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1
المؤلفون: Hartmuth C. Kolb, Stijn Wuyts, Cindy Wintmolders, Leenaerts Joseph Elisabeth, Astrid Bottelbergs, Lieven Declercq, Fengbin Song, Paula te Riele, Chunfang A. Xia, Laura Iturrino, Frederik J. R. Rombouts, José-Ignacio Andrés, Diederik Moechars, Jonas Mariën, Lu Chen, Guy Bormans, Rik Vandenberghe
المصدر: Journal of Medicinal Chemistry. 62:2974-2987
مصطلحات موضوعية: biology, medicine.diagnostic_test, Neurodegeneration, Tau protein, medicine.disease, Biomarker (cell), chemistry.chemical_compound, Nuclear magnetic resonance, chemistry, Positron emission tomography, Drug Discovery, medicine, biology.protein, Molecular Medicine, Structure–activity relationship, Amine gas treating, Cognitive decline, Isoquinoline
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2
المؤلفون: Mark E. Schmidt, Rhys Salter, Cindy Wintmolders, Nigel Austin, Vladimir Chupakhin, Gregor James Macdonald, Astrid Bottelbergs, Paula te Riele, Lu Chen, Katleen Fierens, Diederik Moechars, Andrés A. Trabanco, José-Ignacio Andrés, José Manuel Alonso, Jonas Mariën, Erna Cleiren, Martinez Lamenca Carolina, Frederik J. R. Rombouts, Manuela Ariza, Leenaerts Joseph Elisabeth, Xavier Langlois, Wei Zhang, Alberto Fontana
المصدر: Journal of Medicinal Chemistry. 60:1272-1291
مصطلحات موضوعية: 0301 basic medicine, Tau pathology, tau Proteins, Protein aggregation, Protein Aggregation, Pathological, Mice, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Alzheimer Disease, mental disorders, Drug Discovery, Animals, Humans, Naphthyridines, Pet tracer, Amination, Amyloid beta-Peptides, Chemistry, Quinoline, Brain, Haplorhini, Combinatorial chemistry, First generation, Rats, 030104 developmental biology, Positron-Emission Tomography, Molecular Medicine, Selectivity, 030217 neurology & neurosurgery
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3
المؤلفون: Frederik J R, Rombouts, Lieven, Declercq, José-Ignacio, Andrés, Astrid, Bottelbergs, Lu, Chen, Laura, Iturrino, Joseph E, Leenaerts, Jonas, Mariën, Fengbin, Song, Cindy, Wintmolders, Stijn, Wuyts, Chunfang A, Xia, Paula, Te Riele, Guy, Bormans, Rik, Vandenberghe, Hartmuth, Kolb, Diederik, Moechars
المصدر: Journal of medicinal chemistry. 62(6)
مصطلحات موضوعية: Male, Fluorine Radioisotopes, Pyridines, tau Proteins, Isoquinolines, Macaca mulatta, Rats, Structure-Activity Relationship, Alzheimer Disease, Positron-Emission Tomography, Drug Discovery, Hepatocytes, Animals, Humans, Female, Rats, Wistar, Cells, Cultured
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4
المؤلفون: Jan de Hoon, Guy Bormans, José-Ignacio Andrés, Jesús Alcázar, Paula te Riele, Xavier Langlois, Gil Leurquin-Sterk, Alfons Verbruggen, Mark E. Schmidt, Anne Van Hecken, Sofie Celen, Koen Van Laere, Michel Koole
المصدر: Journal of Nuclear Medicine. 58:110-116
مصطلحات موضوعية: Adult, Male, 0301 basic medicine, Biodistribution, Knockout rat, Metabolic Clearance Rate, Pharmacology, Receptors, Metabotropic Glutamate, Sensitivity and Specificity, Young Adult, 03 medical and health sciences, 0302 clinical medicine, In vivo, Radioligand, Animals, Humans, Tissue Distribution, Radiology, Nuclear Medicine and imaging, Carbon Radioisotopes, Rats, Wistar, Chemistry, Brain, Reproducibility of Results, In vitro, Molecular Imaging, Rats, 030104 developmental biology, Organ Specificity, Isotope Labeling, Positron-Emission Tomography, Radiopharmaceuticals, Metabotropic glutamate receptor 2, Excitatory Amino Acid Antagonists, 030217 neurology & neurosurgery, Ex vivo, Preclinical imaging
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c45e8bc15c80df4046e02dd206ac5bb4
https://doi.org/10.2967/jnumed.116.176628 -
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المؤلفون: Frederik J. R. Rombouts, Lieven Declercq, José-Ignacio Andrés, Astrid Bottelbergs, Lu Chen, Laura Iturrino, Joseph E. Leenaerts, Jonas Mariën, Fengbin Song, Cindy Wintmolders, Stijn Wuyts, Chunfang A. Xia, Paula te Riele, Guy Bormans, Rik Vandenberghe, Hartmuth Kolb, Diederik Moechars
المصدر: Journal of Medicinal Chemistry. 63:1775-1775
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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6
المؤلفون: Xavier Langlois, Nima Davoodi, Paula te Riele
المصدر: European Journal of Pharmacology. 740:669-675
