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1
المؤلفون: Giovanna Bergamini, Stefano Livia, Kenneth David Down, Marcus Bantscheff, Nick Barton, Friedrich B M Reinhard, Paola Grandi, Daniel Thomas, David N. Mallett, Paul Martin Gore, Sophie M. Bertrand, Z.A. Henley, Edith M. Hessel, James E. Rowedder, Mark Price, J. Nicole Hamblin, Birgit Dümpelfeld, Augustin Amour, Steve Keeling, Christina Rau, Máire A. Convery, Chris D. Edwards, Jonathan A. Taylor, Paul Rowland, Aoife C. Maxwell
المصدر: Journal of Medicinal Chemistry. 63:638-655
مصطلحات موضوعية: Models, Molecular, Cell Membrane Permeability, Cell membrane permeability, Class I Phosphatidylinositol 3-Kinases, Biological Availability, Class iii, Crystallography, X-Ray, Binding, Competitive, Structure-Activity Relationship, Drug Discovery, Animals, Humans, Structure–activity relationship, Potency, Phosphoinositide-3 Kinase Inhibitors, Drug discovery, Chemistry, Class III Phosphatidylinositol 3-Kinases, Combinatorial chemistry, Rats, Bioavailability, Isoenzymes, Molecular Docking Simulation, Toxicity, Molecular Medicine, Selectivity
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2
المؤلفون: Kenneth L. Clark, Paul Martin Gore, Panayiotis A. Procopiou, Simon Teanby Hodgson, Alison J. Ford, Clarissa J. Watts, Robert J. Slack, Duncan S. Holmes, Brian Edgar Looker, Ken A. Saunders, Ashley Paul Hancock, Sadie Vile
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:4914-4919
مصطلحات موضوعية: 0301 basic medicine, CYP3A4, Chemistry, Organic Chemistry, Clinical Biochemistry, Sulfonamide (medicine), Pharmaceutical Science, Sulfanilamide, Histamine H1 receptor, Pharmacology, Histamine H1 Antagonists, Biochemistry, Azelastine, Bioavailability, 03 medical and health sciences, 030104 developmental biology, Drug Discovery, medicine, Molecular Medicine, Nasal administration, Molecular Biology, medicine.drug
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3
المؤلفون: Robert J. Slack, Brian Edgar Looker, Sadie Vile, Duncan S. Holmes, Kenneth L. Clark, Clarissa J. Watts, Simon Teanby Hodgson, Panayiotis A. Procopiou, Paul Martin Gore, Ken A. Saunders, Alison J. Ford, James E. Rowedder
المصدر: ACS Medicinal Chemistry Letters. 8:577-581
مصطلحات موضوعية: 0301 basic medicine, Histamine H1 Receptor Antagonists, medicine.medical_specialty, 010405 organic chemistry, Chemistry, Organic Chemistry, Pharmacology, 01 natural sciences, Biochemistry, Azelastine, In vitro, 0104 chemical sciences, Bioavailability, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, Endocrinology, In vivo, Internal medicine, Amide, Drug Discovery, medicine, Nasal administration, Dosing, medicine.drug
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4
المؤلفون: Steven Philip Keeling, Nigel J. Parr, Simon Teanby Hodgson, Ashley Paul Hancock, Duncan S. Holmes, Panayiotis A. Procopiou, James E. Rowedder, Brian Edgar Looker, Robert J. Slack, Paul Martin Gore, Rachael A. Ancliff
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:5855-5859
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Histamine Receptor Antagonists, Pharmacology, 01 natural sciences, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, medicine, Potency, Receptor, Molecular Biology, biology, Chemistry, Organic Chemistry, Quinoline, Azelastine, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 030104 developmental biology, biology.protein, Molecular Medicine, Nasal administration, medicine.drug
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5
المؤلفون: Duncan S. Holmes, Mark J. Bamford, P. Ward, Paul Martin Gore, Jeremy C. Prodger, Victoria Saez
المصدر: Tetrahedron Letters. 36:2339-2342
مصطلحات موضوعية: carbohydrates (lipids), chemistry.chemical_compound, Sialyl-Lewis X, chemistry, Stereochemistry, Organic Chemistry, Drug Discovery, Biochemistry, Sialic acid
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6
المؤلفون: Christopher Browning, Panayiotis A. Procopiou, Paul Martin Gore, Robert J. Slack, Sean M. Lynn, Stephen A. Richards, Steven L. Sollis
المصدر: Bioorganicmedicinal chemistry. 20(20)
مصطلحات موضوعية: ERG1 Potassium Channel, Ketone, Stereochemistry, medicine.drug_class, Pyridines, Clinical Biochemistry, Substituent, Pharmaceutical Science, Stereoisomerism, Biochemistry, Pyrrolidine, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Humans, Receptors, Histamine H1, Molecular Biology, chemistry.chemical_classification, Chemistry, Organic Chemistry, Receptor antagonist, Ether-A-Go-Go Potassium Channels, Pyridazines, Pyrazines, Lipophilicity, Histamine H1 Antagonists, Molecular Medicine, Phthalazines, Mitsunobu reaction, Stereoselectivity, Protein Binding
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7
المؤلفون: Andrew B. McElroy, Paul Martin Gore, P. Ward, Anthony William James Cooper, P.W. Smith, Hilary S. Adams, Richard W. Bell, John Martin Pritchard
المصدر: Bioorganic & Medicinal Chemistry Letters. 4:1951-1956
مصطلحات موضوعية: Chemistry, Stereochemistry, medicine.drug_class, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Nk2 receptor, Pharmacology, Receptor antagonist, Biochemistry, Non peptide, Orally active, Drug Discovery, medicine, Molecular Medicine, Bronchoconstriction, medicine.symptom, Receptor, Molecular Biology
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8
المؤلفون: Linda J. Russell, Paul Martin Gore, Simon Teanby Hodgson, Ashley Paul Hancock, Robert J. Slack, Jennifer M. Buckley, Sadie Vile, Michael Kranz, Steven L. Sollis, Kenneth L. Clark, Brian Edgar Looker, Panayiotis A. Procopiou, Clarissa J. Watts, Duncan S. Holmes, Christopher Browning, Lise C. Fechner, Daniel L. Parton, Karen M. L. Morriss
المصدر: Journal of medicinal chemistry. 54(7)
مصطلحات موضوعية: Models, Molecular, Protein Conformation, Administration, Oral, Nasal congestion, Pharmacology, Drug Discovery, medicine, Potency, Humans, Receptors, Histamine H3, Receptors, Histamine H1, Receptor, Administration, Intranasal, Rhinitis, Chemistry, Azelastine, Bioavailability, Blockade, Immunology, Histamine H1 Antagonists, Molecular Medicine, Phthalazines, Nasal administration, medicine.symptom, Antagonism, medicine.drug, Histamine H3 Antagonists
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9
المؤلفون: Michael Shipman, Jérôme Désiré, Paul Martin Gore, Paul J. Dransfield
المصدر: Synlett. 2001:1329-1331
مصطلحات موضوعية: Chemistry, Organic Chemistry, Organic chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::c6ffa09158f964fd292ccfe2a2e81868
https://doi.org/10.1055/s-2001-16039 -
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المؤلفون: Michael Shipman, Paul Martin Gore, Jérôme Désiré, Paul J. Dransfield
المصدر: ChemInform. 32
مصطلحات موضوعية: Chemistry, Stereochemistry, Organic chemistry, General Medicine