy, 01 natural sciences, Biochemistry, High-performance liquid chromatography, 0104 chemical sciences, Analytical Chemistry, 03 medical and health sciences, 0302 clinical medicine, medicine, Triprolidine, medicine.drug, Chlorpheniramine Maleate
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6
المؤلفون: Nicholas M. Njuguna, Paul M. Njaria, Kelly Chibale, John Okombo
المصدر: Expert Opinion on Therapeutic Patents
مصطلحات موضوعية: hydroxychloroquine, Plasmodium falciparum, malaria, repurposing, Review, chloroquine derivatives, Pharmacology, Patents as Topic, Aminoquinoline, Antimalarials, Chloroquine, Drug Discovery, medicine, cancer, Animals, Humans, Repurposing, Biological evaluation, repositioning, antimalarial, biology, business.industry, Drug Repositioning, Stereoisomerism, aminoquinoline, General Medicine, biology.organism_classification, medicine.disease, patent, Drug Design, business, Malaria, medicine.drug