مصطلحات موضوعية: Male, Agonist, Olanzapine, Indoles, Tetrahydronaphthalenes, medicine.drug_class, medicine.medical_treatment, Pharmacology, Benzodiazepines, chemistry.chemical_compound, Piperidines, Dopamine receptor D3, Tetrahydroisoquinolines, Nitriles, medicine, Haloperidol, Animals, Rats, Wistar, Antipsychotic, Clozapine, 7-OH-DPAT, Receptors, Dopamine D2, business.industry, Receptors, Dopamine D3, Antagonist, Radiography, chemistry, Autoradiography, Dopamine Antagonists, Islands of Calleja, business, Proto-Oncogene Proteins c-fos, Antipsychotic Agents, medicine.drug
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7
المؤلفون: Paula te Riele, Gregor James Macdonald, Luc Peeters, Xavier Langlois, Wilhelmus Drinkenburg, Ilse Biesmans, José Ignacio Andrés, A. Ahnaou, Andrés A. Trabanco, Frank Matthias Dautzenberg, John R. Atack, Cindy Wintmolders, Anton Megens, Robert Johannes Lütjens, Hilde Lavreysen, José María Cid, Ilse Van der Linden
المصدر: Journal of Pharmacology and Experimental Therapeutics. 346:514-527
مصطلحات موضوعية: Cyclopropanes, Male, Agonist, Allosteric modulator, Pyridones, medicine.drug_class, Allosteric regulation, Glycine, CHO Cells, Motor Activity, Biology, Pharmacology, Ligands, Receptors, Metabotropic Glutamate, Tritium, Binding, Competitive, Rats, Sprague-Dawley, Mice, Cricetulus, Piperidines, Cricetinae, Excitatory Amino Acid Agonists, medicine, Radioligand, Animals, Humans, Excitatory Amino Acid Agents, Amino Acids, Receptor, Brain Chemistry, Cerebral Cortex, Chinese hamster ovary cell, Cell Membrane, Glutamate receptor, Rats, Metabotropic receptor, Xanthenes, Guanosine 5'-O-(3-Thiotriphosphate), Isotope Labeling, Autoradiography, Molecular Medicine, Calcium, Sleep
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5995a39c7e77c8c46ae8e3eb699d4276
https://doi.org/10.1124/jpet.113.204990 -
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المؤلفون: Miroslav Cik, John R. Atack, Paula te Riele, Marcel Frans Leopold De Bruyn, Ria Wouters, Gregor James Macdonald, Jef Vermeire, Herman M. R. Hendrickx, Anton Megens, Luc Peeters, Hilde Lavreysen, Xavier Langlois
المصدر: Journal of Pharmacology and Experimental Therapeutics. 342:91-105
مصطلحات موضوعية: Male, Olanzapine, Serotonin, Psychosis, Apomorphine, CHO Cells, Pharmacology, Ligands, Rats, Sprague-Dawley, Benzodiazepines, Piperidines, Cricetinae, Dopamine receptor D2, Muscarinic acetylcholine receptor, medicine, Haloperidol, Animals, Humans, Rats, Wistar, Receptor, Cells, Cultured, Catalepsy, Behavior, Animal, Receptors, Dopamine D2, Chemistry, Brain, medicine.disease, Prolactin, Rats, Pyridazines, Dopamine D2 Receptor Antagonists, Rats, Inbred Lew, Schizophrenia, Dopamine Antagonists, Molecular Medicine, Female, Antagonism, Locomotion, Antipsychotic Agents, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d48a38efd535318d7970257f097b7ea8
https://doi.org/10.1124/jpet.111.190702 -
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المؤلفون: Anton Megens, Wilhelmus Drinkenburg, Koen A. Hens, Xavier Langlois, Jef Vermeire, Brian Joel Hrupka, John R. Atack, Paul F. Jackson, Kenneth J. Rhodes, Paula te Riele, Annemie L. Y. Wellens, Abdallah Ahnaou, Nancy Aerts, Patrick De Haes, Brian C. Shook, Herman M. R. Hendrickx, Stefanie Rassnick
المصدر: ACS chemical neuroscience. 5(10)
مصطلحات موضوعية: Male, Receptor, Adenosine A2A, Physiology, Cognitive Neuroscience, Dopamine, CHO Cells, Pharmacology, Adenosine A1 Receptor Antagonists, Motor Activity, Biochemistry, Dopamine agonist, Antiparkinson Agents, Rats, Sprague-Dawley, Adenosine A1 receptor, Mice, Norepinephrine, Cricetulus, Parkinsonian Disorders, Dopamine receptor D2, medicine, Animals, Humans, Rats, Wistar, Neuropharmacology, Dose-Response Relationship, Drug, Chemistry, Receptor, Adenosine A1, Antagonist, Brain, Cell Biology, General Medicine, Adenosine, Recombinant Proteins, Adenosine A2 Receptor Antagonists, Apomorphine, HEK293 Cells, Pyrimidines, Indenes, medicine.drug
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10
المصدر: Neuropharmacology. 40:242-253
مصطلحات موضوعية: Male, Interpeduncular nucleus, medicine.medical_specialty, Guinea Pigs, Substantia nigra, Striatum, Substance P, Biology, Gerbil, Supraoptic nucleus, Radioligand Assay, Cellular and Molecular Neuroscience, Piperidines, Species Specificity, Internal medicine, medicine, Animals, Rats, Wistar, Receptor, Cerebral Cortex, Pharmacology, Membranes, Brain, Receptors, Neurokinin-3, Peptide Fragments, Rats, medicine.anatomical_structure, Endocrinology, nervous system, Hypothalamus, Autoradiography, Zona incerta, Gerbillinae